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Volumn 20, Issue 2, 2012, Pages

Developing an efficacious diclofenac diethylamine transdermal formulation

Author keywords

Diclofenac diethylamine; Lotion; Oleic acid; Percutaneous absorption; Transdermal

Indexed keywords

DICLOFENAC DIETHYLAMINE; OLEIC ACID; SILICON; TURPENTINE OIL;

EID: 84866113739     PISSN: 10219498     EISSN: None     Source Type: Journal    
DOI: 10.6227/jfda.2012200205     Document Type: Article
Times cited : (20)

References (31)
  • 1
    • 77953592687 scopus 로고    scopus 로고
    • Diclofenac: An update on its mechanism of action and safety profile
    • Gan, T. J. 2010. Diclofenac: an update on its mechanism of action and safety profile. Curr. Med. Res. Opin. 26: 1715-1731.
    • (2010) Curr. Med. Res. Opin. , vol.26 , pp. 1715-1731
    • Gan, T.J.1
  • 3
    • 79953899392 scopus 로고    scopus 로고
    • Development and characterization of sodium alginate-hydroxypropyl methylcellulose-polyester multilayered hydrogel membranes for drug delivery through skin
    • Kulkarni, R. V., Wagh, Y. J., Setty, C. M. and Sa, B. 2011. Development and characterization of sodium alginate-hydroxypropyl methylcellulose-polyester multilayered hydrogel membranes for drug delivery through skin. Polymer-Plastics Technol. Engin. 50: 490-497.
    • (2011) Polymer-Plastics Technol. Engin. , vol.50 , pp. 490-497
    • Kulkarni, R.V.1    Wagh, Y.J.2    Setty, C.M.3    Sa, B.4
  • 4
    • 34247480143 scopus 로고    scopus 로고
    • Ex vivo study of transdermal permeation of four diclofenac salts from different vehicles
    • Minghetti, P., Cilurzo, F., Casiraghi, A., Montanari, L. and Fini, A. 2007. Ex vivo study of transdermal permeation of four diclofenac salts from different vehicles. J. Pharm. Sci. 96: 814-823.
    • (2007) J. Pharm. Sci. , vol.96 , pp. 814-823
    • Minghetti, P.1    Cilurzo, F.2    Casiraghi, A.3    Montanari, L.4    Fini, A.5
  • 5
    • 0036771415 scopus 로고    scopus 로고
    • Design, development, physicochemical, and in vitro and in vivo evaluation of transdermal patches containing diclofenac diethylammonium salt
    • Arora, P. and Mukherjee, B. 2002. Design, development, physicochemical, and In vitro and In vivo evaluation of transdermal patches containing diclofenac diethylammonium salt. J. Pharm. Sci. 91: 2089-2096.
    • (2002) J. Pharm. Sci. , vol.91 , pp. 2089-2096
    • Arora, P.1    Mukherjee, B.2
  • 6
    • 5444241167 scopus 로고    scopus 로고
    • Emerging technologies in transdermal therapeutics
    • Meidan, V. M. and Michniak, B. B. 2004. Emerging technologies in transdermal therapeutics. Am. J. Ther. 11: 312-316.
    • (2004) Am. J. Ther. , vol.11 , pp. 312-316
    • Meidan, V.M.1    Michniak, B.B.2
  • 7
    • 1142297663 scopus 로고    scopus 로고
    • Characterization of caprylocaproyl macrogolglycerides based microemulsion drug delivery vehicles for an amphiphilic drug
    • Djordjevic, L., Primorac, M., Stupar, M. and Krajisnik, D. 2004. Characterization of caprylocaproyl macrogolglycerides based microemulsion drug delivery vehicles for an amphiphilic drug. Int. J. Pharm. 271: 9-11.
    • (2004) Int. J. Pharm. , vol.271 , pp. 9-11
    • Djordjevic, L.1    Primorac, M.2    Stupar, M.3    Krajisnik, D.4
  • 8
    • 7044269444 scopus 로고    scopus 로고
    • Transdermal delivery of diclofenac using microemulsions
    • Kweon, J. H., Chi, S. C. and Park, E. S. 2004. Transdermal delivery of diclofenac using microemulsions. Arch. Pharm. Res. 27: 351-356.
    • (2004) Arch. Pharm. Res. , vol.27 , pp. 351-356
    • Kweon, J.H.1    Chi, S.C.2    Park, E.S.3
  • 9
    • 34247475216 scopus 로고    scopus 로고
    • The physicochemical characterization and in vitro/In vivo evaluation of natural surfactants-based emulsions as vehicles for diclofenac diethylamine
    • Vucinić-Milanković, N., Savić, S., Vuleta, G. and Vucinić, S. 2007. The physicochemical characterization and In vitro/In vivo evaluation of natural surfactants-based emulsions as vehicles for diclofenac diethylamine. Drug Dev. Ind. Pharm. 33: 221-234.
    • (2007) Drug Dev. Ind. Pharm. , vol.33 , pp. 221-234
    • Vucinić-Milanković, N.1    Savić, S.2    Vuleta, G.3    Vucinić, S.4
  • 10
    • 47249114766 scopus 로고    scopus 로고
    • Anti-inflammatory activity of gel containing novel elastic niosomes entrapped with diclofenac diethylammonium
    • Manosroi, A., Jantrawut, P. and Manosroi, J. 2008. Anti-inflammatory activity of gel containing novel elastic niosomes entrapped with diclofenac diethylammonium. Int. J. Pharm. 360: 156-163.
    • (2008) Int. J. Pharm. , vol.360 , pp. 156-163
    • Manosroi, A.1    Jantrawut, P.2    Manosroi, J.3
  • 11
    • 0034028222 scopus 로고    scopus 로고
    • Aqueous solubility of diclofenac diethylamine in the presence of pharmaceutical additives: A comparative study with diclofenac sodium
    • Khalil, E., Najjar, S. and Sallam, A. 2000. Aqueous solubility of diclofenac diethylamine in the presence of pharmaceutical additives: a comparative study with diclofenac sodium. Drug Dev. Ind. Pharm. 26: 375-381.
    • (2000) Drug Dev. Ind. Pharm. , vol.26 , pp. 375-381
    • Khalil, E.1    Najjar, S.2    Sallam, A.3
  • 12
    • 33646243207 scopus 로고    scopus 로고
    • Formulation and evaluation of once-a-day transdermal gels of diclofenac diethylamine
    • Baboota, S., Shakeel, F. and Kohli, K. 2006. Formulation and evaluation of once-a-day transdermal gels of diclofenac diethylamine. Methods Find. Exp. Clin. Pharmacol. 28: 109-114.
    • (2006) Methods Find. Exp. Clin. Pharmacol. , vol.28 , pp. 109-114
    • Baboota, S.1    Shakeel, F.2    Kohli, K.3
  • 13
    • 70350641502 scopus 로고    scopus 로고
    • Effect of O-acylmenthol and salt formation on the skin permeation of diclofenac acid
    • Zhao, L., Li, Y., Fang, L., Ren, C., Xu, Y. and He, Z. 2009. Effect of O-acylmenthol and salt formation on the skin permeation of diclofenac acid. Drug Dev. Ind. Pharm. 35: 814-826.
    • (2009) Drug Dev. Ind. Pharm. , vol.35 , pp. 814-826
    • Zhao, L.1    Li, Y.2    Fang, L.3    Ren, C.4    Xu, Y.5    He, Z.6
  • 14
    • 78650546947 scopus 로고    scopus 로고
    • Optimization and formulation design of gels of Diclofenac and Curcumin for transdermal drug delivery by Box-Behnken statistical design
    • Chaudhary, H., Kohli, K., Amin, S., Rathee, P. and Kumar, V. 2011. Optimization and formulation design of gels of Diclofenac and Curcumin for transdermal drug delivery by Box-Behnken statistical design. J. Pharm. Sci. 100: 580-593.
    • (2011) J. Pharm. Sci. , vol.100 , pp. 580-593
    • Chaudhary, H.1    Kohli, K.2    Amin, S.3    Rathee, P.4    Kumar, V.5
  • 15
  • 17
    • 69249084491 scopus 로고    scopus 로고
    • Chemical Penetration Enhancers for Transdermal Drug Delivery Systems
    • Pathan, I. B. and Setty, C. M. 2009. Chemical Penetration Enhancers for Transdermal Drug Delivery Systems. Trop. J. Pharm. Res. 8: 173-179.
    • (2009) Trop. J. Pharm. Res. , vol.8 , pp. 173-179
    • Pathan, I.B.1    Setty, C.M.2
  • 18
    • 0347804138 scopus 로고    scopus 로고
    • Release rate of nimesulide from different gellants
    • Gupta, G. D. and Gound, R. S. 1999. Release rate of nimesulide from different gellants. Indian J. Pharm. Sci. 61: 229-230.
    • (1999) Indian J. Pharm. Sci. , vol.61 , pp. 229-230
    • Gupta, G.D.1    Gound, R.S.2
  • 19
    • 77649189117 scopus 로고    scopus 로고
    • A two-layer diffusive model for describing the variability of transdermal drug permeation
    • Meidan, V. M. and Pritchard, D. 2010. A two-layer diffusive model for describing the variability of transdermal drug permeation. Eur. J. Pharm. Biopharm. 74: 513-517.
    • (2010) Eur. J. Pharm. Biopharm. , vol.74 , pp. 513-517
    • Meidan, V.M.1    Pritchard, D.2
  • 20
    • 84857003532 scopus 로고    scopus 로고
    • In vitro study of percutaneous absorption of diclofenac in the presence of sodium lauryl sulphate through rabbit skin
    • Shah, S. N. H., Mahboob Rabbani, Muhammad Fakhruddin Amir. 2005. In vitro study of percutaneous absorption of diclofenac in the presence of sodium lauryl sulphate through rabbit skin. J. Res. Sci. 16: 45-50.
    • (2005) J. Res. Sci. , vol.16 , pp. 45-50
    • Shah, S.N.H.1    Rabbani, M.2    Amir, M.F.3
  • 21
    • 78649907180 scopus 로고    scopus 로고
    • Validation of a static Franz diffusion cell system for in vitro permeation studies
    • Ng, S. F., Rouse, J. J., Sanderson, F. D., Meidan, V. and Eccleston, G. M. 2010. Validation of a static Franz diffusion cell system for In vitro permeation studies. AAPS PharmSci. Tech. 11: 1432-1441.
    • (2010) AAPS PharmSci. Tech. , vol.11 , pp. 1432-1441
    • Ng, S.F.1    Rouse, J.J.2    Sanderson, F.D.3    Meidan, V.4    Eccleston, G.M.5
  • 22
    • 0036342912 scopus 로고    scopus 로고
    • Analgesic and anti-inflammatory effects of the aqueous extract of leaves of Persea americana Mill (Lauraceae)
    • Adeyemi, O. O., Okpo, S. O. and Ogunti, O. O. 2002. Analgesic and anti-inflammatory effects of the aqueous extract of leaves of Persea americana Mill (Lauraceae). Fitoterapia. 73: 375-380.
    • (2002) Fitoterapia , vol.73 , pp. 375-380
    • Adeyemi, O.O.1    Okpo, S.O.2    Ogunti, O.O.3
  • 23
    • 0019424939 scopus 로고
    • Studies on cryptolepine II: Inhibition of carrageenan induced oedema by cryptolepine
    • Bamgbose, S. O. and Noamesi, B. K. 1981. Studies on cryptolepine II: Inhibition of carrageenan induced oedema by cryptolepine. Planta Med. 41: 392-396.
    • (1981) Planta Med. , vol.41 , pp. 392-396
    • Bamgbose, S.O.1    Noamesi, B.K.2
  • 24
    • 0017101541 scopus 로고
    • Antinociceptive activity of narcotic agonist and partial agonist analgesics and other agents in the tail-immersion test in mice and rats
    • Sewell, R. D. and Spencer, P. S. 1976. Antinociceptive activity of narcotic agonist and partial agonist analgesics and other agents in the tail-immersion test in mice and rats. Neuropharmacology 15: 683-688.
    • (1976) Neuropharmacology , vol.15 , pp. 683-688
    • Sewell, R.D.1    Spencer, P.S.2
  • 25
    • 0017333312 scopus 로고
    • Restrainer and cell for dermal dosing of small laboratory animals
    • Rice, D. P. and Ketterer, D. J. 1977. Restrainer and cell for dermal dosing of small laboratory animals. Lab. Anim. Sci. 27: 72-75.
    • (1977) Lab. Anim. Sci. , vol.27 , pp. 72-75
    • Rice, D.P.1    Ketterer, D.J.2
  • 26
    • 85015578402 scopus 로고    scopus 로고
    • Dermatotoxicology: Historical perspective and advances
    • Ngo, M. A. and Maibach, H. I.2010. Dermatotoxicology: Historical perspective and advances. Toxicol. Appl. Pharmacol. 243: 225-238.
    • (2010) Toxicol. Appl. Pharmacol. , vol.243 , pp. 225-238
    • Ngo, M.A.1    Maibach, H.I.2
  • 28
    • 84964965548 scopus 로고    scopus 로고
    • Accessed on September 3 (2008).
    • World Medical Association Declaration of Helsinki. Ethical principles of medical research involving human subjects. Accessed on September 3 (2008). http://www.wma.net/en/30publications/10policies/b3/index.html.
    • Ethical Principles of Medical Research Involving Human Subjects
  • 29
    • 0034863372 scopus 로고    scopus 로고
    • Skin delivery of 5-fluorouracil from ultradeformable and standard liposomes in-vitro
    • El Maghraby, G. M. M., Williams, A. C. and Barry, B. W. 2001. Skin delivery of 5-fluorouracil from ultradeformable and standard liposomes in-vitro. J. Pharm. Pharmacol. 53:1069-1077.
    • (2001) J. Pharm. Pharmacol. , vol.53 , pp. 1069-1077
    • El Maghraby, G.M.M.1    Williams, A.C.2    Barry, B.W.3
  • 30
    • 0035043181 scopus 로고    scopus 로고
    • Nutritional skin care: Health effects of micronutrients and fatty acids
    • Boelsma, E., Hendriks, H. F. J. and Roza, L. 2001. Nutritional skin care: health effects of micronutrients and fatty acids. Am. J. Clin. Nutr. 73: 853-864.
    • (2001) Am. J. Clin. Nutr. , vol.73 , pp. 853-864
    • Boelsma, E.1    Hendriks, H.F.J.2    Roza, L.3
  • 31
    • 29244479590 scopus 로고    scopus 로고
    • Interactions of oleic acid and model stratum corneum membranes as seen by 2H NMR
    • Rowat, A. C., Kitson, N. and Thewalt, J. L. 2006. Interactions of oleic acid and model stratum corneum membranes as seen by 2H NMR. Int. J. Pharm. 307: 225-331.
    • (2006) Int. J. Pharm. , vol.307 , pp. 225-331
    • Rowat, A.C.1    Kitson, N.2    Thewalt, J.L.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.