Synthesis and characterization of some new quinoline based derivatives endowed with broad spectrum antimicrobial potency

Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 22, 2012, Pages 6871-6875

  Desai, Nisheeth C ^a   Rajpara, Kiran M ^a   Joshi, Vivek V ^a  

^a BHAVNAGAR UNIVERSITY   (India)

Author keywords

Antimicrobial activity; Morpholine; Pyrazoline; Pyrimidine; Quinoline; Thiazolidinone; Vilsmeier Haack reaction

Indexed keywords

2 (5 (2 CHLORO 6 FLUOROQUINOLIN 3 YL) 3 (ARYL) 4,5 DIHYDRO 1H PYRAZOL 1 YL)THIAZOL 4(5H) ONE DERIVATIVE; ANTIINFECTIVE AGENT; N (4 (2 CHLORO 6 FLUOROQUINOLIN 3 YL) 6 (ARYL)PYRIMIDIN 2 YL) 2 MORPHOLINOACETAMIDE DERIVATIVE; QUINOLONE DERIVATIVE; UNCLASSIFIED DRUG;

ANTIMICROBIAL ACTIVITY; ARTICLE; ASPERGILLUS CLAVATUS; ASPERGILLUS NIGER; BROTH DILUTION; CANDIDA ALBICANS; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; NONHUMAN; PSEUDOMONAS AERUGINOSA; STAPHYLOCOCCUS AUREUS; STREPTOCOCCUS PYOGENES;

ANTI-INFECTIVE AGENTS; FUNGI; GRAM-NEGATIVE BACTERIA; GRAM-POSITIVE BACTERIA; MAGNETIC RESONANCE SPECTROSCOPY; MASS SPECTROMETRY; MICROBIAL SENSITIVITY TESTS; MOLECULAR CONFORMATION; QUINOLINES; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLES;

ASPERGILLUS CLAVATUS; ASPERGILLUS NIGER; CANDIDA ALBICANS; ESCHERICHIA COLI; PSEUDOMONAS AERUGINOSA; STAPHYLOCOCCUS AUREUS; STREPTOCOCCUS PYOGENES;

EID: 84867848258     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2012.09.039     Document Type: Article

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