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Volumn 40, Issue 2, 2013, Pages 289-294

Evaluation of [18F]Nifene biodistribution and dosimetry based on whole-body PET imaging of mice

Author keywords

4 2; 18F Nifene; Biodistribution; Dosimetry; PET; Preclinical

Indexed keywords

NIFENE F 18; TRACER; UNCLASSIFIED DRUG; DIAGNOSTIC AGENT; NIFENE; PYRIDINE DERIVATIVE; PYRROLE DERIVATIVE;

EID: 84872918352     PISSN: 09698051     EISSN: 18729614     Source Type: Journal    
DOI: 10.1016/j.nucmedbio.2012.11.004     Document Type: Article
Times cited : (18)

References (24)
  • 1
    • 79952146830 scopus 로고    scopus 로고
    • Brain imaging of nicotinic receptors in Alzheimer's disease
    • Wu J., Ishikawa M., Zhang J., Hashimoto K. Brain imaging of nicotinic receptors in Alzheimer's disease. Int J Alzheimers Dis 2010, 2010:548913.
    • (2010) Int J Alzheimers Dis , vol.2010 , pp. 548913
    • Wu, J.1    Ishikawa, M.2    Zhang, J.3    Hashimoto, K.4
  • 2
    • 79953765442 scopus 로고    scopus 로고
    • Decreased cerebral alpha4beta2* nicotinic acetylcholine receptor availability in patients with mild cognitive impairment and Alzheimer's disease assessed with positron emission tomography
    • Kendziorra K., Wolf H., Meyer P.M., Barthel H., Hesse S., Becker G.A., et al. Decreased cerebral alpha4beta2* nicotinic acetylcholine receptor availability in patients with mild cognitive impairment and Alzheimer's disease assessed with positron emission tomography. Eur J Nucl Med Mol Imaging 2011, 38:515-525.
    • (2011) Eur J Nucl Med Mol Imaging , vol.38 , pp. 515-525
    • Kendziorra, K.1    Wolf, H.2    Meyer, P.M.3    Barthel, H.4    Hesse, S.5    Becker, G.A.6
  • 3
    • 33847250946 scopus 로고    scopus 로고
    • PET imaging of cortical 11C-nicotine binding correlates with the cognitive function of attention in Alzheimer's disease
    • Kadir A., Almkvist O., Wall A., Langstrom B., Nordberg A. PET imaging of cortical 11C-nicotine binding correlates with the cognitive function of attention in Alzheimer's disease. Psychopharmacology (Berl) 2006, 188:509-520.
    • (2006) Psychopharmacology (Berl) , vol.188 , pp. 509-520
    • Kadir, A.1    Almkvist, O.2    Wall, A.3    Langstrom, B.4    Nordberg, A.5
  • 4
    • 0034576476 scopus 로고    scopus 로고
    • Ligands for in vivo imaging of nicotinic receptor subtypes in Alzheimer brain
    • Sihver W., Langstrom B., Nordberg A. Ligands for in vivo imaging of nicotinic receptor subtypes in Alzheimer brain. Acta Neurol Scand Suppl 2000, 176:27-33.
    • (2000) Acta Neurol Scand Suppl , vol.176 , pp. 27-33
    • Sihver, W.1    Langstrom, B.2    Nordberg, A.3
  • 5
    • 0032857633 scopus 로고    scopus 로고
    • Imaging central nicotinic acetylcholine receptors in baboons with [18F]fluoro-A-85380
    • Valette H., Bottlaender M., Dolle F., Guenther I., Fuseau C., Coulon C., et al. Imaging central nicotinic acetylcholine receptors in baboons with [18F]fluoro-A-85380. J Nucl Med 1999, 40:1374-1380.
    • (1999) J Nucl Med , vol.40 , pp. 1374-1380
    • Valette, H.1    Bottlaender, M.2    Dolle, F.3    Guenther, I.4    Fuseau, C.5    Coulon, C.6
  • 6
    • 32944460294 scopus 로고    scopus 로고
    • Feasibility of 2-deoxy-2-[18F]fluoro-D-glucose- A85380-PET for imaging of human cardiac nicotinic acetylcholine receptors in vivo
    • Bucerius J., Joe A.Y., Schmaljohann J., Gundisch D., Minnerop M., Biersack H.J., et al. Feasibility of 2-deoxy-2-[18F]fluoro-D-glucose- A85380-PET for imaging of human cardiac nicotinic acetylcholine receptors in vivo. Clin Res Cardiol 2006, 95:105-109.
    • (2006) Clin Res Cardiol , vol.95 , pp. 105-109
    • Bucerius, J.1    Joe, A.Y.2    Schmaljohann, J.3    Gundisch, D.4    Minnerop, M.5    Biersack, H.J.6
  • 7
    • 84856388179 scopus 로고    scopus 로고
    • Positron emission tomography experience with 2-[(1)F]fluoro-3-(2(S)-azetidinylmethoxy)pyridine (2-[(1)F]FA) in the living human brain of smokers with paranoid schizophrenia
    • Brasic J.R., Cascella N., Kumar A., Zhou Y., Hilton J., Raymont V., et al. Positron emission tomography experience with 2-[(1)F]fluoro-3-(2(S)-azetidinylmethoxy)pyridine (2-[(1)F]FA) in the living human brain of smokers with paranoid schizophrenia. Synapse 2012, 66:352-368.
    • (2012) Synapse , vol.66 , pp. 352-368
    • Brasic, J.R.1    Cascella, N.2    Kumar, A.3    Zhou, Y.4    Hilton, J.5    Raymont, V.6
  • 8
    • 62749191187 scopus 로고    scopus 로고
    • Baseline expression of alpha4beta2* nicotinic acetylcholine receptors predicts motivation to self-administer nicotine
    • Le Foll B., Chefer S.I., Kimes A.S., Shumway D., Stein E.A., Mukhin A.G., et al. Baseline expression of alpha4beta2* nicotinic acetylcholine receptors predicts motivation to self-administer nicotine. Biol Psychiatry 2009, 65:714-716.
    • (2009) Biol Psychiatry , vol.65 , pp. 714-716
    • Le Foll, B.1    Chefer, S.I.2    Kimes, A.S.3    Shumway, D.4    Stein, E.A.5    Mukhin, A.G.6
  • 9
    • 53749101043 scopus 로고    scopus 로고
    • Greater nicotinic acetylcholine receptor density in smokers than in nonsmokers: a PET study with 2-18F-FA-85380
    • Mukhin A.G., Kimes A.S., Chefer S.I., Matochik J.A., Contoreggi C.S., Horti A.G., et al. Greater nicotinic acetylcholine receptor density in smokers than in nonsmokers: a PET study with 2-18F-FA-85380. J Nucl Med 2008, 49:1628-1635.
    • (2008) J Nucl Med , vol.49 , pp. 1628-1635
    • Mukhin, A.G.1    Kimes, A.S.2    Chefer, S.I.3    Matochik, J.A.4    Contoreggi, C.S.5    Horti, A.G.6
  • 10
    • 53949092571 scopus 로고    scopus 로고
    • Nicotinic acetylcholine receptors and modulation of learning in 4- and 27-month-old rabbits
    • Li J.G., Lehr M., Liu-Chen L.Y., Woodruff-Pak D.S. Nicotinic acetylcholine receptors and modulation of learning in 4- and 27-month-old rabbits. Neuropsychopharmacology 2008, 33:2820-2830.
    • (2008) Neuropsychopharmacology , vol.33 , pp. 2820-2830
    • Li, J.G.1    Lehr, M.2    Liu-Chen, L.Y.3    Woodruff-Pak, D.S.4
  • 11
    • 84857685884 scopus 로고    scopus 로고
    • Nicotinic acetylcholine receptors in rat forebrain that bind (18) F-nifene: relating PET imaging, autoradiography, and behavior
    • Bieszczad K.M., Kant R., Constantinescu C.C., Pandey S.K., Kawai H.D., Metherate R., et al. Nicotinic acetylcholine receptors in rat forebrain that bind (18) F-nifene: relating PET imaging, autoradiography, and behavior. Synapse 2012, 66:418-434.
    • (2012) Synapse , vol.66 , pp. 418-434
    • Bieszczad, K.M.1    Kant, R.2    Constantinescu, C.C.3    Pandey, S.K.4    Kawai, H.D.5    Metherate, R.6
  • 13
    • 33846808976 scopus 로고    scopus 로고
    • Quantification of alpha4beta2* nicotinic receptors in the rat brain with microPET and 2-[18F]F-A-85380
    • Vaupel D.B., Stein E.A., Mukhin A.G. Quantification of alpha4beta2* nicotinic receptors in the rat brain with microPET and 2-[18F]F-A-85380. Neuroimage 2007, 34:1352-1362.
    • (2007) Neuroimage , vol.34 , pp. 1352-1362
    • Vaupel, D.B.1    Stein, E.A.2    Mukhin, A.G.3
  • 14
    • 33646046816 scopus 로고    scopus 로고
    • Nicotinic alpha4beta2 receptor imaging agents: part II. Synthesis and biological evaluation of 2-[18F]fluoro-3-[2-((S)-3-pyrrolinyl)methoxy]pyridine (18F-nifene) in rodents and imaging by PET in nonhuman primate
    • Pichika R., Easwaramoorthy B., Collins D., Christian B.T., Shi B., Narayanan T.K., et al. Nicotinic alpha4beta2 receptor imaging agents: part II. Synthesis and biological evaluation of 2-[18F]fluoro-3-[2-((S)-3-pyrrolinyl)methoxy]pyridine (18F-nifene) in rodents and imaging by PET in nonhuman primate. Nucl Med Biol 2006, 33:295-304.
    • (2006) Nucl Med Biol , vol.33 , pp. 295-304
    • Pichika, R.1    Easwaramoorthy, B.2    Collins, D.3    Christian, B.T.4    Shi, B.5    Narayanan, T.K.6
  • 15
    • 80053908606 scopus 로고    scopus 로고
    • Specific alpha4beta2 nicotinic acetylcholine receptor binding of [F-18]nifene in the rhesus monkey
    • Hillmer A.T., Wooten D.W., Moirano J.M., Slesarev M., Barnhart T.E., Engle J.W., et al. Specific alpha4beta2 nicotinic acetylcholine receptor binding of [F-18]nifene in the rhesus monkey. Synapse 2011, 65:1309-1318.
    • (2011) Synapse , vol.65 , pp. 1309-1318
    • Hillmer, A.T.1    Wooten, D.W.2    Moirano, J.M.3    Slesarev, M.4    Barnhart, T.E.5    Engle, J.W.6
  • 16
    • 84874418635 scopus 로고    scopus 로고
    • Evaluation of F-nifene binding to alpha4beta2 nicotinic receptors in the rat brain using microPET imaging
    • Kant R., Constantinescu C.C., Parekh P., Pandey S.K., Pan M.L., Easwaramoorthy B., et al. Evaluation of F-nifene binding to alpha4beta2 nicotinic receptors in the rat brain using microPET imaging. EJNMMI Res 2011, 1:6.
    • (2011) EJNMMI Res , vol.1 , pp. 6
    • Kant, R.1    Constantinescu, C.C.2    Parekh, P.3    Pandey, S.K.4    Pan, M.L.5    Easwaramoorthy, B.6
  • 17
    • 77950361630 scopus 로고    scopus 로고
    • RADAR realistic animal model series for dose assessment
    • Keenan M.A., Stabin M.G., Segars W.P., Fernald M.J. RADAR realistic animal model series for dose assessment. J Nucl Med 2010, 51:471-476.
    • (2010) J Nucl Med , vol.51 , pp. 471-476
    • Keenan, M.A.1    Stabin, M.G.2    Segars, W.P.3    Fernald, M.J.4
  • 18
    • 79960324659 scopus 로고    scopus 로고
    • RADAR commentary: evolution and current status of dosimetry in nuclear medicine
    • Stabin M.G., Sharkey R.M., Siegel J.A. RADAR commentary: evolution and current status of dosimetry in nuclear medicine. J Nucl Med 2011, 52:1156-1161.
    • (2011) J Nucl Med , vol.52 , pp. 1156-1161
    • Stabin, M.G.1    Sharkey, R.M.2    Siegel, J.A.3
  • 19
    • 0001372627 scopus 로고
    • Radiation-dosimetry of i-131-19-iodocholesterol - pitfalls of using tissue concentration data - reply
    • Kirschner A.S., Ice R.D., Beierwaltes W.H. Radiation-dosimetry of i-131-19-iodocholesterol - pitfalls of using tissue concentration data - reply. J Nucl Med 1975, 16:248-249.
    • (1975) J Nucl Med , vol.16 , pp. 248-249
    • Kirschner, A.S.1    Ice, R.D.2    Beierwaltes, W.H.3
  • 20
    • 67249130006 scopus 로고    scopus 로고
    • In vivo 3D digital atlas database of the adult C57BL/6J mouse brain by Magnetic resonance microscopy
    • Ma Y., Smith D., Hof P.R., Foerster B., Hamilton S., Blackband S.J., et al. In vivo 3D digital atlas database of the adult C57BL/6J mouse brain by Magnetic resonance microscopy. Front Neuroanat 2008, 2:1.
    • (2008) Front Neuroanat , vol.2 , pp. 1
    • Ma, Y.1    Smith, D.2    Hof, P.R.3    Foerster, B.4    Hamilton, S.5    Blackband, S.J.6
  • 21
    • 0038654355 scopus 로고    scopus 로고
    • Biodistribution and radiation dosimetry of 18F-fluoro-A-85380 in healthy volunteers
    • Bottlaender M., Valette H., Roumenov D., Dolle F., Coulon C., Ottaviani M., et al. Biodistribution and radiation dosimetry of 18F-fluoro-A-85380 in healthy volunteers. J Nucl Med 2003, 44:596-601.
    • (2003) J Nucl Med , vol.44 , pp. 596-601
    • Bottlaender, M.1    Valette, H.2    Roumenov, D.3    Dolle, F.4    Coulon, C.5    Ottaviani, M.6
  • 22
    • 84862613906 scopus 로고    scopus 로고
    • Radiation dosimetry of the translocator protein ligands [18F]PBR111 and [18F]PBR102
    • Verschuer J.D., Towson J., Eberl S., Katsifis A., Henderson D., Lam P., et al. Radiation dosimetry of the translocator protein ligands [18F]PBR111 and [18F]PBR102. Nucl Med Biol 2012, 39:742-753.
    • (2012) Nucl Med Biol , vol.39 , pp. 742-753
    • Verschuer, J.D.1    Towson, J.2    Eberl, S.3    Katsifis, A.4    Henderson, D.5    Lam, P.6
  • 23
    • 84878472932 scopus 로고    scopus 로고
    • Evaluation of [18F]Mefway biodistribution and dosimetry based on whole-body PET imaging of mice
    • [Epub ahead of print].
    • Constantinescu C.C., Sevrioukov E., Garcia A., Pan M.-L., Mukherjee J. Evaluation of [18F]Mefway biodistribution and dosimetry based on whole-body PET imaging of mice. Mol Imaging Biol 2012, [Epub ahead of print].
    • (2012) Mol Imaging Biol
    • Constantinescu, C.C.1    Sevrioukov, E.2    Garcia, A.3    Pan, M.-L.4    Mukherjee, J.5
  • 24
    • 84872939155 scopus 로고    scopus 로고
    • Food and Drug Administration
    • National Archives and Records Administration, Office of the Federal Register, Washington DC
    • Food and Drug Administration Title 21 CFR 361.1 Radioactive Drugs for Certain Research Uses 2011, 325-330. National Archives and Records Administration, Office of the Federal Register, Washington DC.
    • (2011) Title 21 CFR 361.1 Radioactive Drugs for Certain Research Uses , pp. 325-330


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