Characterisation of Plasmodium falciparum aspartic protease inhibition by piperidine derivatives

Natural Product Research

Volumn 25, Issue 20, 2011, Pages 1965-1968

  Saify, Zafar Saied ^a   Nisa, Mehrun ^a   Azhar, Kaniz Fizza ^b   Azim, M Kamran ^a   Rasheed, Huma ^a   Mushtaq, Nousheen ^a   Arain, M Arshad ^a   Haider, Shazia ^a   Khanum, Manawar ^a   Ahmed, Waseem ^c  

^a UNIVERSITY OF KARACHI   (Pakistan)

^b PCSIR LABORATORIES COMPLEX   (Pakistan)

^c FEDERAL URDU UNIVERSITY OF ARTS   (Pakistan)

Author keywords

ligand docking; NO 2 group; pepstatin A; piperidine derivatives; plasmepsin

Indexed keywords

1 METHYL 1(4' NITROPHENACYL) 4 HYDROXYPIPERIDINIUM BROMIDE; ASPARTIC PROTEINASE; BENZENE; PIPERIDINE DERIVATIVE; PLASMEPSIN II; PLASMEPSIN INHIBITOR; UNCLASSIFIED DRUG;

ARTICLE; CONCENTRATION (PARAMETERS); DRUG SYNTHESIS; ENZYME ASSAY; ENZYME INHIBITION; PLASMODIUM FALCIPARUM; STRUCTURE ACTIVITY RELATION;

ASPARTIC ACID ENDOPEPTIDASES; ASPARTIC ACID PROTEASES; NITROPHENOLS; PIPERIDINES; PLASMODIUM FALCIPARUM; PROTEIN BINDING; PROTOZOAN PROTEINS;

EID: 84857148549     PISSN: 14786419     EISSN: 14786427     Source Type: Journal    
DOI: 10.1080/14786419.2010.541881     Document Type: Article

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