Synthesis and biological evaluation of andrographolide derivatives as potent anti-HIV agents

Archiv der Pharmazie

Volumn 345, Issue 8, 2012, Pages 647-656

  Tang, Chunlei ^a,b   Liu, Yajuan ^c,d   Wang, Bin ^a,e   Gu, Guolong ^a   Yang, Liumeng ^c   Zheng, Yongtang ^c   Qian, Hai ^a   Huang, Wenlong ^a  

^a CHINA PHARMACEUTICAL UNIVERSITY   (China)

^b JIANGNAN UNIVERSITY   (China)

^c KUNMING INSTITUTE OF ZOOLOGY   (China)

^d UNIVERSITY OF CHINESE ACADEMY OF SCIENCES   (China)

^e Technology Center   (China)

Author keywords

Andrographolide derivatives; Anti HIV; Synthesis

Indexed keywords

19 O TRITYLDEHYDROANDROGRAPHOLIDE; 3 O ICOTINOYL 19 O (1 NAPHTHALENE ACETYL)DEHYDROANDROGRAPHOLIDE; 3 O ICOTINOYL 19 O (3 PHENYLPROPIONYL)DEHYDROANDROGRAPHOLIDE; 3 O NICOTINOYL 19 O (2 ETHYLHEXANOYL)DEHYDROANDROGRAPHOLIDE; 3 O NICOTINOYL 19 O (2 FCHLOROBENZOYL)DEHYDROANDROGRAPHOLIDE; 3 O NICOTINOYL 19 O (2 NITROBENZOYL)DEHYDROANDROGRAPHOLIDE; 3 O NICOTINOYL 19 O (2 QUINOLINEFORMYL)DEHYDROANDROGRAPHOLIDE; 3 O NICOTINOYL 19 O (3,4 DIMETHOXYPHENYLACETYL)DEHYDROANDROGRAPHOLIDE; 3 O NICOTINOYL 19 O (3,5 DINITRYLBENZOYL)DEHYDROANDROGRAPHOLIDE; 3 O NICOTINOYL 19 O (4 FLUOROBENZOYL)DEHYDROANDROGRAPHOLIDE; 3 O NICOTINOYL 19 O (4 METHOXYLBENZOYL))DEHYDROANDROGRAPHOLIDE; 3 O NICOTINOYL 19 O (4 TOLUENESULFONYL)DEHYDROANDROGRAPHOLIDE; 3 O NICOTINOYL 19 O (N BUTYRYL)DEHYDROANDROGRAPHOLIDE; 3 O NICOTINOYL 19 O (N DECANOYL)DEHYDROANDROGRAPHOLIDE; 3 O NICOTINOYL 19 O ACETYLDEHYDROANDROGRAPHOLIDE; 3 O NICOTINOYL 19 O BENZOYLDEHYDROANDROGRAPHOLIDE; 3 O NICOTINOYL 19 O BROMOACETYLDEHYDROANDROGRAPHOLIDE; 3 O NICOTINOYL 19 O PALMITOYLDEHYDROANDROGRAPHOLIDE; 3 O NICOTINOYL 19 O PHENOXYACETYLDEHYDROANDROGRAPHOLIDE; 3 O NICOTINOYL 19 O PHENYLACETYLDEHYDROANDROGRAPHOLIDE; 3 O NICOTINOYL 19 O STEAROYLDEHYDROANDROGRAPHOLIDE; 3 O NICOTINOYL 19 O TRITYLDEHYDROANDROGRAPHOLIDE; 3 O NICOTINOYLDEHYDROANDROGRAPHOLIDE; ANDROGRAPHOLIDE; ANTI HUMAN IMMUNODEFICIENCY VIRUS AGENT; DEHYDROANDROGRAPHOLIDE; UNCLASSIFIED DRUG;

ANTI HUMAN IMMUNODEFICIENCY VIRUS ACTIVITY; ANTIVIRAL ACTIVITY; ARTICLE; DRUG POTENCY; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; IN VITRO STUDY; NONHUMAN; PRIORITY JOURNAL;

ANTI-HIV AGENTS; CELL LINE; DITERPENES; HUMANS; MICROBIAL SENSITIVITY TESTS; MOLECULAR STRUCTURE; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84864606607     PISSN: 03656233     EISSN: 15214184     Source Type: Journal    
DOI: 10.1002/ardp.201200008     Document Type: Article

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