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Volumn 12, Issue 7, 2012, Pages 523-532

Plasma and Cerebrospinal Fluid Pharmacokinetic Parameters After Single-Dose Administration of Intravenous, Oral, or Rectal Acetaminophen

Author keywords

Analgesia; Drug administration routes

Indexed keywords

FEVERALL; PARACETAMOL; UNCLASSIFIED DRUG;

EID: 84865980531     PISSN: 15307085     EISSN: 15332500     Source Type: Journal    
DOI: 10.1111/j.1533-2500.2012.00556.x     Document Type: Article
Times cited : (187)

References (36)
  • 2
    • 34147123764 scopus 로고    scopus 로고
    • Paracetamol (acetaminophen) penetrates readily into the cerebrospinal fluid of children after intravenous administration
    • Kumpulainen E, Kokki H, Halonen T, Heikkinen M, Savolainen J, Laisalmi M. Paracetamol (acetaminophen) penetrates readily into the cerebrospinal fluid of children after intravenous administration. Pediatrics. 2007;119:766-771.
    • (2007) Pediatrics , vol.119 , pp. 766-771
    • Kumpulainen, E.1    Kokki, H.2    Halonen, T.3    Heikkinen, M.4    Savolainen, J.5    Laisalmi, M.6
  • 3
    • 0026653542 scopus 로고
    • Plasma and cerebrospinal fluid concentrations of paracetamol after a single dose of propacetamol
    • Bannwarth B, Netter P, Lapicque F, et al. Plasma and cerebrospinal fluid concentrations of paracetamol after a single dose of propacetamol. Br J Clin Pharmacol. 1992;34:79-81.
    • (1992) Br J Clin Pharmacol , vol.34 , pp. 79-81
    • Bannwarth, B.1    Netter, P.2    Lapicque, F.3
  • 4
    • 79954612747 scopus 로고    scopus 로고
    • A randomized study of the efficacy and safety of intravenous acetaminophen compared to oral acetaminophen for the treatment of fever
    • Peacock WF, Breitmeyer JB, Pan C, Smith WB, Royal MA. A randomized study of the efficacy and safety of intravenous acetaminophen compared to oral acetaminophen for the treatment of fever. Acad Emer Med. 2011;18:360-366.
    • (2011) Acad Emer Med , vol.18 , pp. 360-366
    • Peacock, W.F.1    Breitmeyer, J.B.2    Pan, C.3    Smith, W.B.4    Royal, M.A.5
  • 5
    • 20444364569 scopus 로고    scopus 로고
    • Intravenous acetaminophen reduced the use of opioids compared with oral administration after coronary artery bypass grafting
    • Pettersson PH, Jakobsson J, Owall A. Intravenous acetaminophen reduced the use of opioids compared with oral administration after coronary artery bypass grafting. J Cardiothorac Vasc Anesth. 2005;19(3):306-309.
    • (2005) J Cardiothorac Vasc Anesth , vol.19 , Issue.3 , pp. 306-309
    • Pettersson, P.H.1    Jakobsson, J.2    Owall, A.3
  • 6
    • 84865965630 scopus 로고    scopus 로고
    • Open-label, 4-period, randomized crossover study to determine the comparative pharmacokinetics of oral and intravenous acetaminophen administration in healthy male volunteers. Poster presentation at the 32nd Annual Meeting and Workshops American Society of Regional Anesthesia and Pain (ASRA), April 19-22, Vancouver, Canada.
    • Schutz RA, Fong L, Chang Y, Royal MA. Open-label, 4-period, randomized crossover study to determine the comparative pharmacokinetics of oral and intravenous acetaminophen administration in healthy male volunteers. Poster presentation at the 32nd Annual Meeting and Workshops American Society of Regional Anesthesia and Pain (ASRA), April 19-22, 2007; Vancouver, Canada.
    • (2007)
    • Schutz, R.A.1    Fong, L.2    Chang, Y.3    Royal, M.A.4
  • 7
    • 79953210415 scopus 로고    scopus 로고
    • Randomised controlled trial comparing oral and intravenous paracetamol (acetaminophen) plasma levels when given as preoperative analgesia
    • van der Westhuizen J, Kuo PY, Reed PW, Holder K. Randomised controlled trial comparing oral and intravenous paracetamol (acetaminophen) plasma levels when given as preoperative analgesia. Anaesth Intensive Care. 2011;39:242-246.
    • (2011) Anaesth Intensive Care , vol.39 , pp. 242-246
    • van der Westhuizen, J.1    Kuo, P.Y.2    Reed, P.W.3    Holder, K.4
  • 8
    • 0030449595 scopus 로고    scopus 로고
    • Analgesic efficacy of paracetamol in children using tonsillectomy as a pain model
    • Anderson B, Kanagasundarum S, Woollard G. Analgesic efficacy of paracetamol in children using tonsillectomy as a pain model. Anaesth Intens Care. 1996;24:669-673.
    • (1996) Anaesth Intens Care , vol.24 , pp. 669-673
    • Anderson, B.1    Kanagasundarum, S.2    Woollard, G.3
  • 10
    • 0029847084 scopus 로고    scopus 로고
    • The relative bioavailability of paracetamol in suppositories preparations in comparison to tablets (in German)
    • Blume H, Ali SL, Elze M, Krämer J, Scholz ME. The relative bioavailability of paracetamol in suppositories preparations in comparison to tablets (in German). Arzneimittelforschung. 1996;46(10):975-980.
    • (1996) Arzneimittelforschung , vol.46 , Issue.10 , pp. 975-980
    • Blume, H.1    Ali, S.L.2    Elze, M.3    Krämer, J.4    Scholz, M.E.5
  • 12
    • 0034011991 scopus 로고    scopus 로고
    • High-dose rectal and oral acetaminophen in postoperative patients - serum and saliva concentrations
    • Hahn TW, Mogensen T, Lund C, Schouenborg L, Rasmussen M. High-dose rectal and oral acetaminophen in postoperative patients - serum and saliva concentrations. Acta Anaesthesiol Scand. 2000;44:302-306.
    • (2000) Acta Anaesthesiol Scand , vol.44 , pp. 302-306
    • Hahn, T.W.1    Mogensen, T.2    Lund, C.3    Schouenborg, L.4    Rasmussen, M.5
  • 13
    • 0036725846 scopus 로고    scopus 로고
    • Comparison of oral versus normal and high-dose rectal acetaminophen in the treatment of febrile children
    • Scolnik D, Kozer E, Jacobson S, Diamond S, Young NL. Comparison of oral versus normal and high-dose rectal acetaminophen in the treatment of febrile children. Pediatrics. 2002;110(3):553-556.
    • (2002) Pediatrics , vol.110 , Issue.3 , pp. 553-556
    • Scolnik, D.1    Kozer, E.2    Jacobson, S.3    Diamond, S.4    Young, N.L.5
  • 14
    • 0034912427 scopus 로고    scopus 로고
    • Analgesic efficacy of rectal versus oral acetaminophen in children after major craniofacial surgery
    • van der Marel CD, van Lingen RA, Pluim MAL, et al. Analgesic efficacy of rectal versus oral acetaminophen in children after major craniofacial surgery. Clin Pharmacol Ther. 2001;70(1):82-90.
    • (2001) Clin Pharmacol Ther , vol.70 , Issue.1 , pp. 82-90
    • van der Marel, C.D.1    van Lingen, R.A.2    Pluim, M.A.L.3
  • 15
    • 84865990791 scopus 로고    scopus 로고
    • PK/PD comparison of IV vs rectal acetaminophen administration: a simulation based on a population pharmacokinetic model. Poster presentation at the 111th Annual Meeting of the American Society of Clinical Pharmacology and Therapeutics (ASCPT). March 17-20, Atlanta GA. Poster #PII-82.
    • Breitmeyer JB, Mouksassi S, Gosselin NH, Royal MA. PK/PD comparison of IV vs rectal acetaminophen administration: a simulation based on a population pharmacokinetic model. Poster presentation at the 111th Annual Meeting of the American Society of Clinical Pharmacology and Therapeutics (ASCPT). March 17-20, 2010. Atlanta GA. Poster #PII-82.
    • (2010)
    • Breitmeyer, J.B.1    Mouksassi, S.2    Gosselin, N.H.3    Royal, M.A.4
  • 16
    • 38949212262 scopus 로고    scopus 로고
    • Randomized controlled trial of duration of analgesia following intravenous or rectal acetaminophen after adenotonsillectomy in children
    • Capici F, Ingelmo PM, Davidson A, et al. Randomized controlled trial of duration of analgesia following intravenous or rectal acetaminophen after adenotonsillectomy in children. Paediatrics. 2008;100(2):251-255.
    • (2008) Paediatrics , vol.100 , Issue.2 , pp. 251-255
    • Capici, F.1    Ingelmo, P.M.2    Davidson, A.3
  • 17
    • 33750112852 scopus 로고    scopus 로고
    • Plasma concentrations following repeated rectal of intravenous administration of paracetamol after heart surgery
    • Pettersson PH, Jakobsson J, Öwall A. Plasma concentrations following repeated rectal of intravenous administration of paracetamol after heart surgery. Acta Anaesthesiol Scand. 2006;50:673-677.
    • (2006) Acta Anaesthesiol Scand , vol.50 , pp. 673-677
    • Pettersson, P.H.1    Jakobsson, J.2    Öwall, A.3
  • 18
    • 0027844990 scopus 로고
    • Pharmacokinetics of acetaminophen in the cerebrospinal fluid in elderly population (in French)
    • Moreau X, Le Quay L, Granry JC, Boishardy N, Delhumeau A. Pharmacokinetics of acetaminophen in the cerebrospinal fluid in elderly population (in French). Therapy. 1993;48:393-396.
    • (1993) Therapy , vol.48 , pp. 393-396
    • Moreau, X.1    Le Quay, L.2    Granry, J.C.3    Boishardy, N.4    Delhumeau, A.5
  • 19
    • 33645211311 scopus 로고    scopus 로고
    • Paracetamol concentrations in plasma and cerebrospinal fluid
    • Abstract A-785.
    • Jensen LL, Handberg G, Brøsen K, Schmedes A, Ørding H. Paracetamol concentrations in plasma and cerebrospinal fluid. Eur J Anaesthesiol. 2004;21(S32):193. Abstract A-785.
    • (2004) Eur J Anaesthesiol , vol.21 S , Issue.32 , pp. 193
    • Jensen, L.L.1    Handberg, G.2    Brøsen, K.3    Schmedes, A.4    Ørding, H.5
  • 20
    • 84890724975 scopus 로고    scopus 로고
    • Chapter 6: Analgesia and sedation. In: Arcara K, Tschudy M, eds. 19th ed. Philadelphia, PA: Mosby.
    • Chapter 6: Analgesia and sedation. In: Arcara K, Tschudy M, eds. Johns Hopkins Hospital. The Harriet Lane Handbook. 19th ed. Philadelphia, PA: Mosby; 2012.
    • (2012) Johns Hopkins Hospital. The Harriet Lane Handbook
  • 22
    • 0038186605 scopus 로고    scopus 로고
    • Acetaminophen toxicity in children
    • American Academy of Pedatrics.
    • American Academy of Pedatrics. Acetaminophen toxicity in children. Pediatrics. 2001;108:1020-1024.
    • (2001) Pediatrics , vol.108 , pp. 1020-1024
  • 23
    • 0024267858 scopus 로고
    • Characterization of an "in vitro" blood-brain barrier: effects of molecular size and lipophilicity on cerebrovascular endothelial transport rates of drugs
    • van Bree JB, de Boer AG, Danhof M, Ginsel LA, Breimer DD. Characterization of an "in vitro" blood-brain barrier: effects of molecular size and lipophilicity on cerebrovascular endothelial transport rates of drugs. J Pharmacol Exp Ther. 1988;247(3):1233-1239.
    • (1988) J Pharmacol Exp Ther , vol.247 , Issue.3 , pp. 1233-1239
    • van Bree, J.B.1    de Boer, A.G.2    Danhof, M.3    Ginsel, L.A.4    Breimer, D.D.5
  • 24
    • 0018163621 scopus 로고
    • Aspirin versus acetaminophen: a comparative view
    • Rumack BH. Aspirin versus acetaminophen: a comparative view. Pediatrics. 1978;62:943-946.
    • (1978) Pediatrics , vol.62 , pp. 943-946
    • Rumack, B.H.1
  • 25
    • 84865967136 scopus 로고
    • Pharmacodynamic modeling of the analgesic properties of specific non-opioid analgesics using the dental pain model
    • Hutcheson SJ, Mason WD. Pharmacodynamic modeling of the analgesic properties of specific non-opioid analgesics using the dental pain model. Dissertation Abstracts International. 1993;54(3-B):1354.
    • (1993) Dissertation Abstracts International , vol.54 , Issue.3 , pp. 1354
    • Hutcheson, S.J.1    Mason, W.D.2
  • 26
    • 85030487251 scopus 로고
    • Fort Washington, PA: McNeil Consumer & Specialty Pharmaceuticals;, Submitted to NDA 19-872 as a postapproval commitment.
    • ® Caplets. Fort Washington, PA: McNeil Consumer & Specialty Pharmaceuticals; 1995, Submitted to NDA 19-872 as a postapproval commitment.
    • (1995) ® Caplets
    • Gelotte, C.K.1
  • 28
    • 0029101096 scopus 로고
    • Bioavailability of medication after laparoscopic cholecystectomy
    • Elfant AB, Levine SM, Cencora B, et al. Bioavailability of medication after laparoscopic cholecystectomy. J Laparoendosc Surg. 1995;5(4):237-240.
    • (1995) J Laparoendosc Surg , vol.5 , Issue.4 , pp. 237-240
    • Elfant, A.B.1    Levine, S.M.2    Cencora, B.3
  • 29
    • 0026601632 scopus 로고
    • Gastric emptying after minor gynaecological surgery. The effect of anaesthetic technique
    • Mushambi MC, Rowbotham DJ, Bailey SM. Gastric emptying after minor gynaecological surgery. The effect of anaesthetic technique. Anaesthesia. 1992;47(4):297-299.
    • (1992) Anaesthesia , vol.47 , Issue.4 , pp. 297-299
    • Mushambi, M.C.1    Rowbotham, D.J.2    Bailey, S.M.3
  • 30
    • 0028957311 scopus 로고
    • Bioavailability of medication delivered via nasogastric tube is decreased in the immediate postoperative period
    • Elfant AB, Levine SM, Peikin SR, et al. Bioavailability of medication delivered via nasogastric tube is decreased in the immediate postoperative period. Am J Surg. 1995;169(4):430-432.
    • (1995) Am J Surg , vol.169 , Issue.4 , pp. 430-432
    • Elfant, A.B.1    Levine, S.M.2    Peikin, S.R.3
  • 32
    • 0024145446 scopus 로고
    • Postoperative gastric emptying in outpatient anesthesia: the effect of opioid supplementation
    • Milligan KR, Howe JP, McClean E, Dundee JW. Postoperative gastric emptying in outpatient anesthesia: the effect of opioid supplementation. J Clin Anesth. 1988;1(1):9-11.
    • (1988) J Clin Anesth , vol.1 , Issue.1 , pp. 9-11
    • Milligan, K.R.1    Howe, J.P.2    McClean, E.3    Dundee, J.W.4
  • 33
    • 0028963040 scopus 로고
    • Normal postoperative gastric emptying after orthopaedic surgery with spinal anaesthesia and i.m. ketorolac as the first postoperative analgesic
    • Petring OU, Dawson PJ, Blake DW, et al. Normal postoperative gastric emptying after orthopaedic surgery with spinal anaesthesia and i.m. ketorolac as the first postoperative analgesic. Br J Anaesth. 1995;74(3):257-260.
    • (1995) Br J Anaesth , vol.74 , Issue.3 , pp. 257-260
    • Petring, O.U.1    Dawson, P.J.2    Blake, D.W.3
  • 34
    • 0031787401 scopus 로고    scopus 로고
    • Effects of low-dose morphine on gastric emptying in healthy volunteers
    • Yuan CS, Foss JF, O'Connor M, Roizen MF, Moss J. Effects of low-dose morphine on gastric emptying in healthy volunteers. J Clin Pharmacol. 1998;38(11):1017-1020.
    • (1998) J Clin Pharmacol , vol.38 , Issue.11 , pp. 1017-1020
    • Yuan, C.S.1    Foss, J.F.2    O'Connor, M.3    Roizen, M.F.4    Moss, J.5
  • 35
    • 0020456538 scopus 로고
    • Effect of food on acetaminophen absorption in young and elderly subjects
    • Divoll M, Greenblatt DJ, Ameer B, Abernethy DR. Effect of food on acetaminophen absorption in young and elderly subjects. J Clin Pharmacol. 1982;22(11-12):571-576.
    • (1982) J Clin Pharmacol , vol.22 , Issue.11-12 , pp. 571-576
    • Divoll, M.1    Greenblatt, D.J.2    Ameer, B.3    Abernethy, D.R.4
  • 36
    • 58849114491 scopus 로고    scopus 로고
    • Influence of posture on pharmacokinetics
    • Queckenberg C, Fuhr U. Influence of posture on pharmacokinetics. Eur J Clin Pharmacol. 2009;65(2):109-119.
    • (2009) Eur J Clin Pharmacol , vol.65 , Issue.2 , pp. 109-119
    • Queckenberg, C.1    Fuhr, U.2


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