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Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 12, 2012, Pages 3973-3977

Identification of benzoxazole analogs as novel, S1P3 sparing S1P1 agonists

(11) Deng, Guanghui a Meng, Qinghua a Liu, Qian a Xu, Xuesong a Xu, Qiongfeng a Ren, Feng a Guo, Taylor B a Lu, Hongtao a Xiang, Jia Ning a Elliott, John D a Lin, Xichen a

a GLAXOSMITHKLINE (China)

Author keywords

Agonist; Lymphopenia; Multiple sclerosis; Sphingosine 1 phosphate (S1P)

Indexed keywords

BENZOXAZOLE DERIVATIVE;

ARTICLE; CENTRAL NERVOUS SYSTEM; DRUG EFFICACY; DRUG PENETRATION; DRUG POTENCY; IN VIVO STUDY; PERIPHERAL LYMPHOCYTE; STRUCTURE ACTIVITY RELATION;

ADMINISTRATION, ORAL; ANIMALS; BENZOXAZOLES; BINDING SITES; CALCIUM; IMMUNOSUPPRESSIVE AGENTS; LYMPHOCYTE COUNT; LYMPHOCYTES; MICE; MODELS, MOLECULAR; PROTEIN BINDING; RECEPTORS, LYSOSPHINGOLIPID; SENSITIVITY AND SPECIFICITY; STRUCTURE-ACTIVITY RELATIONSHIP;

MUS;

EID: 84861576687 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2012.04.095 Document Type: Article

Times cited : (7)

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* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.