Contribution of indazolinone tautomers to kinase activity

Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 14, 2012, Pages 4502-4505

  Vasudevan, Anil ^a   Verzal, Mary K ^a   Villamil, Clara I ^a   Stewart, Kent D ^a   Abad Zapatero, Cele ^a   Oie, Tetsuro ^a   Djuric, Stevan W ^a  

^a ABBOTT LABORATORIES   (United States)

Author keywords

Indazolinones; Kdr; Kinase inhibitors; Tautomers

Indexed keywords

INDAZOLE DERIVATIVE; INDAZOLINONE DERIVATIVE; PROTEIN KINASE INHIBITOR; UNCLASSIFIED DRUG;

DRUG DESIGN; DRUG POTENCY; DRUG SYNTHESIS; ENZYME ACTIVITY; HYDROGEN BOND; QUANTUM MECHANICS; REVIEW; STEREOISOMERISM; TAUTOMER;

EID: 84863456422     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2012.06.009     Document Type: Article

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