Kinetic properties and small-molecule inhibition of human myosin-6

FEBS Letters

Volumn 586, Issue 19, 2012, Pages 3208-3214

  Heissler, Sarah M ^a   Selvadurai, Jayashankar ^a   Bond, Lisa M ^b   Fedorov, Roman ^a   Kendrick Jones, John ^c   Buss, Folma ^b   Manstein, Dietmar J ^a  

^a HANNOVER MEDICAL SCHOOL   (Germany)

^b UNIVERSITY OF CAMBRIDGE   (United Kingdom)

^c MRC LABORATORY OF MOLECULAR BIOLOGY   (United Kingdom)

Author keywords

Actin myosin; Allostery; Inhibition; Kinetics

Indexed keywords

2,4,6 TRIIODOPHENOL; F ACTIN; MYOSIN VI; NUCLEOTIDE; PHENOL DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CELL FUSION; CELL MEMBRANE; CELL SECRETION; CONTROLLED STUDY; HUMAN; HUMAN CELL; KINETICS; PRIORITY JOURNAL; PROTEIN DOMAIN; PROTEIN FUNCTION; PROTEIN PROTEIN INTERACTION;

ACTINS; AMINO-ACID N-ACETYLTRANSFERASE; ANIMALS; GENE KNOCKDOWN TECHNIQUES; HELA CELLS; HUMANS; KINETICS; MODELS, BIOLOGICAL; MODELS, MOLECULAR; MOLECULAR MOTOR PROTEINS; MUTAGENESIS, SITE-DIRECTED; MYOSIN HEAVY CHAINS; PHENOLS; PROTEIN INTERACTION DOMAINS AND MOTIFS; RABBITS; RECOMBINANT FUSION PROTEINS; RNA, SMALL INTERFERING;

EID: 84866614795     PISSN: 00145793     EISSN: 18733468     Source Type: Journal    
DOI: 10.1016/j.febslet.2012.07.014     Document Type: Article

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