A uronic acid analogue of isofagomine lactam as a nanomolar glucuronidase inhibitor

Tetrahedron Letters

Volumn 53, Issue 16, 2012, Pages 2045-2047

  Lindbäck, Emil ^a   Zhou, You ^a   López, Óscar ^b   Fernández Bolaños, José G ^b   Pedersen, Christian Marcus ^a   Bols, Mikael ^a  

^a UNIVERSITY OF COPENHAGEN   (Denmark)

^b UNIVERSITY OF SEVILLE   (Spain)

Author keywords

Glucuronidase; Glucuronidase inhibitor; (2,2,6,6 Tetramethyl piperidin 1 yl)oxyl; Bisacetoxyiodobenzene; Selective oxidation

Indexed keywords

5 CARBOXYLIC ACID 3,4 DIHYDROXYPIPERIDIN 2 ONE; BENZENE DERIVATIVE; BETA GLUCURONIDASE; BETA GLUCURONIDASE INHIBITOR; BISACETOXYIODOBENZENE; ENZYME INHIBITOR; GLUCURONIC ACID; ISOFAGOMINE LACTAM URONIC ACID; UNCLASSIFIED DRUG; URONIC 1 DEOXYNOJIRIMYCIN; URONIC ACID;

ARTICLE; CARBON NUCLEAR MAGNETIC RESONANCE; CATALYSIS; CATTLE; CHEMICAL REACTION; CHEMICAL STRUCTURE; ENZYME ACTIVITY; ENZYME INHIBITION; LIVER; MASS SPECTROMETRY; NONHUMAN; OXIDATION; PROTON NUCLEAR MAGNETIC RESONANCE; SYNTHESIS;

BOVINAE;

EID: 84862815653     PISSN: 00404039     EISSN: 18733581     Source Type: Journal    
DOI: 10.1016/j.tetlet.2012.02.009     Document Type: Article

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