Transdermal iontophoresis of ranitidine: An opportunity in paediatric drug therapy

International Journal of Pharmaceutics

Volumn 435, Issue 1, 2012, Pages 27-32

  Djabri, Asma ^a   Guy, Richard H ^a   Delgado Charro, M Begoña ^a  

^a University of Bath   (United Kingdom)

Author keywords

Iontophoresis; Paediatric drug delivery; Ranitidine; Topical gels; Transdermal drug delivery

Indexed keywords

ELECTROLYTE; POLOXAMER; RANITIDINE;

ANIMAL TISSUE; AQUEOUS SOLUTION; ARTICLE; CONDUCTANCE; CONTROLLED STUDY; DRUG DELIVERY SYSTEM; DRUG PENETRATION; DRUG TISSUE LEVEL; IN VITRO STUDY; IONTOPHORESIS; NONHUMAN; PH; PRIORITY JOURNAL; VISCOSITY;

ADMINISTRATION, CUTANEOUS; ANIMALS; CHILD; DRUG DELIVERY SYSTEMS; ELECTRIC CONDUCTIVITY; GELS; HUMANS; IONTOPHORESIS; PERMEABILITY; PHARMACEUTICAL VEHICLES; RANITIDINE; SWINE; VISCOSITY;

EID: 84864282593     PISSN: 03785173     EISSN: 18733476     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2012.03.006     Document Type: Article

References (34)

1. M. Al-Khalili, V.M. Meidan, and B.B. Michniak Iontophoretic transdermal delivery of buspirone hydrochloride in hairless mouse skin AAPS PharmSci 5 2003 E14
2. J.L. Blumer, F.C. Rothstein, B.S. Kaplan, T.S. Yamashita, F.N. Eshelman, C.M. Myers, and M.D. Reed Pharmacokinetic determination of ranitidine pharmacodynamics in pediatric ulcer disease J. Pediatr. 107 1985 301 306 (Pubitemid 15241939)
3. C. Booth, and D. Attwood Effects of block architecture and composition on the association properties of poly(oxyalkylene) copolymers in aqueous solution Macromol. Rapid Commun. 21 2000 501 527
4. H.G. Brittain Profiles of Drug Substances, Excipients and Related Methodology vol. 33 2007 Academic Press London
5. R.R. Burnette, and B. Ongpipattanakul Characterization of the permselective properties of excised human skin during iontophoresis J. Pharm. Sci. 76 1987 765 773
6. A. Cabana, A. AitKadi, and J. Juhasz Study of the gelation process of polyethylene oxide(a) polypropylene oxide(b) polyethylene oxide(a) copolymer (poloxamer 407) aqueous solutions J. Colloid Interf. Sci. 190 1997 307 312 (Pubitemid 27470860)
7. J.H. Collett Monographs poloxamer R.C. Rowe, J. Sheskey, S.C. Owen, Handbook of Pharmaceutical Excipients 2006 Pharmaceutical Press; American Pharmacists Association London 535
8. J.J. Escobar-Chavez, M. Lopez-Cervantes, A. Naik, Y.N. Kalia, D. Quintanar-Guerrero, and A. Ganem-Quintanar Applications of thermo-reversible pluronic f-127 gels in pharmaceutical formulations J. Pharm. Pharm. Sci. 9 2006 339 358 (Pubitemid 46655458)
9. J.Y. Fang, K.C. Sung, J.J. Wang, C.C. Chu, and K.T. Chen The effects of iontophoresis and electroporation on transdermal delivery of buprenorphine from solutions and hydrogels J. Pharm. Pharmacol. 54 2002 1329 1337 (Pubitemid 35174177)
10. D.C. Garg, D.J. Weidler, and F.N. Eshelman Ranitidine bioavailability and kinetics in normal male subjects Clin. Pharm. Ther. 33 1983 445 452 (Pubitemid 13093763)
11. J.W. Goodwin, and R.W. Hughes Rheology for Chemists: An Introduction 2nd ed. 2008 RSC Publishing Cambridge p. 264
12. P. Green, B. Shroot, F. Bernard, W.R. Pilgrim, and R.H. Guy In vitro and in vivo iontophoresis of a tripeptide across nude rat skin J. Control. Release 20 1992 209 217
13. S.K. Gupta, S. Kumar, S. Bolton, C.R. Behl, and A.W. Malick Effect of chemical enhancers and conducting gels on iontophoretic transdermal delivery of cromolyn sodium J. Control. Release 31 1994 229 236 (Pubitemid 24301363)
14. A. Kim, P.G. Green, G. Rao, and R.H. Guy Convective solvent flow across the skin during iontophoresis Pharm. Res. 10 1993 1315 1320 (Pubitemid 23261832)
15. H. Kuhn, H.-D. Försterling, and D.H. Waldeck Principles of Physical Chemistry 2nd ed. 2008 Wiley Hoboken, NJ p. 120
16. R.A. Lugo, A.M. Harrison, J. Cash, J. Sweeley, and D.D. Vernon Pharmacokinetics and pharmacodynamics of ranitidine in critically ill children Crit. Care Med. 29 2001 759 764 (Pubitemid 32299713)
17. A. Luzardo-Alvarez, M. Rodriguez-Fernandez, J. Blanco-Mendez, R.H. Guy, and M.B. Delgado-Charro Iontophoretic permselectivity of mammalian skin: characterization of hairless mouse and porcine membrane models Pharm. Res. 15 1998 984 987 (Pubitemid 28356911)
18. J. Martin British National Formulary for Children revised ed. 2008 BMJ Group, RPS Publishing, and RCPCH Publications London 944
19. C.W. Macosko Rheology: Principles, Measurements, and Applications 1994 VCH Cambridge p. 550
20. A. Malkin Rheology Fundamentals 1994 ChemTec Ontario p. 324
21. D. Marro, R.H. Guy, and M.B. Delgado-Charro Characterization of the iontophoretic permselectivity properties of human and pig skin J. Control. Release 70 2001 213 217 (Pubitemid 32144805)
22. A.C. Moffat, M.D. Osselton, and B. Widdop Clarke's Analysis of Drugs and Poisons: In Pharmaceuticals, Body Fluids and Postmortem Material 3rd ed. 2004 Pharmaceutical Press London
23. C.Y. Oo, R.J. Kuhn, N. Desai, and P.J. Mcnamara Active-transport of cimetidine into human-milk Clin. Pharm. Ther. 58 1995 548 555
24. R.V. Padmanabhan, J.B. Phipps, G.A. Lattin, and R.J. Sawchuk In vitro and in vivo evaluation of transdermal iontophoretic delivery of hydromorphone J. Control. Release 11 1990 123 135 (Pubitemid 20070091)
25. S.R. Patel, H. Zhong, A. Sharma, and Y.N. Kalia In vitro and in vivo evaluation of the transdermal iontophoretic delivery of sumatriptan succinate Eur. J. Pharm. Biopharm. 66 2007 296 301 (Pubitemid 46661905)
26. J.B. Phipps, and J.R. Gyory Transdermal ion migration Adv. Drug Deliv. Rev. 9 1992 137 176
27. P. Santi, and R.H. Guy Reverse iontophoresis - parameters determining electroosmotic flow. 1. pH and ionic strength J. Control. Release 38 1996 159 165 (Pubitemid 26096660)
28. I.R. Schmolka Artificial skin. I. Preparation and properties of pluronic F-127 gels for treatment of burns J. Biomed. Mater. Res. 6 1972 571 582
29. A. Sieg, R.H. Guy, and M.B. Delgado-Charro Electroosmosis in transdermal iontophoresis: implications for noninvasive and calibration-free glucose monitoring Biophys. J. 87 2004 3344 3350 (Pubitemid 40468589)
30. P. Singh, S. Boniello, P. Liu, and S. Dinh Transdermal iontophoretic delivery of methylphenidate HCl in vitro Int. J. Pharm. 178 1999 121 128 (Pubitemid 29074414)
31. S.F. Taveira, A. Nomizo, and R.F. Lopez Effect of the iontophoresis of a chitosan gel on doxorubicin skin penetration and cytotoxicity J. Control. Release 134 2009 35 40
32. R. Van der Geest, M. Danhof, and H.E. Bodde Iontophoretic delivery of apomorphine. I: in vitro optimization and validation Pharm. Res. 14 1997 1798 1803
33. A.M. Vanhecken, T.B. Tjandramaga, A. Mullie, R. Verbesselt, and P.J. Deschepper Ranitidine - single dose pharmacokinetics and absolute bioavailability in man Brit. J. Clin. Pharm. 14 1982 195 200 (Pubitemid 13141876)
34. L. Wearley, L. Jue-Chen, and Y.W. Chien Iontophoresis-facilitated transdermal delivery of verapamil. 1. In vitro evaluation and mechanistic studies J. Control. Release 8 1989 237 250 (Pubitemid 19099002)