Anti-ischemic effects of multivalent dendrimeric A 3 adenosine receptor agonists in cultured cardiomyocytes and in the isolated rat heart

Pharmacological Research

Volumn 65, Issue 3, 2012, Pages 338-346

  Chanyshev, Bella ^a   Shainberg, Asher ^a   Isak, Ahuva ^a   Litinsky, Alexandra ^a   Chepurko, Yelena ^b   Tosh, Dilip K ^c   Phan, Khai ^c   Gao, Zhan Guo ^c   Hochhauser, Edith ^b   Jacobson, Kenneth A ^c  

^a BAR ILAN UNIVERSITY   (Israel)

^b TEL AVIV UNIVERSITY   (Israel)

^c NATIONAL INSTITUTE OF DIABETES AND DIGESTIVE AND KIDNEY DISEASES   (United States)

Author keywords

Adenosine receptor; Cardiomyocyte; Dendrimer; Ischemia; Isolated heart; Rat

Indexed keywords

2 CHLORO 6 N (3 IODOBENZYL)ADENOSINE 5' N METHYLCARBOXAMIDE; 5 PROPYL 2 ETHYL 4 PROPYL 3 (ETHYLSULFANYLCARBONYL) 6 PHENYLPYRIDINE 5 CARBOXYLATE; 6 ETHYL 2 PHENYL 4 PROPYL 3 PYRIDINECARBOXYLIC ACID 5 THIOCARBOXYLIC ACID 5 ETHYL 3 PROPYL ESTER; 6 N (3 IODOBENZYL)ADENOSINE 5' N METHYLCARBOXAMIDE; ADENOSINE A3 RECEPTOR; ADENOSINE A3 RECEPTOR AGONIST; ADENOSINE A3 RECEPTOR ANTAGONIST; MRS 5216; MRS 5246; MRS 5539; POLYAMIDOAMINE; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; CELL CULTURE; CELL SURFACE; CONTROLLED STUDY; DRUG CONJUGATION; DRUG POTENCY; DRUG STRUCTURE; ENZYME ACTIVATION; HEART CONTRACTION; HEART INFARCTION SIZE; HEART MUSCLE CELL; HEART MUSCLE ISCHEMIA; HEART MUSCLE RELAXATION; HEART PROTECTION; HEART VENTRICLE PRESSURE; ISOLATED HEART; MALE; NONHUMAN; PRIORITY JOURNAL; RAT; RECEPTOR AFFINITY;

ADENOSINE; ADENOSINE A3 RECEPTOR AGONISTS; ANIMALS; CARDIOTONIC AGENTS; CELLS, CULTURED; DENDRIMERS; HEART; MALE; MYOCARDIAL ISCHEMIA; MYOCYTES, CARDIAC; RATS; RATS, SPRAGUE-DAWLEY; RECEPTOR, ADENOSINE A3;

EID: 84857062597     PISSN: 10436618     EISSN: 10961186     Source Type: Journal    
DOI: 10.1016/j.phrs.2011.11.013     Document Type: Article

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