Synthesis and anti-HIV activity of alkylated quinoline 2,4-diols

Bioorganic and Medicinal Chemistry

Volumn 18, Issue 8, 2010, Pages 2872-2879

  Ahmed, Nafees ^a   Brahmbhatt, Keyur G ^a   Sabde, Sudeep ^b   Mitra, Debashis ^b   Singh, Inder Pal ^a   Bhutani, Kamlesh K ^a  

^a NATIONAL INSTITUTE OF PHARMACEUTICAL EDUCATION AND RESEARCH NIPER   (India)

^b NATIONAL CENTRE FOR CELL SCIENCE   (India)

Author keywords

Alkylation; Anti HIV activity; CEM GFP cells; Quinoline 2,4 diol

Indexed keywords

3 (3 METHYLBUT 2 ENYL) 4 (3 METHYLBUT 2 ENYLOXY)QUINOLIN 2 OL; 3 (4 METHYLPENT 3 ENYL) 4 (4 METHYLPENT 3 ENYLOXY)QUINOLIN 2 OL; 3 (PROP 2 YNYL) 4 (PROP 2 YNYLOXY)QUINOLIN 2 OL; 4 (ISOPENTYLOXY)QUINOLIN 2 OL; 4 (PROP 2 YNYLOXY)QUINOLIN 2 OL; ALKALOID; BUCHAPINE; QUINOLONE DERIVATIVE; UNCLASSIFIED DRUG;

ALKYLATION; ANTIVIRAL ACTIVITY; ARTICLE; CD4+ T LYMPHOCYTE; CONTROLLED STUDY; DRUG CYTOTOXICITY; DRUG STRUCTURE; DRUG SYNTHESIS; HUMAN; HUMAN CELL; HUMAN IMMUNODEFICIENCY VIRUS; HUMAN IMMUNODEFICIENCY VIRUS 1; IC 50;

ALKYLATION; ANTI-HIV AGENTS; CD4-POSITIVE T-LYMPHOCYTES; ENZYME-LINKED IMMUNOSORBENT ASSAY; HUMANS; QUINOLINES; STRUCTURE-ACTIVITY RELATIONSHIP;

HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 77950629689     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2010.03.015     Document Type: Article

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