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Volumn 6, Issue 1, 1996, Pages 87-92

Synthesis and biological evaluation of 2,3-diarylthiophenes as selective Cox-2 inhibitors. Part II: Replacing the heterocycle

Author keywords

[No Author keywords available]

Indexed keywords

1,2,3 THIADIAZOLE DERIVATIVE; 5 BROMO 2 (4 FLUOROPHENYL) 3 (4 METHYLSULFONYLPHENYL)THIOPHENE; CYCLOOXYGENASE 2; INDOMETACIN; ISOENZYME; PROSTAGLANDIN SYNTHASE; PROSTAGLANDIN SYNTHASE INHIBITOR; THIADIAZOLE DERIVATIVE; THIOPHENE DERIVATIVE; UNCLASSIFIED DRUG;

EID: 0030029368     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/0960-894X(95)00564-A     Document Type: Article
Times cited : (59)

References (23)
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    • Hla, T.; Neilson, K. Proc. Natl. Acad. Sci. U.S.A. 1992, 89, 7384; Xie, W.; Chipman, J.G.; Robertson, D. L.; Erickson, R. L.; Simmons, D. L. Proc. Natl. Acad. Sci. U.S.A. 1991, 88, 2692; Kujubu, D. A.; Fletcher, B. S.; Varnum, B. C.; Lim, R.W.; Herschman, H. R. J. Biol. Chem. 1991, 266, 12866.
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    • WO 95/00501
    • Ducharme, Y.; Gauthier, J. Y.; Prasit, P.; Leblanc, Y.; Wang, Z.; Léger, S.; Thérien, M. World Patent Application, 1995, WO 95/00501. For a related study with indenes and benzofurans, see: Huang, H. C.; Chamberlain, T. S.; Seibert, K.; Koboldt, C. M.; Isakson, P. C.; Reitz, D. B. Bioorg. Med. Chem. Lett. 1995, 5, 2377. For a study of pyrroles, see: Wilkerson, W. W.; Copeland, R. A.; Covington, M.; Trzaskos, J. M. J. Med. Chem. 1995, 38, 3895.
    • (1995) World Patent Application
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    • Ducharme, Y.; Gauthier, J. Y.; Prasit, P.; Leblanc, Y.; Wang, Z.; Léger, S.; Thérien, M. World Patent Application, 1995, WO 95/00501. For a related study with indenes and benzofurans, see: Huang, H. C.; Chamberlain, T. S.; Seibert, K.; Koboldt, C. M.; Isakson, P. C.; Reitz, D. B. Bioorg. Med. Chem. Lett. 1995, 5, 2377. For a study of pyrroles, see: Wilkerson, W. W.; Copeland, R. A.; Covington, M.; Trzaskos, J. M. J. Med. Chem. 1995, 38, 3895.
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    • Ducharme, Y.; Gauthier, J. Y.; Prasit, P.; Leblanc, Y.; Wang, Z.; Léger, S.; Thérien, M. World Patent Application, 1995, WO 95/00501. For a related study with indenes and benzofurans, see: Huang, H. C.; Chamberlain, T. S.; Seibert, K.; Koboldt, C. M.; Isakson, P. C.; Reitz, D. B. Bioorg. Med. Chem. Lett. 1995, 5, 2377. For a study of pyrroles, see: Wilkerson, W. W.; Copeland, R. A.; Covington, M.; Trzaskos, J. M. J. Med. Chem. 1995, 38, 3895.
    • (1995) J. Med. Chem. , vol.38 , pp. 3895
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* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.