메뉴 건너뛰기




Volumn 37, Issue 3, 2012, Pages 225-231

Transepithelial transport of rosuvastatin and effect of ursolic acid on its transport in Caco-2 monolayers

Author keywords

Caco 2 cell monolayers; Rosuvastatin; Ursolic acid

Indexed keywords

1,2,3,4,6,7,12,12A OCTAHYDRO 6 ISOBUTYL 9 METHOXY 1,4 DIOXOPYRAZINO[1',2':1,6]PYRIDO[3,4 B]INDOLE 3 PROPANOIC ACID TERT BUTYL ESTER; BREAST CANCER RESISTANCE PROTEIN; MULTIDRUG RESISTANCE PROTEIN; MULTIDRUG RESISTANCE PROTEIN 2; ROSUVASTATIN; TALINOLOL; URSOLIC ACID;

EID: 84871335784     PISSN: 03787966     EISSN: 21070180     Source Type: Journal    
DOI: 10.1007/s13318-012-0094-9     Document Type: Article
Times cited : (14)

References (19)
  • 1
    • 0035286778 scopus 로고    scopus 로고
    • Caco-2 monolayers inexperimental and theoretical predictions of drug transport
    • Artursson P, Palm K, Luthman K (2001) Caco-2 monolayers inexperimental and theoretical predictions of drug transport. Adv Drug Deliv Rev 46:27-43
    • (2001) Adv Drug Deliv Rev , vol.46 , pp. 27-43
    • Artursson, P.1    Palm, K.2    Luthman, K.3
  • 2
    • 1242296077 scopus 로고    scopus 로고
    • Optimizing the pharmacology of statins: Characteristics of rosuvastatin
    • discussion 36-37
    • Chapman MJ, Taggart FM (2002) Optimizing the pharmacology of statins: characteristics of rosuvastatin. Atheroscler Suppl 2:33-36 discussion 36-37
    • (2002) Atheroscler , Issue.SUPPL. 2 , pp. 33-36
    • Chapman, M.J.1    Taggart, F.M.2
  • 3
    • 77953403463 scopus 로고    scopus 로고
    • Development of a cell-based high-throughput assay to screen for inhibitors of organic anion transporting polypeptides 1B1 and 1B3
    • Chunshan G, Amanda O, Rathnam C, Bruno H (2010) Development of a cell-based high-throughput assay to screen for inhibitors of organic anion transporting polypeptides 1B1 and 1B3. Curr Chem Genomics 4:1-8
    • (2010) Curr Chem Genomics , vol.4 , pp. 1-8
    • Chunshan, G.1    Amanda, O.2    Rathnam, C.3    Bruno, H.4
  • 5
    • 84871340288 scopus 로고    scopus 로고
    • Inhibition of the function of p-glycoprotein by ursolic acid
    • Huayi R (2009) Inhibition of the function of p-glycoprotein by ursolic acid. Central South Pharm 7(7):493-496
    • (2009) Central South Pharm , vol.7 , Issue.7 , pp. 493-496
    • Huayi, R.1
  • 6
    • 16344366327 scopus 로고    scopus 로고
    • Food-drug interaction between ferulic acid and nateglinide involving the fluorescein/H? cotransport system
    • Itagaki S, Kobayashi Y, Otsuka Y, Kubo S, Kobayashi M, Hirano T, Iseki K (2005) Food-drug interaction between ferulic acid and nateglinide involving the fluorescein/H? cotransport system. J Agric Food Chem 53:2499-2502
    • (2005) J Agric Food Chem , vol.53 , pp. 2499-2502
    • Itagaki, S.1    Kobayashi, Y.2    Otsuka, Y.3    Kubo, S.4    Kobayashi, M.5    Hirano, T.6    Iseki, K.7
  • 7
    • 79959434557 scopus 로고    scopus 로고
    • Use of transporter knockdown Caco-2 cells to investigate the in vitro efflux of statin drugs
    • Li J, Volpe DA, Wang Y, Zhang W, Bode C, Owen A, Hidalgo IJ (2011) Use of transporter knockdown Caco-2 cells to investigate the in vitro efflux of statin drugs. Drug Metab Dispos 39(7):1196-1202
    • (2011) Drug Metab Dispos , vol.39 , Issue.7 , pp. 1196-1202
    • Li, J.1    Volpe, D.A.2    Wang, Y.3    Zhang, W.4    Bode, C.5    Owen, A.6    Hidalgo, I.J.7
  • 8
    • 33645829284 scopus 로고    scopus 로고
    • ATP-dependent transport of rosuvastatin in membrane vesicles expressing breast cancer resistance protein
    • Liyue Hu, Yi W, Scott G (2006) ATP-dependent transport of rosuvastatin in membrane vesicles expressing breast cancer resistance protein. Drug Metab Dispos 34:738-742
    • (2006) Drug Metab Dispos , vol.34 , pp. 738-742
    • Liyue, Hu.1    Yi, W.2    Scott, G.3
  • 9
    • 0242509092 scopus 로고    scopus 로고
    • Absolute oral bioavailability of rosuvastatin in healthy white adult male volunteers
    • Martin PD, Warwick MJ, Dane AL, Brindley C, Short T (2003a) Absolute oral bioavailability of rosuvastatin in healthy white adult male volunteers. Clin Ther 25:2553-2563
    • (2003) Clin Ther , vol.25 , pp. 2553-2563
    • Martin, P.D.1    Warwick, M.J.2    Dane, A.L.3    Brindley, C.4    Short, T.5
  • 11
    • 7444272089 scopus 로고    scopus 로고
    • Transepithelial permeation of tolbutamide across the human intestinal cell line, Caco-2
    • Nobuhiro N, Kohji N, Tomochika U, Hidenari H, Kikuo I (2004) Transepithelial permeation of tolbutamide across the human intestinal cell line, Caco-2. DrugMetab Pharmacokin 19(1):48-54
    • (2004) DrugMetab Pharmacokin , vol.19 , Issue.1 , pp. 48-54
    • Nobuhiro, N.1    Kohji, N.2    Tomochika, U.3    Hidenari, H.4    Kikuo, I.5
  • 12
    • 84992920491 scopus 로고    scopus 로고
    • Rosuvastatin demonstrates greater reduction of low-density lipoprotein cholesterol compared with pravastatin and simvastatin in hypercholesterolaemic patients: A randomized, double blind study
    • Paoletti R, Fahmy M, Mahla G, Mizan J, Southworth H (2001) Rosuvastatin demonstrates greater reduction of low-density lipoprotein cholesterol compared with pravastatin and simvastatin in hypercholesterolaemic patients: a randomized, double blind study. J Cardiovasc Risk 8:383-890
    • (2001) J Cardiovasc Risk , vol.8 , pp. 383-890
    • Paoletti, R.1    Fahmy, M.2    Mahla, G.3    Mizan, J.4    Southworth, H.5
  • 13
    • 52949104006 scopus 로고    scopus 로고
    • Involvement of multiple transporters in the hepatobiliary transport of rosuvastatin
    • Satoshi K, Kazuya M, Yi W, Yuichi S (2008) Involvement of multiple transporters in the hepatobiliary transport of rosuvastatin. Drug Metab Dispos 36(10):2014-2023
    • (2008) Drug Metab Dispos , vol.36 , Issue.10 , pp. 2014-2023
    • Satoshi, K.1    Kazuya, M.2    Yi, W.3    Yuichi, S.4
  • 14
    • 84856237147 scopus 로고    scopus 로고
    • The effect of herbal medicine danshensu and ursolic acid on pharmacokinetics of rosuvastatin in rats
    • Wen JH, Xiong YQ (2011) The effect of herbal medicine danshensu and ursolic acid on pharmacokinetics of rosuvastatin in rats. Eur J Drug Metab Pharmacokinet 36:205-211
    • (2011) Eur J Drug Metab Pharmacokinet , vol.36 , pp. 205-211
    • Wen, J.H.1    Xiong, Y.Q.2
  • 17
    • 78651252487 scopus 로고    scopus 로고
    • Quantitation of ursolic acid in human plasma by ultra performance liquid chromatography tandem mass spectrometry and its pharmacokinetic study
    • 879
    • Xia Y, Wei G, Si D, Liu C (2011) Quantitation of ursolic acid in human plasma by ultra performance liquid chromatography tandem mass spectrometry and its pharmacokinetic study. J Chromatogr B Analyt Technol Biomed Life Sci 15 879(2):219-224
    • (2011) J Chromatogr B Analyt Technol Biomed Life Sci , vol.15 , Issue.2 , pp. 219-224
    • Xia, Y.1    Wei, G.2    Si, D.3    Liu, C.4
  • 18
    • 84860394704 scopus 로고    scopus 로고
    • Transport characteristics of tryptanthrin and its inhibitory effect on P-gp and MRP2 in Caco-2 cells
    • Xingang Z, Xuelian Z, Guo M, Junkai Y, Honghai W, Qing Y (2011) Transport characteristics of tryptanthrin and its inhibitory effect on P-gp and MRP2 in Caco-2 cells. J Pharm Pharmaceut Sci 14(3):325-335. http://www.cspsCanada.org
    • (2011) J Pharm Pharmaceut Sci , vol.14 , Issue.3 , pp. 325-335
    • Xingang, Z.1    Xuelian, Z.2    Guo, M.3    Junkai, Y.4    Honghai, W.5    Qing, Y.6


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.