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Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 6, 2012, Pages 2235-2238

Novel 5-substituted 1H-tetrazoles as cyclooxygenase-2 (COX-2) inhibitors

(4) Al Hourani, Baker Jawabrah a,b Sharma, Sai Kiran a Suresh, Mavanur a Wuest, Frank a

a UNIVERSITY OF ALBERTA (Canada)

b AMERICAN UNIVERSITY OF MADABA (Jordan)

Author keywords

5 Substituted 1H tetrazoles; COX 2 inhibitors; Cyclooxygenase

Indexed keywords

1 [4 (AMINOSULFONYL)PHENYL] 5 (4 CHLOROPHENYL) 1H TETRAZOLE; 1 [4 (AMINOSULFONYL)PHENYL] 5 (4 DIMETHYLAMINOPHENYL) 1H TETRAZOLE; 1 [4 (AMINOSULFONYL)PHENYL] 5 (4 FLUOROPHENYL) 1H TETRAZOLE; 1 [4 (AMINOSULFONYL)PHENYL] 5 (4 METHOXYPHENYL) 1H TETRAZOLE; 1 [4 (AMINOSULFONYL)PHENYL] 5 (4 NITROPHENYL) 1H TETRAZOLE; 1 [4 (AMINOSULFONYL)PHENYL] 5 (4 TRIFLUOROMETHYLPHENYL) 1H TETRAZOLE; 1 [4 (AMINOSULFONYL)PHENYL] 5 4 TOLYL 1H TETRAZOLE; 1 [4 (AMINOSULFONYL)PHENYL] 5 PHENYL 1H TETRAZOLE; 1 [4 (METHYLSULFONYL)PHENYL] 5 (4 DIMETHYLAMINOPHENYL)1H TETRAZOLE; 1 [4 (METHYLSULFONYL)PHENYL] 5 (4 NITROPHENYL) 1H TETRAZOLE; 1 [4 (METHYLSULFONYL)PHENYL] 5 PHENYL 1H TETRAZOLE; 4 (METHYLSULFONYL)PHENYL] 5 4 TOLYL 1H TETRAZOLE; 5 (4 FLUOROPHENYL) 1 [4 (METHYLSULFONYL)PHENYL] 1H TETRAZOLE; 5 (4 METHOXYPHENYL) 1 [4 (METHYLSULFONYL)PHENYL] 1H TETRAZOLE; CELECOXIB; CYCLOOXYGENASE 1; CYCLOOXYGENASE 2; CYCLOOXYGENASE 2 INHIBITOR; TETRAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; DRUG POTENCY; ENZYME ASSAY; ENZYME INHIBITION; IC 50; SUBSTITUTION REACTION;

AMIDES; BIOLOGICAL ASSAY; CHLORIDES; CYCLOOXYGENASE 2; CYCLOOXYGENASE 2 INHIBITORS; DRUG DESIGN; HUMANS; MODELS, MOLECULAR; PYRAZOLES; SILICON COMPOUNDS; SODIUM AZIDE; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONAMIDES; TETRAZOLES;

EID: 84863397494 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2012.01.093 Document Type: Article

Times cited : (39)

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