Cholorpheniramine tannate complexes: Physicochemical, chemometric, and taste masking evaluation

International Journal of Pharmaceutics

Volumn 436, Issue 1-2, 2012, Pages 582-592

  Rahman, Ziyaur ^a,c   Zidan, Ahmed S ^a,b   Khan, Saeed R ^a   Reddy, Indra K ^c   Khan, Mansoor A ^a  

^a CENTER FOR DRUG EVALUATION AND RESEARCH   (United States)

^b Zagazig University   (Egypt)

^c TEXAS A AND M HEALTH SCIENCE CENTER   (United States)

Author keywords

Bitter taste; Chemometric model; Cholorpheniramine maleate; Complex; Dissolution; Solubility; Tannic acid

Indexed keywords

CHLORPHENIRAMINE MALEATE; MICROCRYSTALLINE CELLULOSE; TANNIN;

ACCURACY; ARTICLE; BITTER TASTE; CHEMOMETRIC ANALYSIS; COMPLEX FORMATION; DRUG FORMULATION; DRUG SCREENING; DRUG SOLUBILITY; EVAPORATION; INFRARED SPECTROSCOPY; MASKING; PH; PHYSICAL CHEMISTRY; PRIORITY JOURNAL; SUSTAINED DRUG RELEASE; X RAY DIFFRACTION;

ANTI-ALLERGIC AGENTS; CALORIMETRY, DIFFERENTIAL SCANNING; CELLULOSE; CHLORPHENIRAMINE; DELAYED-ACTION PREPARATIONS; DIAGNOSTIC EQUIPMENT; EXCIPIENTS; MICROSCOPY, ELECTRON, SCANNING; POWDER DIFFRACTION; SOLUBILITY; SPECTROSCOPY, FOURIER TRANSFORM INFRARED; SPECTROSCOPY, NEAR-INFRARED; TASTE; X-RAY DIFFRACTION;

EID: 84865289881     PISSN: 03785173     EISSN: 18733476     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2012.07.037     Document Type: Article

References (37)

1. R. Agarwal, R. Mittal, and A. Singh Studies of ion-exchange resin complex of chloroquine phosphate Drug Dev. Ind. Pharm. 26 2000 773 776
2. M.G. Albu, M.V. Ghica, M. Leca, L. Popa, C. Borlescu, E. Cremenescu, M. Giurginca, and V. Trandafir Doxycycline delivery from collagen matrices crosslinked with tannic acid Mol. Cryst. Liq. Cryst. 523 2010 97 105
3. G.M.O. Barra, S.J. Crespo, J.R. Bertolino, V. Soldi, and A.T.N. Pires Maleic anhydride grafting on EPDM: qualitative and quantitative determination J. Braz. Chem. Soc. 10 1999 31 34
4. S.K. Baveja, K.V.R. Rao, R. Kumar, and K.P. Devi Sustained release tablet formulation of diethylcarbamazine. Part II Int. J. Pharm. 24 1985 355 358
5. T.K. Bhat, B. Singh, and O.P. Sharma Microbial degradation of tannins - current perspective Biodegradation 9 1998 343 357
6. S. Burgalassi, L. Panichi, M.F. Saettone, J. Jacobsen, and M.R. Rassing Development and in vitro/in vivo testing of mucoadhesive buccal patches releasing benzydamine and lidocaine Int. J. Pharm. 133 1996 1 7
7. C.J. Cavallito, L. Chafetz, and L.D. Miller Some studies of a sustained release principle J. Pharm. Sci. 52 1963 259 263
8. C.J. Cavallito, and R. Jewell Modification of rates of gastrointestinal absorption of drugs. I. Amines J. Am. Pharm. Assoc. 47 1958 165 168
9. R. Chopra, G. Alderborn, J.M. Newton, and F. Podczeck The influence of film coating on pellet properties Pharm. Dev. Technol. 7 2002 59 68
10. C. Dollery Therapeutic Drugs 1991 Churchill Living Stones New York pp. 198-200
11. A.E. Hagerman, and L.G. Butler The specificity of proanthocyanidin- protein interaction J. Biol. Chem. 256 1981 4494 4497
12. R. Herrera-Becerra, J.L. Rius, and C. Zorrilla Tannin biosynthesis of iron oxide nanoparticles Appl. Phys. A 100 2010 453 459
13. B.T. Hiep, C. Fernandez, M. Tod, H. Banide, A. Thuillier, B. Lacour, R. Farinotti, and R. Gimenez Intestinal absorption and metabolism of chlorpheniramine enantiomers in rat Chirality 13 2001 207 213
14. I.S. Iman, A.S. Nadia, and M.A. Ebtsam Formulation and stability study of chlorpheniramine maleate transdermal patch Asian J. Pharm. 4 2010 17 23
15. J.C. Isenburg, N.V. Karamchandani, D.T. Simionescu, and N.R. Vyavahare Structural requirements for stabilization of vascular elastin by polyphenolic tannins Biomaterials 27 2006 3645 3651
16. International conference of harmonization-validation of analytical procedures Q2(R1), 2005.
17. B.G. Katzung Basic and Clinical Pharmacology 2007 McGraw Hill Boston pp. 1043-1049
18. N.S. Khan, A. Ahmad, and S.M. Hadi Anti-oxidant, pro-oxidant properties of tannic acid and its binding to DNA Chem. Biol. Interact. 125 2000 177 189
19. B.S. Kim, H.I. Lee, Y. Min, Z. Poon, and P.T. Hammond Hydrogen bonded multilayer of pH-responsive polymeric micelles with tannic acid for surface drug delivery Chem. Commun. 28 2009 4194 4196
20. P. Li, S.E. Tabibi, and S.H. Yalkowsky Solubilization of flavopiridol by pH control combined with cosolvents, surfactants, or complexants J. Pharm. Sci. 88 1999 945 947
21. J.K. Lorenz, J.P. Reo, O. Hendl, J.H. Worthington, and V.D. Petrossian Evaluation of a taste sensor instrument (electronic tongue) for use in formulation development Int. J. Pharm. 367 2009 65 72
22. M. Martinez-Gomez, S. Sagrado, R.M. Villanueva-Camanas, and M.J. Medina-Hernandez Enantiomeric quality control of antihistamines in pharmaceuticals by affinity electrokinetic chromatography with human serum albumin as chiral selector Anal. Chim. Acta 592 2007 202 209
23. a of the antihistaminic drug chlorpheniramine maleate by supramolecular interactions with water-soluble polymers Polymer 48 2007 799 804
24. N. Ono, Y. Miyamoto, T. Ishiguro, K. Motoyama, F. Hirayama, D. Iohara, H. Seo, S. Tsuruta, H. Arima, and K. Uekama Reduction of bitterness of antihistaminic drugs by complexation with β-cyclodextrins J. Pharm. Sci. 100 2011 1935 1943
25. M. Otsuka, and H. Kinoshita Quantitative determination of hydrate content of theophylline powder by chemometric X-ray powder diffraction analysis AAPS PharmSciTech 11 2010 204 211
26. Y. Raghunathan, L. Amsel, O. Hinsvark, and W. Bryant Sustained-release drug delivery system I: coated ion-exchange resin system for phenylpropanolamine and other drugs J. Pharm. Sci. 70 1981 379 384
27. Z. Rahman, A.S. Zidan, R.T. Berendt, and M.A. Khan Tannate complexes of antihistaminic drug: sustained release and taste masking approaches Int. J. Pharm. 422 2012 91 100
28. Z. Rahman, A.S. Zidan, and M.A. Khan Non-destructive methods of characterization of risperidone solid lipid nanoparticles Eur. J. Pharm. Biopharm. 76 2010 127 137
29. M. Rani, A. Agarwal, and Y.S. Negi Characterization and biodegradation studies for interpenetrating polymeric network (IPN) of chitosan-amino acid beads J. Biomat. Nanobiotechnol. 2 2011 71 84
30. 1 receptor antagonist drugs New Engl. J. Med. 330 1994 1663 1670
31. M.O. Taha, W. Nasser, A. Ardakani, and H.S. AlKhatib Sodium lauryl sulfate impedes drug release from zinc-crosslinked alginate beads: switching from enteric coating release into biphasic profiles Int. J. Pharm. 350 2008 291 300
32. J. Varshosaz, A. Pardakhty, and S.M.H. Baharanchi Sorbitan monopalmitate-based proniosomes for transdermal delivery of chlorpheniramine maleate Drug Deliv. 12 2005 75 82
33. K. Woertz, C. Tissen, P. Kleinebudde, and J. Breitkreutz A comparative study on two electronic tongues for pharmaceutical formulation development J. Pharm. Biomed. Anal. 55 2011 272 281
34. Z.Q. Zhang, C.H. Pan, and D. Chung Tannic acid cross-linked gelatin-gum arabic coacervate microspheres for sustained release of allyl isothiocyanate: characterization and in vitro release study Food Res. Int. 44 2011 1000 1007
35. J.Y. Zheng, and M.P. Keeney Taste masking analysis in pharmaceutical formulation development using an electronic tongue Int. J. Pharm. 310 2006 118 124
36. Y. Zhu, N.H. Shah, A.W. Malick, M.H. Infeld, and J.W. McGinity Solid-state plasticization of an acrylic polymer with chlorpheniramine maleate and triethyl citrate Int. J. Pharm. 241 2002 301 310
37. A.S. Zidan, C. Spinks, J. Fortunak, M. Habib, and M.A. Khan Near-infrared investigations of novel anti-HIV tenofovir liposomes AAPS J. 12 2010 202 214