G protein-coupled receptor biased agonism: Development towards future selective therapeutics

Mini-Reviews in Medicinal Chemistry

Volumn 12, Issue 9, 2012, Pages 803-

  Maudsley, Stuart ^a  

^a NATIONAL INSTITUTE ON AGING   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ANGIOTENSIN 1 RECEPTOR; G PROTEIN COUPLED RECEPTOR; GONADORELIN RECEPTOR; PARATHYROID HORMONE RECEPTOR;

DRUG TARGETING; EDITORIAL; PROTEIN CONFORMATION; SIGNAL TRANSDUCTION;

HUMANS; MOLECULAR TARGETED THERAPY; PROTEIN CONFORMATION; RECEPTORS, G-PROTEIN-COUPLED;

EID: 84862881048     PISSN: 13895575     EISSN: 18755607     Source Type: Journal    
DOI: 10.2174/138955712800959161     Document Type: Editorial

References (5)

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2. Gesty-Palmer, D.; Luttrell, L.M. Heptahelical terpsichory. Who calls the tune? J. Recept. Signal Transduct. Res. 2008, 28(1-2), 39-58.
3. Maudsley, S.; Martin, B.; Luttrell, L.M. G protein-coupled receptor signaling complexity in neuronal tissue: implications for novel therapeutics. Curr. Alzheimer Res. 2007, 4(1), 3-19.
4. Maudsley, S.; Martin, B.; Luttrell, L.M. The origins of diversity and specificity in g protein-coupled receptor signaling. J. Pharmacol. Exp. Ther. 2005, 314(2), 485-494.
5. Maurice, P.; Guillaume, J.L.; Benleulmi-Chaachoua, A.; Daulat, A.M.; Kamal, M.; Jockers, R. GPCR-Interacting Proteins, Major Players of GPCR Function. Adv. Pharmacol. 2011, 62, 349-380.