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Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 2, 2012, Pages 1103-1106

Synthesis of new praziquantel analogues: Potential candidates for the treatment of schistosomiasis

(6) Sadhu, Partha Sarathi a Kumar, Singam Naveen a Chandrasekharam, Malapaka a Pica Mattoccia, Livia b Cioli, Donato b Rao, Vaidya Jayathirtha a

a INDIAN INSTITUTE OF CHEMICAL TECHNOLOGY (India)

b CNR (Italy)

Author keywords

Antischistosomal; Praziquantel analogues; Schistosoma mansoni; Schistosomiasis

Indexed keywords

4 TOLUENE SULFONYL; 4 TRIFLUOROMETHYLBENZOYL; AMIDE; ANTISCHISTOSOMAL AGENT; AROMATIC COMPOUND; DIMETHOXY TETRAHYDROISOQUINOLINE DERIVATIVE; PIPERAZINE; PRAZIQUANTEL; TRYPTOLINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; DRUG ACTIVITY; DRUG SYNTHESIS; NONHUMAN; SCHISTOSOMA MANSONI; SCHISTOSOMIASIS; STRUCTURE ACTIVITY RELATION;

ANIMALS; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG DESIGN; MOLECULAR STRUCTURE; PRAZIQUANTEL; SCHISTOSOMA MANSONI; SCHISTOSOMIASIS; SCHISTOSOMICIDES; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP;

SCHISTOSOMA MANSONI;

EID: 84855660079 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2011.11.108 Document Type: Article

Times cited : (36)

References (36)

1
- 0034706868
- L. Chitsulo, D. Engels, A. Montresor, and L. Savioli Acta Trop. 77 2000 41
- (2000) Acta Trop. , vol.77 , pp. 41
- Chitsulo, L.¹ Engels, D.² Montresor, A.³ Savioli, L.⁴

2
- 1842458494
- L. Savioli, D. Engels, J.B. Roungou, A. Frenwick, and H. Endo Lancet 363 2004 658
- (2004) Lancet , vol.363 , pp. 658
- Savioli, L.¹ Engels, D.² Roungou, J.B.³ Frenwick, A.⁴ Endo, H.⁵

3
- 0036824166
- Y.-X. He, L. Chen, and K. Ramaswamy Exp. Parasitol. 102 2002 99
- (2002) Exp. Parasitol. , vol.102 , pp. 99
- He, Y.-X.¹ Chen, L.² Ramaswamy, K.³

4
- 0037847426
- M.J. Van der Werf, S.J. De Vlas, S. Brooker, C.W. Looman, N.J. Nagelkerke, J.D. Habbema, and D. Engels Acta Trop. 86 2003 125
- (2003) Acta Trop. , vol.86 , pp. 125
- Van Der Werf, M.J.¹ De Vlas, S.J.² Brooker, S.³ Looman, C.W.⁴ Nagelkerke, N.J.⁵ Habbema, J.D.⁶ Engels, D.⁷

5
- 0028895250
- D. Cioli, L. Pica-Mattoccia, and S. Archer Pharmacol. Ther. 68 1995 35
- (1995) Pharmacol. Ther. , vol.68 , pp. 35
- Cioli, D.¹ Pica-Mattoccia, L.² Archer, S.³

6
- 0142227135
- A. Fenwick, L. Savioli, D. Engels, R. Bergquist, and M.H. Todd Trends. Parasitol. 19 2003 509
- (2003) Trends. Parasitol. , vol.19 , pp. 509
- Fenwick, A.¹ Savioli, L.² Engels, D.³ Bergquist, R.⁴ Todd, M.H.⁵

7
- 84855672510
- http://www.schisto.org/.

8
- 11344254337
- L.-A.T. Tchuenté, D.J. Shaw, L. Polla, D. Cioli, and J. Vercruysse Am. J. Trop. Hyg. 71 2004 778
- (2004) Am. J. Trop. Hyg. , vol.71 , pp. 778
- Tchuenté, L.-A.T.¹ Shaw, D.J.² Polla, L.³ Cioli, D.⁴ Vercruysse, J.⁵

9
- 0033662883
- D. Cioli Curr. Opin. Infect. Dis. 13 2000 659
- (2000) Curr. Opin. Infect. Dis. , vol.13 , pp. 659
- Cioli, D.¹

10
- 0029955908
- S.Q. Murray-Smith, B.J. Scott, D.P. Barton, and P.A. Wienstein Med. J. Aust. 165 1996 458
- (1996) Med. J. Aust. , vol.165 , pp. 458
- Murray-Smith, S.Q.¹ Scott, B.J.² Barton, D.P.³ Wienstein, P.A.⁴

11
- 79961172802
- J. Utzinger, E.K. N'goran, C.R. Caffrey, and J. Keiser Acta. Trop. 120s 2011 s121
- (2011) Acta. Trop. , vol.120 S , pp. 121
- Utzinger, J.¹ N'Goran, E.K.² Caffrey, C.R.³ Keiser, J.⁴

12
- 70449568249
- M.H. Abdulla, D.S. Ruelas, B. Wolff, J. Snedecor, K.-C. Lim, F. Xu, A.R. Renslo, J. Williams, J.H. McKerrow, and C.R. Caffrey PLoS Negl. Trop. Dis. 3 2009 e478
- (2009) PLoS Negl. Trop. Dis. , vol.3 , pp. 478
- Abdulla, M.H.¹ Ruelas, D.S.² Wolff, B.³ Snedecor, J.⁴ Lim, K.-C.⁵ Xu, F.⁶ Renslo, A.R.⁷ Williams, J.⁸ McKerrow, J.H.⁹ Caffrey, C.R.¹⁰

13
- 33846697738
- M.H. Abdulla, M. Sajid, K.-C. Lim, J.H. McKerrow, and C.R. Caffrey PLoS Med. 4 2007 e14
- (2007) PLoS Med. , vol.4 , pp. 14
- Abdulla, M.H.¹ Sajid, M.² Lim, K.-C.³ McKerrow, J.H.⁴ Caffrey, C.R.⁵

14
- 70449510166
- S.D. Melman, M.L. Steinauer, C. Cunningham, L.S. Kubatko, I.N. Mwangi, N.B. Wynn, M.W. Mutuku, D.M.S. Karanja, D.G. Colley, C.L. Black, W.E. Secor, G.M. Mkoji, and E.S. Loker PLoS Negl. Trop. Dis. 3 2009 e504
- (2009) PLoS Negl. Trop. Dis. , vol.3 , pp. 504
- Melman, S.D.¹ Steinauer, M.L.² Cunningham, C.³ Kubatko, L.S.⁴ Mwangi, I.N.⁵ Wynn, N.B.⁶ Mutuku, M.W.⁷ Karanja, D.M.S.⁸ Colley, D.G.⁹ Black, C.L.¹⁰ Secor, W.E.¹¹ Mkoji, G.M.¹² Loker, E.S.¹³

15
- 0017410779
- J. Seubert, R. Pohlke, and F. Loebich Experientia 33 1977 1036
- (1977) Experientia , vol.33 , pp. 1036
- Seubert, J.¹ Pohlke, R.² Loebich, F.³

16
- 85042910533
- D. Frehel, and J.-P. Maffrand Heterocycles 20 1983 1731
- (1983) Heterocycles , vol.20 , pp. 1731
- Frehel, D.¹ Maffrand, J.-P.²

17
- 0001401343
- W.F. Berkowitz, and T.V. John J. Org. Chem. 49 1984 5269
- (1984) J. Org. Chem. , vol.49 , pp. 5269
- Berkowitz, W.F.¹ John, T.V.²

18
- 0022570771
- F. Yuste, Y. Pallas, H. Barrios, B. Oritz, and R.J. Sanchez-Obregon Heterocyl. Chem. 23 1986 189
- (1986) Heterocyl. Chem. , vol.23 , pp. 189
- Yuste, F.¹ Pallas, Y.² Barrios, H.³ Oritz, B.⁴ Sanchez-Obregon, R.J.⁵

19
- 0032565993
- J.H. Kim, Y.S. Lee, H. Park, and H.S. Kim Tetrahedron 54 1998 7395
- (1998) Tetrahedron , vol.54 , pp. 7395
- Kim, J.H.¹ Lee, Y.S.² Park, H.³ Kim, H.S.⁴

20
- 0037077002
- M.H. Todd, C. Ndubaku, and P.A. Bartlett J. Org. Chem. 67 2002 3985
- (2002) J. Org. Chem. , vol.67 , pp. 3985
- Todd, M.H.¹ Ndubaku, C.² Bartlett, P.A.³

21
- 84855672511
- German Patent 2, 362, 539
- Seubert, J.; Thomas, H.; Andrews, P. German Patent 2, 362, 539, 1975.
- (1975)
- Seubert, J.¹ Thomas, H.² Andrews, P.³

22
- 2942567749
- C. Ma, Q.-F. Zhang, Y.-B. Tan, and L.J. Wang Chem. Res. 2004 186
- (2004) Chem. Res. , pp. 186
- Ma, C.¹ Zhang, Q.-F.² Tan, Y.-B.³ Wang, L.J.⁴

23
- 84855698523
- P. Roszkowski, J.K. Maurin, and Z. Czarnocki Tetrahedron: Asymmetry 2006 1415 17
- (1415) Tetrahedron: Asymmetry , vol.2006 , pp. 17
- Roszkowski, P.¹ Maurin, J.K.² Czarnocki, Z.³

24
- 30944452978
- S. El-Fayyoumy, M. Mansour, and M.H. Todd Tetrahedron Lett. 47 2006 1287
- (2006) Tetrahedron Lett. , vol.47 , pp. 1287
- El-Fayyoumy, S.¹ Mansour, M.² Todd, M.H.³

25
- 0020525864
- P. Andrews, H. Thomas, R. Pholke, and J. Seubert Med. Res. Rev. 3 1983 147
- (1983) Med. Res. Rev. , vol.3 , pp. 147
- Andrews, P.¹ Thomas, H.² Pholke, R.³ Seubert, J.⁴

26
- 34347387279
- F. Ronketti, A.V. Ramana, X. Chao-Ming, L. Pica-Mattoccia, D. Cioli, and M.H. Todd Biorg.Med. Chem. Lett. 17 2007 4154
- (2007) Biorg.Med. Chem. Lett. , vol.17 , pp. 4154
- Ronketti, F.¹ Ramana, A.V.² Chao-Ming, X.³ Pica-Mattoccia, L.⁴ Cioli, D.⁵ Todd, M.H.⁶

27
- 77950267287
- Y. Dong, J. Chollet, M. Vargas, N.R. Mansour, Q. Bickle, Y. Alnouti, J. Huang, J. Keiser, and J.L. Vennerstrom Biorg. Med. Chem. Lett. 20 2010 2481
- (2010) Biorg. Med. Chem. Lett. , vol.20 , pp. 2481
- Dong, Y.¹ Chollet, J.² Vargas, M.³ Mansour, N.R.⁴ Bickle, Q.⁵ Alnouti, Y.⁶ Huang, J.⁷ Keiser, J.⁸ Vennerstrom, J.L.⁹

28
- 33746533902
- P. Narender, U. Srinivas, M. Ravinder, B. Anand Rao, C. Ramesh, K. Harakishore, B. Gangadasu, U.S.N. Murthy, and V. Jayathirtha Rao Bioorg. Med. Chem. 14 2006 4600
- (2006) Bioorg. Med. Chem. , vol.14 , pp. 4600
- Narender, P.¹ Srinivas, U.² Ravinder, M.³ Anand Rao, B.⁴ Ramesh, C.⁵ Harakishore, K.⁶ Gangadasu, B.⁷ Murthy, U.S.N.⁸ Jayathirtha Rao, V.⁹

29
- 27644582509
- P. Narender, U. Srinivas, B. Gangadasu, S. Biswas, and V. Jayathirtha Rao Bioorg. Med. Chem. Lett. 15 2005 5378
- (2005) Bioorg. Med. Chem. Lett. , vol.15 , pp. 5378
- Narender, P.¹ Srinivas, U.² Gangadasu, B.³ Biswas, S.⁴ Jayathirtha Rao, V.⁵

30
- 0141853234
- M.C. Elliott, and E. Williams Org. Bio. Chem. 2003 3038
- (2003) Org. Bio. Chem. , pp. 3038
- Elliott, M.C.¹ Williams, E.²

31
- 34547785059
- F. Werner, N. Blank, and T. Opatz Euro. J. Org. Chem. 2007 3911
- (2007) Euro. J. Org. Chem. , pp. 3911
- Werner, F.¹ Blank, N.² Opatz, T.³

32
- 0003663443
- N.J. Whittaker Chem. Soc. C 1969 85
- (1969) Chem. Soc. C , pp. 85
- Whittaker, N.J.¹

33
- 33744978812
- N.L. Sergovskaya, and S.A. Chernyak Khim. Geterotsikl. Soedin. 8 1991 1107
- (1991) Khim. Geterotsikl. Soedin. , vol.8 , pp. 1107
- Sergovskaya, N.L.¹ Chernyak, S.A.²

34
- 69549101621
- H. Liu, and A. Domling J. Org. Chem. 74 2009 6895
- (2009) J. Org. Chem. , vol.74 , pp. 6895
- Liu, H.¹ Domling, A.²

35
- 65549111256
- T. Meyer, H. Sekljic, S. Fuchs, H. Bothe, D. Schollmeyer, and C. Miculka PLoS Negl. Trop. Dis. 3 2009 e357
- (2009) PLoS Negl. Trop. Dis. , vol.3 , pp. 357
- Meyer, T.¹ Sekljic, H.² Fuchs, S.³ Bothe, H.⁴ Schollmeyer, D.⁵ Miculka, C.⁶

36
- 1542358686
- L. Pica-Mattoccia, and D. Cioli Int. J. Parasitol. 34 2004 527
- (2004) Int. J. Parasitol. , vol.34 , pp. 527
- Pica-Mattoccia, L.¹ Cioli, D.²

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