An efficient, solvent-free microwave-assisted synthesis and antimicrobial screening of 1,6-dihydropyrimidine analogues

Medicinal Chemistry Research

Volumn 21, Issue 12, 2012, Pages 4412-4421

  Desai, N C ^a   Pandya, D D ^a   Satodiya, H M ^a   Rajpara, K M ^a   Joshi, V V ^a   Vaghani, H V ^a  

^a BHAVNAGAR UNIVERSITY   (India)

Author keywords

1,6 Dihydropyrimidine analogues; Antimicrobial activity; Conventional and microwave method; MIC

Indexed keywords

1,6 DIHYDROPYRIMIDINE DERIVATIVE; 2 (6 (4 AMINOPHENYL) 2 MERCAPTO 3,4 DIHYDROPYRIMIDIN 4 YL)PHENOL; 3 (6 (4 AMINOPHENYL) 2 MERCAPTO 3,4 DIHYDROPYRIMIDIN 4 YL)PHENOL; 4 (4 (4 AMINOPHENYL) 6 (2 HYDROXYPHENYL) 1,6 DIHYDROPYRIMIDIN 2 YLTHIO)BUTANENITRILE; 4 (4 (4 AMINOPHENYL) 6 (3 HYDROXYPHENYL) 1,6 DIHYDROPYRIMIDIN 2 YLTHIO)BUTANENITRILE; 4 (4 (4 AMINOPHENYL) 6 (4 (DIMETHYLAMINO)PHENYL) 1,6 DIHYDROPYRIMIDIN 2 YLTHIO)BUTANENITRILE; 4 (4 (4 AMINOPHENYL) 6 (4 CHLOROPHENYL) 1,6 DIHYDROPYRIMIDIN 2 YLTHIO)BUTANENITRILE; 4 (4 (4 AMINOPHENYL) 6 (4 HYDROXY 3 METHOXYPHENYL) 1,6 DIHYDROPYRIMIDIN 2 YLTHIO)BUTANENITRILE; 4 (4 (4 AMINOPHENYL) 6 (4 HYDROXYPHENYL) 1,6 DIHYDROPYRIMIDIN 2 YLTHIO)BUTANENITRILE; 4 (4 (4 AMINOPHENYL) 6 (4 NITROPHENYL) 1,6 DIHYDROPYRIMIDIN 2 YLTHIO)BUTANENITRILE; 4 (4 (4 AMINOPHENYL) 6 3 TOLYL 1,6 DIHYDROPYRIMIDIN 2 YLTHIO)BUTANENITRILE; 4 (4 (4 AMINOPHENYL) 6 4 METHOXYPHENYL) 1,6 DIHYDROPYRIMIDIN 2 YLTHIO)BUTANENITRILE; 4 (4 (4 AMINOPHENYL) 6 4 TOLYL 1,6 DIHYDROPYRIMIDIN 2 YLTHIO)BUTANENITRILE; 4 (4 (4 AMINOPHENYL) 6 O TOLYL 1,6 DIHYDROPYRIMIDIN 2 YLTHIO)BUTANENITRILE; 4 (4 (4 AMINOPHENYL) 6 PHENYL 1,6 DIHYDROPYRIMIDIN 2 YLTHIO)BUTANENITRILE; 4 (4 AMINOPHENYL) 6 (3 NITROPHENYL) 1,6 DIHYDROPYRIMIDINE 2 THIOL; 4 (4 AMINOPHENYL) 6 (4 (DIMETHYLAMINO)PHENYL) 1,6 DIHYDROPYRIMIDINE 2 THIOL; 4 (4 AMINOPHENYL) 6 (4 CHLOROPHENYL) 1,6 DIHYDROPYRIMIDINE 2 THIOL; 4 (4 AMINOPHENYL) 6 (4 METHOXYPHENYL) 1,6 DIHYDROPYRIMIDINE 2 THIOL; 4 (4 AMINOPHENYL) 6 3 TOLYL 1,6 DIHYDROPYRIMIDINE 2 THIOL; 4 (4 AMINOPHENYL) 6 4 TOLYL 1,6 DIHYDROPYRIMIDINE 2 THIOL; 4 (4 AMINOPHENYL) 6 O TOLYL 1,6 DIHYDROPYRIMIDINE 2 THIOL; 4 (4 AMINOPHENYL) 6 PHENYL 1,6 DIHYDROPYRIMIDINE 2 THIOL; 4 (6 (4 AMINOPHENYL) 2 MERCAPTO 3,4 DIHYDROPYRIMIDIN 4 YL) 2 METHOXYPHENOL; 4 (6 (4 AMINOPHENYL) 2 MERCAPTO 3,4 DIHYDROPYRIMIDIN 4 YL)PHENOL; AMPICILLIN; ANTIINFECTIVE AGENT; GRISEOFULVIN; UNCLASSIFIED DRUG;

ANTIMICROBIAL ACTIVITY; ARTICLE; BACTERIAL STRAIN; BROTH DILUTION; CARBON NUCLEAR MAGNETIC RESONANCE; DRUG STRUCTURE; DRUG SYNTHESIS; ESCHERICHIA COLI; FUNGAL STRAIN; INFRARED SPECTROSCOPY; MICROWAVE ASSISTED SYNTHESIS; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; PROTON NUCLEAR MAGNETIC RESONANCE; PSEUDOMONAS AERUGINOSA; STREPTOCOCCUS PYOGENES;

EID: 84856462255     PISSN: 10542523     EISSN: 15548120     Source Type: Journal    
DOI: 10.1007/s00044-012-9980-6     Document Type: Article

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