Anti-inflammatory activity of gel containing novel elastic niosomes entrapped with diclofenac diethylammonium

International Journal of Pharmaceutics

Volumn 360, Issue 1-2, 2008, Pages 156-163

  Manosroi, A ^a   Jantrawut, P ^a   Manosroi, J ^a  

^a CHIANG MAI UNIVERSITY   (Thailand)

Author keywords

Anti inflammatory; Diclofenac; Elastic niosomes; Ethanol; Rat skin transdermal; Tween 61

Indexed keywords

ALCOHOL; BENZENE DERIVATIVE; CARBOMER; CHOLESTEROL; DICLOFENAC DERIVATIVE; DICLOFENAC DIETHYLAMMONIUM; NIOSOME; PHENYLBUTAZONE; POLYSORBATE 60; SORBITAN STEARATE;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ANTIINFLAMMATORY ACTIVITY; ARTICLE; BILAYER MEMBRANE; CONTROLLED STUDY; DERMIS; DIFFUSION; DRUG ABSORPTION; DRUG FORMULATION; DRUG STRUCTURE; EDEMA; ELASTICITY; EPIDERMIS; GEL; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; IN VITRO STUDY; IN VIVO STUDY; MALE; NONHUMAN; PARTICLE SIZE; PRIORITY JOURNAL; QUANTITATIVE ANALYSIS; RAT; SEDIMENTATION; SEPARATION TECHNIQUE; SKIN ABSORPTION; STRATUM CORNEUM; ZETA POTENTIAL;

ADMINISTRATION, CUTANEOUS; ANIMALS; ANTI-INFECTIVE AGENTS, LOCAL; ANTI-INFLAMMATORY AGENTS, NON-STEROIDAL; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; DICLOFENAC; DRUG COMPOUNDING; DRUG STABILITY; ELASTICITY; ELECTROCHEMISTRY; ETHANOL; GELS; LIPID BILAYERS; LIPOSOMES; MALE; MICROSCOPY, ELECTRON, SCANNING; PARTICLE SIZE; RATS; RATS, SPRAGUE-DAWLEY; SKIN ABSORPTION; SOLVENTS;

EID: 47249114766     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2008.04.033     Document Type: Article

References (27)

1. Bangham A.D., Standish M.M., and Walkins J.C. Diffusion of univalent ions across the lamellar of swollen phospholipids. J. Mol. Biol. 13 (1965) 238-252
2. Barry A.L., and Cullis P.R. Direct NMR evidence for ethanol binding to the lipid-water interface of phospholipid bilayers. Biochemistry 33 (1995) 8082-8088
3. Brattsand R., Thalen A., Roempke K., Kallstrom L., and Gruvstad E. Influence of 16α, 17α-acetal substitution and steroid nucleus fluorination on the topical to systemic activity ratio of glucocorticoids. J. Steroid Biochem. 16 (1982) 779-786
4. Bochot A., Fattal E., and Gulik A. Liposomes dispersed within a thermosensitive gel: a new dosage form for ocular delivery of oligonucleotides. Pharm. Res. 15 (1998) 1364-1369
5. Burnham R., Gregy R., Healy P., and Steadward R. The effectiveness of topical diclofenac for lateral epicondylitis. Clin. J. Sport Med. 8 (1998) 78-81
6. Cevc G. Transfersomes, liposomes and other lipid suspensions on the skin: permeation enhancement, vesicle penetration, and transdermal drug delivery. Crit. Rev. Ther. Drug Carrier Syst. 13 (1996) 257-388
7. Cevc G., Blume G., Schätzlein A., Gebauer D., and Paul A. The skin: a pathway for systemic treatment with patches and lipid-based agent carriers. Adv. Drug Rev. 18 (1996) 349-378
8. Cevc G., Blume G., and Schatzlein A. J. Control. Rel. 45 (1997) 211-226
9. Dayan N., and Touitou E. Carriers for skin delivery of trihexyphenidyl HCl: ethosomes vs. liposomes. Biomaterials 21 (2000) 1879-1885
10. Dubey V., Mishra D., and Jain N.K. Melatonin loaded ethanolic liposomes: physico-chemical characterization and enhanced transdermal delivery. Eur. J. Pharm. Biopharm. 67 (2007) 398-405
11. Friberg S.E., and Osborne D.W. Small angle X-ray diffraction patterns of stratum corneum and a model structure for its lipids. J. Disper. Sci. Technol. 6 (1985) 485-495
12. Glavas-Dodov M., Goracinova K., and Mladenovska K. Release profile of lidocaine HCl from topical liposomal gel formulation. Int. J. Pharm. 242 (2002) 381-384
13. Grace D., Rogers J., Skeith K., and Anderson K. Topical diclofenac versus placebo: a double blind, randomized clinical trial in patients with oesteoarthritis of the knee. J. Rheumatol. 26 (1999) 2659-2663
14. Jain S., Jain P., Umamaheshwari R.B., and Jain N.K. Drug. Dev. Ind. Pharm. 29 (2003) 1013-1026
15. Kirjavainen M., Urtti A., Valjakka-Koskela R., Kiesvaara J., and Monkkonen J. Liposome-skin interactions and their effects on the skin permeation of drugs. Eur. J. Pharm. Sci. 7 (1999) 279-286
16. Lasic D., Weiner N., Riaz M., and Martin F. Liposomes. In: Lieberman A., Rieger M., and Banker G. (Eds). Pharmaceutical Dosage Forms: Disperse Systems vol. 3 (1998), Marcel Dekker, NY 8-43
17. Castanho M.A.R.B., Santos N.C., and Loura L.M.S. Separating the turbidity spectra of vesicles from the absorption spectra of membrane probes and other chromophores. Eur. Biophys. J. 26 (1997) 253-259
18. Namdeo A., and Jain N.K. Niosomes as drug carriers. Ind. J. Pharm. Sci. 58 (1996) 41-46
19. Nishihata T., Kotera K., Nakano Y., and Yamazaki M. Rat percutaneous transport of diclofenac and influence of hydrogenated soya phospholipids. Chem. Pharm. Bull. 35 (1987) 3807-3812
20. Obata Y.T., Takayama K., Maitaini Y., Machida Y., and Nagai T. Int. J. Pharm. 89 (1993) 91-98
21. Plessis J., Egbaria K., and Weiner N. Influence of formulation factors on the deposition of liposomal components into the different strata of the skin. J. Soc. Cosmet. Chem. 43 (1992) 93-100
22. Raja-Naresh R.A., Singh U.V., Udupa N., and Pillai G.K. Anti-inflammatory activity of niosome encapsulated diclofenac sodium in rats. Ind. Drugs 30 (1993) 275-278
23. Ruel-Gariepy E., Leclair G., and Hildgen P. Thermosensitive chitosan based on hydrogel containing liposomes for the delivery of hydrophilic molecules. J. Control. Rel. 30 (1994) 1-15
24. Touitou E., Dayan N., Bergelson L., Godin B., and Eliaz M. Ethosomes-novel vesicular carriers: characterization and delivery properties. J. Control. Rel. 65 (2000) 403-418
25. Valjakka-Koskela R., Kirjavainen M., Mönkkönen J., Urtti A., and Kiesvaara J. Enhancement of percutaneous absorption of naproxen by phospholipids. Int. J. Pharm. 175 (1998) 225-230
26. Van, D., Bergh, B.A.I., 1999. Elastic liquid state vesicles as a tool for topical drug delivery. Thesis. Leiden University, The Netherlands, pp. 49-80.
27. Young J.M., Wagner B.M., and Spires D.A. Tachyphylaxis in 12-O-tetradecanoylphobal acetate- and arachidonic acid-induced ear edema. J. Invest. Dermatol. 80 (1983) 48-52