Comparative study of conventional and microwave-assisted synthesis of some Schiff bases and their potential as antimicrobial agents

Medicinal Chemistry Research

Volumn 21, Issue 6, 2012, Pages 844-852

  Pandey, Vikas ^a   Chawla, Viney ^a   Saraf, Shailendra K ^a  

^a Northern India Engineering College   (India)

Author keywords

Antibacterial; Antifungal; Green chemistry; Microwave assisted synthesis; Schiff base

Indexed keywords

(3 METHYLPYRIDIN 2 YL)NAPHTHALEN 1 YLMETHYLENE AMINE; (4 CHLOROPHENYL)NAPHTHALEN 1 YLMETHYLENE AMINE; (4 CHLOROPHENYL)THIOPHEN 2 YLMETHYLENE AMINE; (5 METHYL 5H ISOXAZOL 2 YL)NAPHTHALEN 1 YLMETHYLENE AMINE; 3 [(1H [1,2,4]TRIAZOL 3 YLIMINO)METHYL]CHROMEN 4 ONE; 3 [(4 CHLOROPHENYLIMINO)METHYL]CHROMEN 4 ONE; ANTIINFECTIVE AGENT; FURAN 2 YLMETHYLENE (1H [1,2,4]TRIAZOL 3 YL)AMINE; NAPHTHALEN 1 YLMETHYLENE (1H [1,2,4]TRIAZOL 3 YL)AMINE; NAPHTHALEN 1 YLMETHYLENE PYRIDIN 2 YLAMINE; SCHIFF BASE; THIOPHEN 2 YLMETHYLENE (1H [1,2,4]TRIAZOL 3 YL)AMINE; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ARTICLE; ASPERGILLUS NIGER; BACILLUS PUMILUS; BACILLUS SUBTILIS; COMPARATIVE STUDY; DRUG SYNTHESIS; ESCHERICHIA COLI; INFRARED SPECTROSCOPY; MASS SPECTROMETRY; MICROCOCCUS LUTEUS; MICROWAVE RADIATION; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; PENICILLIUM CHRYSOGENUM; PROTON NUCLEAR MAGNETIC RESONANCE; PSEUDOMONAS AERUGINOSA; PSEUDOMONAS FLUORESCENS;

EID: 84861883795     PISSN: 10542523     EISSN: 15548120     Source Type: Journal    
DOI: 10.1007/s00044-011-9592-6     Document Type: Article

References (22)

1. Andrews JM (2001) Determination of minimum inhibitory concentrations. J Antimicrob Chemother 48S:5-16
2. Bharti SK, Nath G, Tilak R, Singh SK (2010) Synthesis, anti-bacterial and anti-fungal activities of some novel Schiff bases containing 2,4-disubstituted thiazole ring. Eur J Med Chem 45:651-660
3. Biological assay, Indian Pharmacopoeia (1996), vol 2, Govt. of India, Delhi, pp A100-102
4. Burczyk A, Loupy A, Bogdal D, Petit A (2005) Improvement in the synthesis of metallophthalocyanines using microwave irradiation. Tetrahedron 61:179-188 (Pubitemid 39573416)
5. Byrnes RW, Mohan M, Antholine WE, Xu RX, Petering DH (1990) Oxidative stress induced by a copper-thiosemicarbazone complex. Biochemistry 29:7046-7053 (Pubitemid 20241151)
6. Clayden J, Greeves N, Warren S, Wothers P (2001) Organic chemistry, 1st edn. Oxford University Press Inc, New York, pp 1385-1387
7. Curini M, Epifano F, Maltese F, Marcotullio MC (2002) Novel chiral Schiff base ligands from amino acid amides and salicylaldehyde. Tetrahedron Lett 43:3821-3823 (Pubitemid 34463039)
8. Hodnett EM, Dunn WJ (1970) Structure-antitumor activity correlation of some Schiff bases. J Med Chem 13:768-770
9. Kamel MM, Ali HI, Anwar MM, Mohamed NA, Soliman AMM (2010) Synthesis, antitumour activity and molecular docking study of novel sulphonamide-Schiff's bases, thiazolidinones, benzothiazones and their C-nucleoside derivatives. Eur J Med Chem 45:572-580
10. Kosower EM, Miyadera T (1972) Glutathione.6. Probable mechanism of action of diazene antibiotics. J Med Chem 15:307-312
11. Lidstorm P, Tierney J, Wathey B, Westman J (2001) Microwave assisted organic synthesis-a review. Tetrahedron 57:9225-9283 (Pubitemid 33016768)
12. Liu MC, Lin TS, Sartorelli AC (1992) Synthesis and antitumor activity of amino derivatives of pyridine-2-carboxaldehyde thiosemicarbazone. J Med Chem 35:3672-3677
13. Loupy A (2002) Microwaves in organic synthesis. Wiley, Weinheim
14. Mladenova R, Ignatova M, Manolova N, Petrova T, Rashkov I (2002) Preparation, characterization and biological activity of Schiff base compounds derived from 8-hydoxy quinoline-2-carboxaldehyde and Jeffamines ED®. Eur Polym J 38:989-999 (Pubitemid 34200973)
15. Pannerselvam P, Nair RR, Vijayalakshmi G, Subramanian EH, Sridhar SK (2005) Synthesis of Schiff bases of 4-(4-aminophenyl)-morpholine as potential antimicrobial agents. Eur J Med Chem 40:225-229 (Pubitemid 40203164)
16. Sridhar SK, Saravanan M, Ramesh A (2001) Synthesis and antibacterial screening of hydrazones, Schiff and Mannich bases of hydrazone derivatives. Eur J Med Chem 36:615-625 (Pubitemid 32964732)
17. Tenorio RP, Carvalho CS, Pessanha CS, Delima JG (2005) Synthesis of thiosemicarbazone and 4-thiazolidinone derivatives and their in vitro anti-Toxoplasma gondii activity. Bioorg Med Chem Lett 15:2575-2578 (Pubitemid 40614991)
18. Varma RS, Dahiya R, Kumar S (1997) Clay catalyzed synthesis of imines and enamines under solvent-free conditions using microwave irradiation. Tetrahedron Lett 38:2039-2042 (Pubitemid 27117740)
19. Vass A, Dudas J, Varma RS (1999) Solvent-free synthesis of N-sulfonylimines using microwave irradiation. Tetrahedron Lett 40:4951-4954 (Pubitemid 29287340)
20. Walsh OM, Meegan MJ, Prendergast RM, Nakib TA (1996) Synthesis of 3-acetoxy-azetidin-2-ones and 3-hydoxy-azetidin-2-ones with antifungal and antibacterial activity. Eur J Med Chem 31:989-1000 (Pubitemid 26418443)
21. Yadav LDS, Yadav BS, Rai VK (2004) A novel salicylaldehyde based mineral supported expedient synthesis of benzoxazinone nucleosides. Tetrahedron Lett 45:5351-5353 (Pubitemid 38781852)
22. Yang HJ, Sun WH, Li ZL, Ma Z (2002) The rapid synthesis of Schiffbase without solvent under microwave irradiation. Chin Chem Lett 13:3-6