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Volumn 53, Issue 3, 2012, Pages 248-250

Prevalence of TMC278 (rilpivirine) associated mutations in the Frankfurt Resistance Database

Author keywords

Drug resistance; Prevalence; Rilpivirine; TMC278

Indexed keywords

RILPIVIRINE;

EID: 84856964209     PISSN: 13866532     EISSN: 18735967     Source Type: Journal    
DOI: 10.1016/j.jcv.2011.12.012     Document Type: Article
Times cited : (11)

References (16)
  • 1
    • 35348995999 scopus 로고    scopus 로고
    • Is it safe to switch between efavirenz and nevirapine in the event of toxicity?
    • Mehta U., Maartens G. Is it safe to switch between efavirenz and nevirapine in the event of toxicity?. Lancet Infect Dis 2007, 7(11):733-738.
    • (2007) Lancet Infect Dis , vol.7 , Issue.11 , pp. 733-738
    • Mehta, U.1    Maartens, G.2
  • 2
    • 75149149567 scopus 로고    scopus 로고
    • Safety and tolerability of etravirine
    • Portilla J. Safety and tolerability of etravirine. Enferm Infecc Microbiol Clin 2009, 27(Suppl. 2):21-26.
    • (2009) Enferm Infecc Microbiol Clin , vol.27 , Issue.SUPPL. 2 , pp. 21-26
    • Portilla, J.1
  • 3
    • 0035903010 scopus 로고    scopus 로고
    • Female sex and the use of anti-allergic agents increase the risk of developing cutaneous rash associated with nevirapine therapy
    • Antinori A., Baldini F., Girardi E., Cingolani A., Zaccarelli M., Di Giambenedetto S., et al. Female sex and the use of anti-allergic agents increase the risk of developing cutaneous rash associated with nevirapine therapy. AIDS 2001, 15(12):1579-1581.
    • (2001) AIDS , vol.15 , Issue.12 , pp. 1579-1581
    • Antinori, A.1    Baldini, F.2    Girardi, E.3    Cingolani, A.4    Zaccarelli, M.5    Di Giambenedetto, S.6
  • 4
    • 34347327010 scopus 로고    scopus 로고
    • DUET-1 study group. Efficacy and safety of TMC125 (etravirine) in treatment-experienced HIV-1-infected patients in DUET-1: 24-week results from a randomised, double-blind, placebo-controlled trial
    • Madruga J.V., Cahn P., Grinsztejn B., Haubrich R., Lalezari J., Mills A., et al. DUET-1 study group. Efficacy and safety of TMC125 (etravirine) in treatment-experienced HIV-1-infected patients in DUET-1: 24-week results from a randomised, double-blind, placebo-controlled trial. Lancet 2007, 370(9581):29-38.
    • (2007) Lancet , vol.370 , Issue.9581 , pp. 29-38
    • Madruga, J.V.1    Cahn, P.2    Grinsztejn, B.3    Haubrich, R.4    Lalezari, J.5    Mills, A.6
  • 5
    • 34347354196 scopus 로고    scopus 로고
    • Efficacy and safety of TMC125 (etravirine) in treatment-experienced HIV-1-infected patients in DUET-2: 24-week results from a randomised, double-blind, placebo-controlled trial
    • Lazzarin A., Campbell T., Clotet B., Johnson M., Katlama C., Moll A., et al. Efficacy and safety of TMC125 (etravirine) in treatment-experienced HIV-1-infected patients in DUET-2: 24-week results from a randomised, double-blind, placebo-controlled trial. Lancet 2007, 370(9581):39-48.
    • (2007) Lancet , vol.370 , Issue.9581 , pp. 39-48
    • Lazzarin, A.1    Campbell, T.2    Clotet, B.3    Johnson, M.4    Katlama, C.5    Moll, A.6
  • 6
    • 77649254869 scopus 로고    scopus 로고
    • Resistance profile of etravirine: combined analysis of baseline genotypic and phenotypic data from the randomized, controlled Phase III clinical studies
    • Vingerhoets J., Tambuyzer L., Azijn H., Hoogstoel A., Nijs S., Peeters M., et al. Resistance profile of etravirine: combined analysis of baseline genotypic and phenotypic data from the randomized, controlled Phase III clinical studies. AIDS 2010, 24(4):503-514.
    • (2010) AIDS , vol.24 , Issue.4 , pp. 503-514
    • Vingerhoets, J.1    Tambuyzer, L.2    Azijn, H.3    Hoogstoel, A.4    Nijs, S.5    Peeters, M.6
  • 7
    • 79960346744 scopus 로고    scopus 로고
    • Rilpivirine: a step forward in tailored HIV treatment
    • July
    • Schrijvers R., Ayele Desimmie B., Debyser Z. Rilpivirine: a step forward in tailored HIV treatment. Lancet 2011, 378(July (9787)):201-203.
    • (2011) Lancet , vol.378 , Issue.9787 , pp. 201-203
    • Schrijvers, R.1    Ayele Desimmie, B.2    Debyser, Z.3
  • 8
    • 20144366006 scopus 로고    scopus 로고
    • Synthesis of novel diarylpyrimidine analogues and their antiviral activity against human immunodeficiency virus type 1
    • Guillemont J., Pasquier E., Palandjian P., Vernier D., Gaurrand S., Lewi P.J., et al. Synthesis of novel diarylpyrimidine analogues and their antiviral activity against human immunodeficiency virus type 1. J Med Chem 2005, 48:2072-2079.
    • (2005) J Med Chem , vol.48 , pp. 2072-2079
    • Guillemont, J.1    Pasquier, E.2    Palandjian, P.3    Vernier, D.4    Gaurrand, S.5    Lewi, P.J.6
  • 9
    • 20144372481 scopus 로고    scopus 로고
    • In search of a novel anti-HIV drug: multidisciplinary coordination in the discovery of 4-[[4-[[4-[(1E)-2-cyanoethenyl]-2,6-dimethylphenyl]amino]-2-pyrimidinyl]amino]benzonitrile (R278474, rilpivirine)
    • Janssen P.A., Lewi P.J., Arnold E., Daeyaert F., de Jonge M., Heeres J., et al. In search of a novel anti-HIV drug: multidisciplinary coordination in the discovery of 4-[[4-[[4-[(1E)-2-cyanoethenyl]-2,6-dimethylphenyl]amino]-2-pyrimidinyl]amino]benzonitrile (R278474, rilpivirine). J Med Chem 2005, 48:1901-1909.
    • (2005) J Med Chem , vol.48 , pp. 1901-1909
    • Janssen, P.A.1    Lewi, P.J.2    Arnold, E.3    Daeyaert, F.4    de Jonge, M.5    Heeres, J.6
  • 10
    • 75749118495 scopus 로고    scopus 로고
    • TMC278, a next-generation nonnucleoside reverse transcriptase inhibitor (NNRTI), active against wild-type and NNRTI-resistant HIV-1
    • Azijn H., Tirry I., Vingerhoets J., de Béthune M.P., Kraus G., Boven K., et al. TMC278, a next-generation nonnucleoside reverse transcriptase inhibitor (NNRTI), active against wild-type and NNRTI-resistant HIV-1. Antimicrob Agents Chemother 2010, 54(2):718-727.
    • (2010) Antimicrob Agents Chemother , vol.54 , Issue.2 , pp. 718-727
    • Azijn, H.1    Tirry, I.2    Vingerhoets, J.3    de Béthune, M.P.4    Kraus, G.5    Boven, K.6
  • 11
    • 83655163698 scopus 로고    scopus 로고
    • Genotypic and phenotypic characterization of HIV-1 isolates obtained from patients on rilpivirine therapy experiencing virologic failure in the phase 3 ECHO and THRIVE studies: 48-week analysis
    • [Epub ahead of print], November
    • Rimsky L., Vingerhoets J., Van Eygen V., Eron J., Clotet B., Hoogstoel A., et al. Genotypic and phenotypic characterization of HIV-1 isolates obtained from patients on rilpivirine therapy experiencing virologic failure in the phase 3 ECHO and THRIVE studies: 48-week analysis. J Acquir Immune Defic Syndr 2011, (November). [Epub ahead of print].
    • (2011) J Acquir Immune Defic Syndr
    • Rimsky, L.1    Vingerhoets, J.2    Van Eygen, V.3    Eron, J.4    Clotet, B.5    Hoogstoel, A.6
  • 12
    • 79960381844 scopus 로고    scopus 로고
    • ECHO study group. Rilpivirine versus efavirenz with tenofovir and emtricitabine in treatment-naive adults infected with HIV-1 (ECHO): a phase 3 randomised double-blind active-controlled trial
    • Molina J.M., Cahn P., Grinsztejn B., Lazzarin A., Mills A., Saag M., et al. ECHO study group. Rilpivirine versus efavirenz with tenofovir and emtricitabine in treatment-naive adults infected with HIV-1 (ECHO): a phase 3 randomised double-blind active-controlled trial. Lancet 2011, 378(9787):238-246.
    • (2011) Lancet , vol.378 , Issue.9787 , pp. 238-246
    • Molina, J.M.1    Cahn, P.2    Grinsztejn, B.3    Lazzarin, A.4    Mills, A.5    Saag, M.6
  • 13
    • 79960358849 scopus 로고    scopus 로고
    • THRIVE study group. Rilpivirine versus efavirenz with two background nucleoside or nucleotide reverse transcriptase inhibitors in treatment-naive adults infected with HIV-1 (THRIVE): a phase 3, randomised, non-inferiority trial
    • Cohen C.J., Andrade-Villanueva J., Clotet B., Fourie J., Johnson M.A., Ruxrungtham K., et al. THRIVE study group. Rilpivirine versus efavirenz with two background nucleoside or nucleotide reverse transcriptase inhibitors in treatment-naive adults infected with HIV-1 (THRIVE): a phase 3, randomised, non-inferiority trial. Lancet 2011, 378(9787):229-237.
    • (2011) Lancet , vol.378 , Issue.9787 , pp. 229-237
    • Cohen, C.J.1    Andrade-Villanueva, J.2    Clotet, B.3    Fourie, J.4    Johnson, M.A.5    Ruxrungtham, K.6
  • 14
    • 0346252370 scopus 로고    scopus 로고
    • Variety of interpretation systems for human immunodeficiency virus type 1 genotyping: confirmatory information or additional confusion?
    • Stürmer M., Doerr H.W., Preiser W. Variety of interpretation systems for human immunodeficiency virus type 1 genotyping: confirmatory information or additional confusion?. Curr Drug Targets Infect Disord 2003, 3(4):373-382.
    • (2003) Curr Drug Targets Infect Disord , vol.3 , Issue.4 , pp. 373-382
    • Stürmer, M.1    Doerr, H.W.2    Preiser, W.3
  • 15
    • 0142182292 scopus 로고    scopus 로고
    • Modifications and substitutions of the RNA extraction module in the ViroSeq HIV-1 genotyping system version 2: effects on sensitivity and complexity of the assay
    • Stürmer M., Berger A., Doerr H.W. Modifications and substitutions of the RNA extraction module in the ViroSeq HIV-1 genotyping system version 2: effects on sensitivity and complexity of the assay. J Med Virol 2003, 71(4):475-479.
    • (2003) J Med Virol , vol.71 , Issue.4 , pp. 475-479
    • Stürmer, M.1    Berger, A.2    Doerr, H.W.3
  • 16
    • 62549083388 scopus 로고    scopus 로고
    • Etravirine and rilpivirine: nonnucleoside reverse transcriptase inhibitors with activity against human immunodeficiency virus type 1 strains resistant to previous nonnucleoside agents
    • Fulco P.P., McNicholl I.R. Etravirine and rilpivirine: nonnucleoside reverse transcriptase inhibitors with activity against human immunodeficiency virus type 1 strains resistant to previous nonnucleoside agents. Pharmacotherapy 2009, 29(3):281-294.
    • (2009) Pharmacotherapy , vol.29 , Issue.3 , pp. 281-294
    • Fulco, P.P.1    McNicholl, I.R.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.