Microstructural investigation to the controlled release kinetics of monolith osmotic pump tablets via synchrotron radiation X-ray microtomography

International Journal of Pharmaceutics

Volumn 427, Issue 2, 2012, Pages 270-275

  Li, Haiyan ^a   Yin, Xianzhen ^a   Ji, Junqiu ^b   Sun, Lixin ^c   Shao, Qun ^d   York, Peter ^d   Xiao, Tiqiao ^e   He, You ^e   Zhang, Jiwen ^a  

^a SHANGHAI INSTITUTE OF MATERIA MEDICA   (China)

^b Hefei Lifeon Medication Group   (China)

^c SHENYANG PHARMACEUTICAL UNIVERSITY   (China)

^d UNIVERSITY OF BRADFORD   (United Kingdom)

^e SHANGHAI INSTITUTE OF APPLIED PHYSICS   (China)

Author keywords

Drug release kinetics; Microtomography; Osmotic drug delivery system; Surface area; Synchrotron radiation X ray computed; Three dimensional reconstruction

Indexed keywords

FELODIPINE;

ARTICLE; CHEMICAL STRUCTURE; CONTROLLED RELEASE FORMULATION; DRUG DELIVERY SYSTEM; HYDRATION; MICRO-COMPUTED TOMOGRAPHY; MORPHOLOGY; OSMOTIC PUMP; PRIORITY JOURNAL; SURFACE PROPERTY; SYNCHROTRON RADIATION X RAY COMPUTED MICROTOMOGRAPHY; TABLET FORMULATION; THREE DIMENSIONAL IMAGING;

ALGORITHMS; CALCIUM CHANNEL BLOCKERS; DELAYED-ACTION PREPARATIONS; DRUG DELIVERY SYSTEMS; FELODIPINE; IMAGE PROCESSING, COMPUTER-ASSISTED; IMAGING, THREE-DIMENSIONAL; OSMOSIS; SOLUBILITY; SYNCHROTRONS; TABLETS; TOMOGRAPHY, X-RAY COMPUTED; X-RAY MICROTOMOGRAPHY;

EID: 84862820773     PISSN: 03785173     EISSN: 18733476     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2012.02.017     Document Type: Article

References (35)

1. M. Ansari, and F. Stepanek Formation of hollow core granules by fluid bed in situ melt granulation: modelling and experiments Int. J. Pharm. 321 2006 108 116
2. D. Bass, M. Prevo, and D. Waxman Gastrointestinal safety of an extended release, nondeformable, oral dosage form (OROS (R)) - a retrospective study Drug Saf. 25 2002 1021 1033
3. W. Charman, H. Chan, B. Finnin, and S. Charman Drug delivery: a key factor in realizing the full therapeutic potential of drugs Drug Dev. Res. 46 1999 316 327
4. G. Chauve, F. Raverielle, and R. Marchessault Comparative imaging of a slow release starch exciplent tablet: evidence of membrane formation Carbohydrate Polym. 70 2007 61 67
5. R. Conley, S. Gupta, and G. Sathyan Clinical spectrum of the osmotic-controlled release oral delivery system (OROS), an advanced oral delivery form Curr. Med. Res. Opin. 22 2006 1879 1892
6. T. Donath Quantitative X-ray Microtomography with Synchrotron Radiation 2007 GKSS-ForschungszentrumBibliothek Geesthacht pp. 1-221
7. R. Dwarakanadha, and D. Swarnalatha Recent advances in novel drug delivery systems Int. J. Pharm. Technol. Res. 2 2010 2025 2027
8. X. Fu, M. Dutt, A. Bentham, B. Hancock, R. Cameron, and J. Elliott Investigation of particle packing in model pharmaceutical powders using X ray microtomography and discrete element method Powder Technol. 167 2006 134 140
9. H. Gupta, D. Bhandari, and A. Sharma Recent trends in oral drug delivery: a review Recent Pat. Drug Deliv. Formul. 3 2009 162 173
10. R. Gupta, R. Gupta, P. Basniwal, and G. Rathore Osmotically controlled oral drug delivery systems: a review Int. J. Pharm. Technol. Res. 1 2009 269 275
11. B. Hancock, and M. Mullarney X-ray microtomography of solid dosage forms Pharm. Technol. 2 2005 92 100
12. E. Karakosta, P. Jenneson, R. Sear, and P. McDonald Observations of coarsening of air voids in a polymer-highly-soluble crystalline matrix during dissolution Phys. Rev. E74 2006 011504-1-011504-7
13. A. Kaushal, and S. Garg An update on osmotic drug delivery patents Pharm. Technol. 27 2003 38-40, 42-44, 9797
14. J. Kerc, S. Srcic, B. Kofler, and J. Smid-Korbar Molar solubility of felodipine in different aqueous systems Int. J. Pharm. 81 1992 R1 R4
15. W. Ketjinda, N. Sinchaipanid, P. Limsuwan, H. Leuenberger, and A. Mitrevej Development of push-pull osmotic tablets using Chitosan-Poly(Acrylic Acid) interpolymer complex as an osmopolymer A. A. P. S. Pharm. Sci. Tech. 12 2010 132 140
16. P. Kumar, and B. Mishra An overview of recent patents on oral osmotic drug delivery systems Recent Pat. Drug Deliv. Formul. 1 2007 236 255
17. L. Liu, G. Khang, J. Rhee, and H. Lee Monolithic osmotic tablet system for nifedipine delivery J. Control. Release 67 2000 309 322
18. E. Lu, Z. Jiang, Q. Zhang, and X. Jiang A water-insoluble drug monolithic osmotic tablet system utilizing gum Arabic as an osmotic, suspending and expanding agent J. Control. Release 92 2003 375 382
19. V. Malaterre, J. Ogorka, N. Loggia, and R. Gurny Oral osmotically driven systems: 30 years of development and clinical use Eur. J. Pharm. Biopharm. 73 2009 311 323
20. E. Mehuys, and C. Vervaet Oral controlled release dosage forms J. Pharm. Belg. 2 2010 34 38
21. A. Nokhodchi, M. Momin, J. Shokri, M. Shahsavari, and P. Rashidi Factors affecting the release of nifedipine from a swellable elementary osmotic pump Drug Deliv. 15 2008 43 48
22. S. Rose, and J. Nelson A continuous long term injector Aust. J. Exp. Bio. Med. Sci. 33 1955 415 420
23. G. Santus, and R. Baker Osmotic drug delivery: a review of the patent literature J. Control. Release 35 1995 1 21
24. B. Singh Modified-release solid formulations for colonic delivery Recent Pat. Drug Deliv. Formul. 1 2007 53 63
25. I. Sinka, S. Burch, J. Tweed, and J. Cunningham Measurement of density variations in tablets using X-ray computed tomography Int. J. Pharm. 271 2004 215 224
26. Y. Tokudome, H. Ohshima, and M. Otsuka Non-invasive and rapid analysis for observation of internal structure of press-coated tablet using X-ray computed tomography Drug Dev. Ind. Pharm. 35 2009 678 682
27. D. Traini, G. Loretit, A. Jones, and P. Young X-ray computed microtomography for the study of modified release systems Micros. Anal. 22 2008 13 17
28. R. Verma, S. Arora, and S. Garg Osmotic pumps in drug delivery Crit. Rev. Ther. Drug Carrier Syst. 21 2004 477 520
29. R. Verma, D. Krishna, and S. Garg Formulation aspects in the development of osmotically controlled oral drug delivery systems J. Control. Release 79 2002 7 27
30. R. Verma, B. Mishra, and S. Garg Osmotically controlled oral drug delivery Drug Dev. Ind. Pharm. 26 2000 695 708
31. Y. Wang, D. Wertheim, A. Jones, and A. Coombes Micro-CT in drug delivery Eur. J. Pharm. Biopharm. 74 2010 41 49
32. Y. Wang, D. Wertheim, A. Jones, H. Chang, and A. Coombes Micro-CT analysis of matrix-type drug delivery devices and correlation with protein release behaviour J. Pharm. Sci. 99 2010 2854 2862
33. H. Wen, and K. Park Oral Controlled Release Formulation Design and Drug Delivery, Theory to Practice 2010 Wiley
34. P. Young, K. Nguyen, A. Jones, and D. Traini Microstructural analysis of porous composite materials: dynamic imaging of drug dissolution and diffusion through porous matrices A. A. P. S. J. 10 2008 560 564
35. J. Zeitler, and L. Gladden In vitro tomography and non-destructive imaging at depth of pharmaceutical solid dosage forms Eur. J. Pharm. Biopharm. 71 2009 2 22