Linear trifluoroethylamine RGD peptidomimetics: Stereoselective synthesis and integrin αvβ3 affinity

Synlett

Volumn 23, Issue 20, 2012, Pages 2899-2902

  Piras, Monica ^a   Fleming, Ian N ^a   Harrison, William T A ^a   Zanda, Matteo ^a  

^a UNIVERSITY OF ABERDEEN   (United Kingdom)

Author keywords

integrins; peptidomimetics; RGD; trifluoroethylamine

Indexed keywords

ARGINYLGLYCYLASPARTIC ACID; ETHYLAMINE; HYDROGEN; PEPTIDOMIMETIC AGENT; TRIFLUOROETHYLAMINE; UNCLASSIFIED DRUG; VITRONECTIN RECEPTOR;

ARTICLE; BINDING AFFINITY; CHEMICAL ANALYSIS; CHEMICAL BOND; CHEMICAL STRUCTURE; DIASTEREOISOMER; PROTEIN INTERACTION; STEREOCHEMISTRY; SYNTHESIS;

EID: 84869479583     PISSN: 09365214     EISSN: 14372096     Source Type: Journal    
DOI: 10.1055/s-0032-1317557     Document Type: Article

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