Synthesis and in vitro antiplasmodial activities of fluoroquinolone analogs

European Journal of Medicinal Chemistry

Volumn 51, Issue , 2012, Pages 52-59

  Dixit, Sandeep K ^a   Mishra, Nidhi ^a   Sharma, Manish ^a   Singh, Shailja ^a   Agarwal, Alka ^b   Awasthi, Satish K ^a   Bhasin, V K ^a  

^a UNIVERSITY OF DELHI   (India)

^b BANARAS HINDU UNIVERSITY   (India)

Author keywords

Antimalarial activity; Fluoroquinolones; In vitro; Plasmodium falciparum

Indexed keywords

CHLORO 6 FLUORO 4 OXO 1 (1H [1,2,3]TRIAZOL 4 YLMETHYL) 1,4 DIHYDROQUINOLINE 3 CARBOXYLIC ACID ETHYL ESTER; CIPROFLOXACIN; QUINOLINE DERIVED ANTIINFECTIVE AGENT; UNCLASSIFIED DRUG; ANTIMALARIAL AGENT; QUINOLONE DERIVATIVE; TRIAZOLE DERIVATIVE;

ALKYLATION; ANTIMALARIAL ACTIVITY; ARTICLE; CLICK CHEMISTRY; CONTROLLED STUDY; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; IC 50; IN VITRO STUDY; NONHUMAN; PLASMODIUM; PLASMODIUM FALCIPARUM; CELL STRAIN HEK293; CELL SURVIVAL; CHEMISTRY; DRUG EFFECT; HUMAN; SYNTHESIS;

ANTIMALARIALS; CELL SURVIVAL; CHEMISTRY TECHNIQUES, SYNTHETIC; FLUOROQUINOLONES; HEK293 CELLS; HUMANS; INHIBITORY CONCENTRATION 50; PLASMODIUM FALCIPARUM; TRIAZOLES;

EID: 84862824408     PISSN: 02235234     EISSN: 17683254     Source Type: Journal    
DOI: 10.1016/j.ejmech.2012.02.006     Document Type: Article

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