Preparation of evodiamine solid dispersions and its pharmacokinetics

Indian Journal of Pharmaceutical Sciences

Volumn 73, Issue 3, 2011, Pages 276-281

  Xu, H ^a,b   Zhang, T ^a   Yang, H ^b   Xiao, X ^a,c   Bian, Y ^c   Si, D ^a   Liu, C ^a  

^a TIANJIN INSTITUTE OF PHARMACEUTICAL RESEARCH   (China)

^b INSTITUTE OF CHINESE MATERIA MEDICA   (China)

^c TIANJIN UNIVERSITY OF TRADITIONAL CHINESE MEDICINE   (China)

Author keywords

Dissolution rate; evodiamine; pharmacokinetics; solid dispersions; X ray powder diffraction

Indexed keywords

EVODIAMINE; POVIDONE;

ARTICLE; DOG; DRUG ABSORPTION; DRUG CAPSULE; DRUG ISOLATION; DRUG SOLUBILITY; EVODIA; SINGLE DRUG DOSE; X RAY POWDER DIFFRACTION;

EID: 84863284796     PISSN: 0250474X     EISSN: 19983743     Source Type: Journal    
DOI: 10.4103/0250-474X.93511     Document Type: Article

References (31)

1. Pharmacopoeia of People's Republic of China, (in Chinese). Vol. 1. Beijing: Chemical Industry Press; 2002.
2. Lin H, Tsai SC, Chen JJ, Chiao YC, Wang SW, Wang GJ, et al. Effect of evodiamine on the secretion of testosterone in rat testicular interstitial cells. Metabolism 1999;48:1532-5.
3. Yoshizumi M, Houchi H, Ishimura Y, Hirose M, Kitagawa T, Tsuchiya K, et al. Effect of evodiamine on catecholamine secretion from bovine adrenal medulla. J Med Invest 1997;44:79-82. (Pubitemid 127495237)
4. Kobayashi Y. The nociceptive and anti-nociceptive effects of evodiamine from fruits of Evodia rutaecarpa in mice. Planta Med 2003;69:425-8. (Pubitemid 36774182)
5. Chiou WF, Sung YJ, Liao JF, Shum AY, Chen CF. Inhibitory effect of dehydroevodiamine and evodiamine on nitric oxide production in cultured murine macrophages. J Nat Prod 1997;60:708-11. (Pubitemid 27318419)
6. Kobayashi Y, Nakano Y, Kizaki M, Hoshikuma K, Yokoo Y, Kamiya T. Capsaicin-like anti-obese activities of evodiamine from fruits of Evodia rutaecarpa, a vanilloid receptor agonist. Planta Med 2001;67:628-33. (Pubitemid 32929573)
7. Chiou WF, Chou CJ, Shum AY, Chen CF. The vasorelaxant effect of evodiamine in rat isolated mesenteric arteries: Mode of action. Eur J Pharmacol 1992;215:277-83.
8. Tsai TH, Lee TF, Chen CF, Wang LC. Thermoregulatory effects of alkaloids isolated from Wu-chu-yu in afebrile and febrile rats. Pharmacol Biochem Behav 1995;50:293-8.
9. King CL, Kong YC, Wong NS, Yeung HW, Fong HH, Sankawa U. Uterotonic effect of Evodia rutaecarpa alkaloids. J Nat Prod 1980;43:577-82.
10. Ogasawara M, Matsubara T, Suzuki H. Screening of natural compounds for inhibitory activity on colon cancer cell migration. Biol Pharm Bull 2001;24:720-3. (Pubitemid 32586670)
11. Liao CH, Pan SL, Guh JH, Chang YL, Pai HC, Lin CH, et al. Antitumor mechanism of evodiamine, a constituent from Chinese herb Evodiae fructus, in human multiple-drug resistant breast cancer NCI/ADR-RES cells in vitro and in vivo. Carcinogenesis 2005;26:968-75.
12. Kan SF, Yu CH, Pu HF, Hsu JM, Chen MJ, Wang PS. Anti-proliferative effects of evodiamine on human prostate cancer cell lines DU145 and PC3. J Cell Biochem 2007;101:44-56. (Pubitemid 46652571)
13. Huang DM, Guh JH, Huang YT, Chueh SC, Chiang PC, Teng CM. Induction of mitotic arrest and apoptosis in human prostate cancer PC-3 cells by evodiamine. J Urol 2005;173:256-61.
14. Kang SF, Huang WJ, Lin LC, Wang PS. Inhibitory effects of evodiamine on the growth of human prostate cancer cell line LNCaP. Int J Cancer 2004;110:641-51. (Pubitemid 38746021)
15. Lee TJ, Kim EJ, Kim S, Jung EM, Park JW, Jeong SH, et al. Caspase-dependent and caspase-independent apoptosis induced by evodiamine in human eukemic U937 cells. Mol Cancer Ther 2006;5:2398-407. (Pubitemid 44530477)
16. Huang YC, Guh JH, Teng CM. Induction of mitotic arrest and apoptosis by evodiamine in human leukemic T-lymphocytes. Life Sci 2004;75:35-49.
17. Wang C, Wang MW, Tashiro S, Onodera S, Ikejima T. Evodiamine induced human melanoma A375-S2 cell death partially through interleukin 1 mediated pathway. Biol Pharm Bull 2005;28:984-9. (Pubitemid 40880301)
18. Fei XF, Wang BX, Li TJ, Tashiro S, Minami M, Xing DJ, et al. Evodiamine, a constituent of Evodiae fructus, induces anti-proliferating effects in tumor cells. Cancer Sci 2003;94:92-8. (Pubitemid 36575865)
19. Ogasawara M, Matsubara T, Suzuki H. Inhibitory effects of evodiamine on in vitro invasion and experimental lung metastasis of murine colon cancer cells. Biol Pharm Bull 2001;24:917-20. (Pubitemid 32750318)
20. Ogasawara M, Matsubara T, Takahashi S, Saiki I, Suzuki H. Anti-invasive and metastatic activities of evodiamine. Biol Pharm Bull 2002;25:1491-3. (Pubitemid 39663174)
21. Shyr MH, Lin LC, Lin TY, Tsai TY. Determination and pharmacokinetics of evodiamine in the plasma and feces of conscious rats. Anal Chim Acta 2006;3:16-21.
22. Yamashita K, Nakate T, Okimoto K, Ohike A, Tokunaga Y, Ibuki R, et al. Establishment of new preparation method for solid, dispersion formulation of tacrolimus. Int J Pharm 2003;267:79-91. (Pubitemid 37352952)
23. Chiou WL, Riegelman S. Pharmaceutical applications of solid dispersions. J Pharm Sci 1971;60:1281-302.
24. Ford JL. The current status of solid dispersions. Pharm Acta Helv 1986;61:69-88. (Pubitemid 16134014)
25. Craig DQ. Polyethylene glycols and drug release. Drug Dev Ind Pharm 1990;16:2501-27.
26. Serajuddin AT. Solid dispersions of poorly water-soluble drugs: Early promises, subsequent problems, and recent breakthroughs. J Pharm Sci 1999;88:1058-66.
27. Craig DQ. The mechanisms of drug release from solid dispersions in water-soluble polymers. Int J Pharm 2002;231:131-44. (Pubitemid 34033673)
28. Craig C, Duncan QM. The mechanisms of drug release from solid dispersions in water soluble polymers. Int J Pharm 2002;32:213-6.
29. Pandit JK, Khakurel BK. In vitro and in vivo evaluation of some fast release dosage forms of hydrochlorothiazide. Drug Dev Ind Pharm 1984;10:1709-24. (Pubitemid 15127392)
30. Leuner C, Dressman J. Improving drug solubility for oral delivery using solid dispersions. Eur J Pharm Biopharm 2000;50:47-60. (Pubitemid 30326688)
31. Chauhan B, Shimpi S, Paradkar A. Preparation and evaluation of libenclamide-polyglycolized glycerides solid dispersions with silicon dioxide by spray drying technique. Eur J Pharm Sci 2005;26:219-30. (Pubitemid 41169805)