Biased agonism of the angiotensin II type 1 receptor

Mini-Reviews in Medicinal Chemistry

Volumn 12, Issue 9, 2012, Pages 812-816

  Godin, C M ^a   Ferguson, S S G ^a  

^a ROBARTS RESEARCH INSTITUTE   (Canada)

Author keywords

Angiotensin II; Biased agonism; G protein; GPCR; SII

Indexed keywords

ANGIOTENSIN 1 RECEPTOR; ANGIOTENSIN II; ANGIOTENSIN II [1 SARCOSINE 8 ISOLEUCINE]; BETA ARRESTIN; CALPASTATIN; EPIDERMAL GROWTH FACTOR RECEPTOR; G PROTEIN COUPLED RECEPTOR; LOSARTAN; MITOGEN ACTIVATED PROTEIN KINASE; MITOGEN ACTIVATED PROTEIN KINASE 1; MITOGEN ACTIVATED PROTEIN KINASE 3; PROTEIN C JUN; PROTEIN KINASE D;

ARTICLE; BINDING AFFINITY; CARDIOVASCULAR DISEASE; CELL STRAIN HEK293; ENDOCYTOSIS; GENE CONTROL; GENETIC TRANSCRIPTION; HUMAN; INTERNALIZATION; INTRACELLULAR SIGNALING; ISOTOPE LABELING; MICROARRAY ANALYSIS; MYOTATIC REFLEX; PROTEIN BINDING; PROTEIN EXPRESSION; PROTEIN PHOSPHORYLATION;

1-SARCOSINE-8-ISOLEUCINE ANGIOTENSIN II; ANGIOTENSIN II; ANGIOTENSIN II TYPE 1 RECEPTOR BLOCKERS; ARRESTINS; HEK293 CELLS; HUMANS; LIGANDS; LOSARTAN; MAP KINASE SIGNALING SYSTEM; PROTEIN CONFORMATION; RECEPTOR, ANGIOTENSIN, TYPE 1; STRESS, MECHANICAL;

EID: 84862864947     PISSN: 13895575     EISSN: 18755607     Source Type: Journal    
DOI: 10.2174/138955712800959134     Document Type: Article

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