Effect of amorphization method on telmisartan solubility and the tableting process

European Journal of Pharmaceutics and Biopharmaceutics

Volumn 83, Issue 1, 2013, Pages 114-121

  Lepek, P ^a   Sawicki, W ^a   Wlodarski, K ^a   Wojnarowska, Z ^b   Paluch, M ^b   Guzik, L ^a  

^a MEDICAL UNIVERSITY OF GDANSK   (Poland)

^b UNIVERSITY OF SILESIA   (Poland)

Author keywords

Amorphous telmisartan; Cryogenic grinding; Glassy state; Melt quench technique; Vitrification

Indexed keywords

TELMISARTAN;

ARTICLE; DIFFERENTIAL SCANNING CALORIMETRY; DRUG SOLUBILITY; DRUG STABILITY; DRUG SYNTHESIS; GLASS TRANSITION TEMPERATURE; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; PHYSICAL CHEMISTRY; TABLET FORMULATION; VITRIFICATION; X RAY POWDER DIFFRACTION;

ANGIOTENSIN II TYPE 1 RECEPTOR BLOCKERS; BENZIMIDAZOLES; BENZOATES; CALORIMETRY, DIFFERENTIAL SCANNING; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; CRYSTALLIZATION; DRUG STABILITY; DRUG STORAGE; SOLUBILITY; TABLETS; TEMPERATURE; TIME FACTORS; X-RAY DIFFRACTION;

EID: 84871919738     PISSN: 09396411     EISSN: 18733441     Source Type: Journal    
DOI: 10.1016/j.ejpb.2012.09.019     Document Type: Article

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