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Volumn 20, Issue 19, 2012, Pages 5980-5985

Synthesis and comparison of antiplasmodial activity of (+), (-) and racemic 7-chloro-4-(N-lupinyl)aminoquinoline

(8) Rusconi, Chiara a Vaiana, Nadia a Casagrande, Manolo a Basilico, Nicoletta a Parapini, Silvia a Taramelli, Donatella a Romeo, Sergio a Sparatore, Anna a

a UNIVERSITY OF MILAN (Italy)

Author keywords

Enzymatic resolution; Lipase; Lupinine; Malaria; Quinoline

Indexed keywords

7 CHLORO 4 (N LUPINYL)AMINOQUINOLINE; 7 CHLORO 4 [N [(OCTAHYDRO 2H QUINOLIZIN 1 YL)METHYL]AMINO]QUINOLINE; ANTIMALARIAL AGENT; CHLOROQUINE; LUPININE; TRIACYLGLYCEROL LIPASE; UNCLASSIFIED DRUG;

ANTIMALARIAL ACTIVITY; ARTICLE; CATALYSIS; CONTROLLED STUDY; CYTOTOXICITY; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME KINETICS; HUMAN; HUMAN CELL; IC 50; IN VITRO STUDY; NONHUMAN; PHARMACOLOGICAL PARAMETERS; PLASMODIUM FALCIPARUM; RACEMIC MIXTURE; THERAPEUTIC INDEX;

AMINOQUINOLINES; ANTIMALARIALS; CELL LINE; CELL SURVIVAL; HUMANS; INHIBITORY CONCENTRATION 50; LUPINUS; PLASMODIUM FALCIPARUM; SPARTEINE; STEREOISOMERISM;

LUPINUS LUTEUS; PLASMODIUM FALCIPARUM;

EID: 84866395906 PISSN: 09680896 EISSN: 14643391 Source Type: Journal
DOI: 10.1016/j.bmc.2012.07.041 Document Type: Article

Times cited : (12)

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