메뉴 건너뛰기




Volumn 56, Issue 6, 2012, Pages 3114-3120

Sterilizing activities of novel combinations lacking first- and second-line drugs in a murine model of tuberculosis

Author keywords

[No Author keywords available]

Indexed keywords

6,7 DIHYDRO 2 NITRO 6 (4 TRIFLUOROMETHOXYBENZYLOXY) 5H IMIDAZO[2,1 B][1,3]OXAZINE; BEDAQUILINE; CLOFAZIMINE; ISONIAZID; MOXIFLOXACIN; PYRAZINAMIDE; RIFAMPICIN; RIFAPENTINE; SUTEZOLID;

EID: 84861137329     PISSN: 00664804     EISSN: 10986596     Source Type: Journal    
DOI: 10.1128/AAC.00384-12     Document Type: Article
Times cited : (136)

References (47)
  • 1
    • 58149394712 scopus 로고    scopus 로고
    • Increasing incidence of fluoroquinolone-resistant Mycobacterium tuberculosis in Mumbai, India
    • Agrawal D, Udwadia ZF, Rodriguez C, Mehta A. 2009. Increasing incidence of fluoroquinolone-resistant Mycobacterium tuberculosis in Mumbai, India. Int. J. Tuberc. Lung Dis. 13:79-83.
    • (2009) Int. J. Tuberc. Lung Dis. , vol.13 , pp. 79-83
    • Agrawal, D.1    Udwadia, Z.F.2    Rodriguez, C.3    Mehta, A.4
  • 2
    • 79958826429 scopus 로고    scopus 로고
    • Effectiveness of tuberculosis chemotherapy correlates with resistance to Mycobacterium tuberculosis infection in animal models
    • Ahmad Z, et al. 2011. Effectiveness of tuberculosis chemotherapy correlates with resistance to Mycobacterium tuberculosis infection in animal models. J. Antimicrob. Chemother. 66:1560-1566.
    • (2011) J. Antimicrob. Chemother. , vol.66 , pp. 1560-1566
    • Ahmad, Z.1
  • 3
    • 79952346767 scopus 로고    scopus 로고
    • Susceptibility of clinical Mycobacterium tuberculosis isolates to a potentially less toxic derivate of linezolid, PNU-100480
    • Alffenaar JW, et al. 2011. Susceptibility of clinical Mycobacterium tuberculosis isolates to a potentially less toxic derivate of linezolid, PNU-100480. Antimicrob. Agents Chemother. 55:1287-1289.
    • (2011) Antimicrob. Agents Chemother. , vol.55 , pp. 1287-1289
    • Alffenaar, J.W.1
  • 6
    • 63349091494 scopus 로고    scopus 로고
    • Moxifloxacin versus ethambutol in the initial treatment of tuberculosis: A double-blind, randomised, controlled phase II trial
    • Conde MB, et al. 2009. Moxifloxacin versus ethambutol in the initial treatment of tuberculosis: a double-blind, randomised, controlled phase II trial. Lancet 373:1183-1189.
    • (2009) Lancet , vol.373 , pp. 1183-1189
    • Conde, M.B.1
  • 7
    • 70350322939 scopus 로고    scopus 로고
    • Noninvasive pulmonary [18F]-2-fluoro-deoxy-Dglucose positron emission tomography correlates with bactericidal activity of tuberculosis drug treatment
    • Davis SL, et al. 2009. Noninvasive pulmonary [18F]-2-fluoro-deoxy- Dglucose positron emission tomography correlates with bactericidal activity of tuberculosis drug treatment. Antimicrob. Agents Chemother. 53:4879-4884.
    • (2009) Antimicrob. Agents Chemother. , vol.53 , pp. 4879-4884
    • Davis, S.L.1
  • 8
    • 79952336855 scopus 로고    scopus 로고
    • Comparative studies evaluating mouse models used for efficacy testing of experimental drugs against Mycobacterium tuberculosis
    • De Groote MA, et al. 2011. Comparative studies evaluating mouse models used for efficacy testing of experimental drugs against Mycobacterium tuberculosis. Antimicrob. Agents Chemother. 55:1237-1247.
    • (2011) Antimicrob. Agents Chemother. , vol.55 , pp. 1237-1247
    • De Groote, M.A.1
  • 9
    • 84856077753 scopus 로고    scopus 로고
    • Importance of confirming data on the in vivo efficacy of novel antibacterial drug regimens against various strains of Mycobacterium tuberculosis
    • De Groote MA, et al. 2012. Importance of confirming data on the in vivo efficacy of novel antibacterial drug regimens against various strains of Mycobacterium tuberculosis. Antimicrob. Agents Chemother. 56:731-738.
    • (2012) Antimicrob. Agents Chemother. , vol.56 , pp. 731-738
    • De Groote, M.A.1
  • 10
    • 80053972438 scopus 로고    scopus 로고
    • Course of murine tuberculosis and response to first-line therapy depends on route of infection and inoculum size
    • de Steenwinkel JE, et al. 2011. Course of murine tuberculosis and response to first-line therapy depends on route of infection and inoculum size. Int. J. Tuberc. Lung Dis. 15:1478-1484.
    • (2011) Int. J. Tuberc. Lung Dis. , vol.15 , pp. 1478-1484
    • De Steenwinkel, J.E.1
  • 11
    • 66649090346 scopus 로고    scopus 로고
    • The diarylquinoline TMC207 for multidrugresistant tuberculosis
    • Diacon AH, et al. 2009. The diarylquinoline TMC207 for multidrugresistant tuberculosis. N. Engl. J. Med. 360:2397-2405.
    • (2009) N. Engl. J. Med. , vol.360 , pp. 2397-2405
    • Diacon, A.H.1
  • 13
    • 0037417012 scopus 로고    scopus 로고
    • Mycobacterium tuberculosis in the extracellular compartment: An underestimated adversary
    • DOI 10.1128/AAC.47.3.833-836.2003
    • Grosset J. 2003. Mycobacterium tuberculosis in the extracellular compartment: an underestimated adversary. Antimicrob. Agents Chemother. 47:833-836. (Pubitemid 36254203)
    • (2003) Antimicrobial Agents and Chemotherapy , vol.47 , Issue.3 , pp. 833-836
    • Grosset, J.1
  • 14
    • 84856301870 scopus 로고    scopus 로고
    • Mouse model of necrotic tuberculosis granulomas develops hypoxic lesions
    • Harper J, et al. 2012. Mouse model of necrotic tuberculosis granulomas develops hypoxic lesions. J. Infect. Dis. 205:595-602.
    • (2012) J. Infect. Dis. , vol.205 , pp. 595-602
    • Harper, J.1
  • 15
    • 79952847428 scopus 로고    scopus 로고
    • Location of intra- and extracellular M. tuberculosis populations in lungs of mice and guinea pigs during disease progression and after drug treatment
    • Hoff DR, et al. 2011. Location of intra- and extracellular M. tuberculosis populations in lungs of mice and guinea pigs during disease progression and after drug treatment. PLoS One 6:e17550.
    • (2011) PLoS One , vol.6
    • Hoff, D.R.1
  • 17
    • 0028102968 scopus 로고
    • Effectiveness of various antimicrobial agents against Mycobacterium avium complex in the beige mouse model
    • Ji B, Lounis N, Truffot-Pernot C, Grosset J. 1994. Effectiveness of various antimicrobial agents against Mycobacterium avium complex in the beige mouse model. Antimicrob. Agents Chemother. 38:2521-2529. (Pubitemid 24332580)
    • (1994) Antimicrobial Agents and Chemotherapy , vol.38 , Issue.11 , pp. 2521-2529
    • Ji, B.1    Lounis, N.2    Truffot-Pernot, C.3    Grosset, J.4
  • 18
    • 84555220645 scopus 로고    scopus 로고
    • Patterns of pncA mutations in drug-resistant Mycobacterium tuberculosis isolated from patients in South Korea
    • Kim HJ, et al. 2012. Patterns of pncA mutations in drug-resistant Mycobacterium tuberculosis isolated from patients in South Korea. Int. J. Tuberc. Lung Dis. 16:98-103.
    • (2012) Int. J. Tuberc. Lung Dis. , vol.16 , pp. 98-103
    • Kim, H.J.1
  • 19
    • 49049106807 scopus 로고    scopus 로고
    • Prevention of drug carryover effects in studies assessing antimycobacterial efficacy of TMC207
    • Lounis N, et al. 2008. Prevention of drug carryover effects in studies assessing antimycobacterial efficacy of TMC207. J. Clin. Microbiol. 46:2212-2215.
    • (2008) J. Clin. Microbiol. , vol.46 , pp. 2212-2215
    • Lounis, N.1
  • 21
    • 80054681349 scopus 로고    scopus 로고
    • Pyrazinoic acid decreases the proton motive force, respiratory ATP synthesis activity, and cellular ATP levels
    • Lu P, et al. 2011. Pyrazinoic acid decreases the proton motive force, respiratory ATP synthesis activity, and cellular ATP levels. Antimicrob. Agents Chemother. 55:5354-5357.
    • (2011) Antimicrob. Agents Chemother. , vol.55 , pp. 5354-5357
    • Lu, P.1
  • 22
    • 80054700266 scopus 로고    scopus 로고
    • Clofazimine analogs with efficacy against experimental tuberculosis and reduced potential for accumulation
    • Lu Y, et al. 2011. Clofazimine analogs with efficacy against experimental tuberculosis and reduced potential for accumulation. Antimicrob. Agents Chemother. 55:5185-5193.
    • (2011) Antimicrob. Agents Chemother. , vol.55 , pp. 5185-5193
    • Lu, Y.1
  • 23
    • 33845323336 scopus 로고    scopus 로고
    • OPC-67683, a nitro-dihydro-imidazooxazole derivative with promising action against tuberculosis in vitro and in mice
    • Matsumoto M, et al. 2006. OPC-67683, a nitro-dihydro-imidazooxazole derivative with promising action against tuberculosis in vitro and in mice. PLoS Med. 3:e466.
    • (2006) PLoS Med. , vol.3
    • Matsumoto, M.1
  • 24
    • 84873075127 scopus 로고    scopus 로고
    • Combination therapy with novel TB drugs
    • Progr. Abstr. Virology Education B.V., Utrecht, The Netherlands
    • Mdluli K. 2011. Combination therapy with novel TB drugs. Progr. Abstr. Fourth Int. Workshop Clin. Pharmacol. Tuberculosis Drugs, Chicago, IL, 16 September 2011. Virology Education B.V., Utrecht, The Netherlands. http://regist2.virology-education.com/2011/4TB-PK/docs/07-Mdluli.pdf.
    • (2011) Fourth Int. Workshop Clin. Pharmacol. Tuberculosis Drugs, Chicago, IL, 16 September 2011
    • Mdluli, K.1
  • 25
    • 53649111744 scopus 로고    scopus 로고
    • Pyrazinamide resistance among South African multidrug-resistant Mycobacterium tuberculosis isolates
    • Mphahlele M, et al. 2008. Pyrazinamide resistance among South African multidrug-resistant Mycobacterium tuberculosis isolates. J. Clin. Microbiol. 46:3459 -3464.
    • (2008) J. Clin. Microbiol. , vol.46 , pp. 3459-3464
    • Mphahlele, M.1
  • 28
    • 84855706343 scopus 로고    scopus 로고
    • Fluoroquinolone and pyrazinamide resistance in multidrug-resistant tuberculosis
    • Pierre-Audigier C, et al. 2012. Fluoroquinolone and pyrazinamide resistance in multidrug-resistant tuberculosis. Int. J. Tuberc. Lung Dis. 16:221-223.
    • (2012) Int. J. Tuberc. Lung Dis. , vol.16 , pp. 221-223
    • Pierre-Audigier, C.1
  • 32
    • 38049038389 scopus 로고    scopus 로고
    • Daily dosing of rifapentine cures tuberculosis in three months or less in the murine model
    • Rosenthal IM, et al. 2007. Daily dosing of rifapentine cures tuberculosis in three months or less in the murine model. PLoS Med. 4:e344.
    • (2007) PLoS Med. , vol.4
    • Rosenthal, I.M.1
  • 33
    • 84857157134 scopus 로고    scopus 로고
    • Pharmacokinetics-pharmacodynamics of TMC207 and its N-desmethyl metabolite in a murine model of tuberculosis
    • Rouan MC, et al. 2012. Pharmacokinetics-pharmacodynamics of TMC207 and its N-desmethyl metabolite in a murine model of tuberculosis. Antimicrob. Agents Chemother. 56:1444-1451.
    • (2012) Antimicrob. Agents Chemother. , vol.56 , pp. 1444-1451
    • Rouan, M.C.1
  • 35
    • 77952357833 scopus 로고    scopus 로고
    • New initiative speeds tuberculosis drug development: Novel drug regimens become possible in years, not decades
    • Spigelman M, Woosley R, Gheuens J. 2010. New initiative speeds tuberculosis drug development: novel drug regimens become possible in years, not decades. Int. J. Tuberc. Lung Dis. 14:663-664.
    • (2010) Int. J. Tuberc. Lung Dis. , vol.14 , pp. 663-664
    • Spigelman, M.1    Woosley, R.2    Gheuens, J.3
  • 36
    • 81555221113 scopus 로고    scopus 로고
    • Sterilizing activity of novel TMC207- And PA-824-containing regimens in a murine model of tuberculosis
    • Tasneen R, et al. 2011. Sterilizing activity of novel TMC207- and PA-824-containing regimens in a murine model of tuberculosis. Antimicrob. Agents Chemother. 55:5485-5492.
    • (2011) Antimicrob. Agents Chemother. , vol.55 , pp. 5485-5492
    • Tasneen, R.1
  • 37
    • 54049098833 scopus 로고    scopus 로고
    • Enhanced bactericidal activity of rifampin and/or pyrazinamide when combined with PA-824 in a murine model of tuberculosis
    • Tasneen R, Tyagi S, Williams K, Grosset J, Nuermberger E. 2008. Enhanced bactericidal activity of rifampin and/or pyrazinamide when combined with PA-824 in a murine model of tuberculosis. Antimicrob. Agents Chemother. 52:3664-3668.
    • (2008) Antimicrob. Agents Chemother. , vol.52 , pp. 3664-3668
    • Tasneen, R.1    Tyagi, S.2    Williams, K.3    Grosset, J.4    Nuermberger, E.5
  • 39
    • 77952365008 scopus 로고    scopus 로고
    • Short, highly effective, and inexpensive standardized treatment of multidrug-resistant tuberculosis
    • van Deun A, et al. 2010. Short, highly effective, and inexpensive standardized treatment of multidrug-resistant tuberculosis. Am. J. Respir. Crit. Care Med. 182:684-692.
    • (2010) Am. J. Respir. Crit. Care Med. , vol.182 , pp. 684-692
    • Van Deun, A.1
  • 40
    • 0030887404 scopus 로고    scopus 로고
    • Riminophenazine compounds: Pharmacology and anti-neoplastic potential
    • DOI 10.1016/S1040-8428(96)00229-6, PII S1040842896002296
    • van Rensburg CE, Anderson R, O'Sullivan JF. 1997. Riminophenazine compounds: pharmacology and anti-neoplastic potential. Crit. Rev. Oncol. Hematol. 25:55-67. (Pubitemid 27138048)
    • (1997) Critical Reviews in Oncology/Hematology , vol.25 , Issue.1 , pp. 55-67
    • Van Rensburg, C.E.J.1    Anderson, R.2    O'Sullivan, J.F.3
  • 41
    • 78751693374 scopus 로고    scopus 로고
    • Biomarker-assisted dose selection for safety and efficacy in early development of PNU-100480 for tuberculosis
    • Wallis RS, et al. 2011. Biomarker-assisted dose selection for safety and efficacy in early development of PNU-100480 for tuberculosis. Antimicrob. Agents Chemother. 55:567-574.
    • (2011) Antimicrob. Agents Chemother. , vol.55 , pp. 567-574
    • Wallis, R.S.1
  • 42
    • 84855928950 scopus 로고    scopus 로고
    • Rapid evaluation in whole blood culture of regimens for XDR-TB containing PNU-100480 (Sutezolid), TMC207, PA-824, SQ109, and pyrazinamide
    • Wallis RS, et al. 2012. Rapid evaluation in whole blood culture of regimens for XDR-TB containing PNU-100480 (Sutezolid), TMC207, PA-824, SQ109, and pyrazinamide. PLoS One 7:e30479.
    • (2012) PLoS One , vol.7
    • Wallis, R.S.1
  • 43
    • 77955706291 scopus 로고    scopus 로고
    • Pharmacokinetics and whole-blood bactericidal activity against Mycobacterium tuberculosis of single doses of PNU-100480 in healthy volunteers
    • Wallis RS, et al. 2010. Pharmacokinetics and whole-blood bactericidal activity against Mycobacterium tuberculosis of single doses of PNU-100480 in healthy volunteers. J. Infect. Dis. 202:745-751.
    • (2010) J. Infect. Dis. , vol.202 , pp. 745-751
    • Wallis, R.S.1
  • 44
    • 68849115048 scopus 로고    scopus 로고
    • Addition of PNU-100480 to first-line drugs shortens the time needed to cure murine tuberculosis
    • Williams KN, et al. 2009. Addition of PNU-100480 to first-line drugs shortens the time needed to cure murine tuberculosis. Am. J. Respir. Crit. Care Med. 180:371-376.
    • (2009) Am. J. Respir. Crit. Care Med. , vol.180 , pp. 371-376
    • Williams, K.N.1
  • 45
    • 65649089528 scopus 로고    scopus 로고
    • Promising antituberculosis activity of the oxazolidinone PNU-100480 relative to that of linezolid in a murine model
    • Williams KN, et al. 2009. Promising antituberculosis activity of the oxazolidinone PNU-100480 relative to that of linezolid in a murine model. Antimicrob. Agents Chemother. 53:1314 -1319.
    • (2009) Antimicrob. Agents Chemother. , vol.53 , pp. 1314-1319
    • Williams, K.N.1
  • 46
    • 79953218013 scopus 로고    scopus 로고
    • Reduction of clofazimine by mycobacterial type 2 NADH:quinone oxidoreductase: A pathway for the generation of bactericidal levels of reactive oxygen species
    • Yano T, et al. 2011. Reduction of clofazimine by mycobacterial type 2 NADH:quinone oxidoreductase: a pathway for the generation of bactericidal levels of reactive oxygen species. J. Biol. Chem. 286:10276-10287.
    • (2011) J. Biol. Chem. , vol.286 , pp. 10276-10287
    • Yano, T.1
  • 47
    • 80052916123 scopus 로고    scopus 로고
    • Short-course chemotherapy with TMC207 and rifapentine in a murine model of latent tuberculosis infection
    • Zhang T, Li SY, Williams KN, Andries K, Nuermberger EL. 2011. Short-course chemotherapy with TMC207 and rifapentine in a murine model of latent tuberculosis infection. Am. J. Respir. Crit. Care Med. 184:732-737.
    • (2011) Am. J. Respir. Crit. Care Med. , vol.184 , pp. 732-737
    • Zhang, T.1    Li, S.Y.2    Williams, K.N.3    Andries, K.4    Nuermberger, E.L.5


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.