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Volumn 65, Issue 5, 2011, Pages 700-706

Synthesis and in vitro antimicrobial activity of new 3-(2- morpholinoquinolin-3-yl) substituted acrylonitrile and propanenitrile derivatives

Author keywords

2 morpholinoquinoline; Antimicrobial activity; MIC; Nitrile

Indexed keywords


EID: 83455187850     PISSN: 03666352     EISSN: 13369075     Source Type: Journal    
DOI: 10.2478/s11696-011-0048-8     Document Type: Conference Paper
Times cited : (10)

References (27)
  • 1
    • 67649836274 scopus 로고    scopus 로고
    • Comparative studies on conventional and microwave-assisted synthesis of a series of 2,4-di and 2,3,4-trisubstituted benzimidazo[1,2-a]pyrimidines and their antimicrobial activ-ities
    • DOI: 10.2478/s11532-009-0023-1
    • Algul, O., Meric, A., Polat, S., Yuksek, N. D., & Serin, M. S. (2009). Comparative studies on conventional and microwave-assisted synthesis of a series of 2,4-di and 2,3,4-trisubstituted benzimidazo[1,2-a]pyrimidines and their antimicrobial activ-ities. Central European Journal of Chemistry, 7, 337-342. DOI: 10.2478/s11532-009-0023-1
    • (2009) Central European Journal of Chemistry , vol.7 , pp. 337-342
    • Algul, O.1    Meric, A.2    Polat, S.3    Yuksek, N.D.4    Serin, M.S.5
  • 2
    • 36549058379 scopus 로고    scopus 로고
    • Synthesis and antioxidant capacities of some new benzimidazole derivatives
    • DOI 10.1002/ardp.200700088
    • Ayhan-Kilcǧil, G., Ku̧s, C., Ozdamar, E. D., Can-Eke, B., & I̧scan, M. (2007). Synthesis and antioxidant capacities of some new benzimidazole derivatives. Archiv der Pharmazie, 340, 607-611. DOI: 10.1002/ardp.200700088. (Pubitemid 350178679)
    • (2007) Archiv der Pharmazie , vol.340 , Issue.11 , pp. 607-611
    • Ayhan-Kilcigil, G.1    Kus, C.2    Ozdamar, E.D.3    Can-Eke, B.4    Ican, M.5
  • 4
    • 25444504491 scopus 로고    scopus 로고
    • Synthesis and antimalarial activity of E-2-quinolinylbenzocycloalcanones
    • DOI 10.1016/j.ejmech.2005.03.013, PII S0223523405000954
    • Charris, J. E., Domínguez, J. N., Gamboa, N., Rodrigues, J. R., & Angel, J. E. (2005). Synthesis and antimalarial activity of E-2-quinolinylbenzocycloalcanones. European Journal of Medicinal Chemistry, 40, 875-881. DOI: 10.1016/j.ejmech. 2005.03.013. (Pubitemid 41376302)
    • (2005) European Journal of Medicinal Chemistry , vol.40 , Issue.9 , pp. 875-881
    • Charris, J.E.1    Dominguez, J.N.2    Gamboa, N.3    Rodrigues, J.R.4    Angel, J.E.5
  • 5
    • 36849087457 scopus 로고    scopus 로고
    • A facile tandem synthesis of α-benzyl benzimidazole acetoni-triles
    • Dubey, P. K., Prasada Reddy, P. V. V., & Srinivas, K. (2007). A facile tandem synthesis of α-benzyl benzimidazole acetoni-triles. ARKIVOC, 2007(xv), 192-198.
    • (2007) ARKIVOC , vol.2007 , Issue.15 , pp. 192-198
    • Dubey, P.K.1    Prasada Reddy, P.V.V.2    Srinivas, K.3
  • 6
    • 0031834393 scopus 로고    scopus 로고
    • Legal issues associated with antimicrobial drug resistance
    • Fidler, D. P. (1998). Legal issues associated with antimicrobial drug resistance. Emerging Infectious Diseases, 4, 169-177. (Pubitemid 28311203)
    • (1998) Emerging Infectious Diseases , vol.4 , Issue.2 , pp. 169-177
    • Fidler, D.P.1
  • 7
    • 33645539695 scopus 로고    scopus 로고
    • Lanthanide(III) and yttrium(III) complexes of benzimidazole-2-acetic acid: Synthesis, characterisation and effect of La(III) complex on germination of wheat
    • DOI 10.1155/BCA/2006/75612
    • Gudasi, K. B., Shenoy, R. V., Vadavi, R. S., Patil, M. S., Patil, S. A., Hanchinal, R. R., Desai, S. A., & Lohithaswa, H. (2006). Lanthanide(III) and yttrium(III) complexes of benzimidazole-2-acetic acid: synthesis, characterisation and effect of La(III) complex on germination of wheat. Bioinor-ganic Chemistry and Applications, 2006, art. ID 75612. DOI: 10.1155/BCA/2006/75612. (Pubitemid 43509056)
    • (2006) Bioinorganic Chemistry and Applications , vol.2006 , pp. 75612
    • Gudasi, K.B.1    Shenoy, R.V.2    Vadavi, R.S.3    Patil, M.S.4    Patil, S.A.5    Hanchinal, R.R.6    Desai, S.A.7    Lohithaswa, H.8
  • 8
    • 0035271615 scopus 로고    scopus 로고
    • Discovery of gemifloxacin (Factive, LB20304a): A quinolone of new a generation
    • DOI 10.1016/S0014-827X(01)01017-5, PII S0014827X01010175
    • Hong, C. Y. (2001). Discovery of gemifloxacin (Factive, LB20304a): a quinolone of new a generation. Il Farmaco, 56, 41-44. DOI: 10.1016/s0014- 827X(01)01017-5. (Pubitemid 32372581)
    • (2001) Farmaco , vol.56 , Issue.1-2 , pp. 41-44
    • Hong, C.Y.1
  • 10
    • 77951234594 scopus 로고    scopus 로고
    • A con-venient one-pot synthesis of some new 3-(2-phenyl-6-(2-thienyl)-4- pyridyl)hydroquinolin-2-ones under microwave ir-radiation and their antimicrobial activities
    • DOI: 10.1080/10426500902915507
    • Ladani, N. K., Patel, M. P., & Patel, R. G. (2010). A con-venient one-pot synthesis of some new 3-(2-phenyl-6-(2-thienyl)-4-pyridyl)hydroquinolin- 2-ones under microwave ir-radiation and their antimicrobial activities. Phosphorus, Sul-fur, and Silicon and the Related Elements, 185, 658-662. DOI: 10.1080/10426500902915507.
    • (2010) Phosphorus, Sul-fur, and Silicon and the Related Elements , vol.185 , pp. 658-662
    • Ladani, N.K.1    Patel, M.P.2    Patel, R.G.3
  • 11
    • 67651111969 scopus 로고    scopus 로고
    • A convenient one-pot synthesis of series of 3-(2,6-diphenyl-4-pyridyl) hydroquinolin-2-one under microwave irradiation and their antimicrobial activities
    • Ladani, N. K., Patel, M. P., & Patel, R. G. (2009a). A convenient one-pot synthesis of series of 3-(2,6-diphenyl-4-pyridyl)hydroquinolin-2-one under microwave irradiation and their antimicrobial activities. Indian Journal of Chemistry, 48B, 261-266.
    • (2009) Indian Journal of Chemistry , vol.48 B , pp. 261-266
    • Ladani, N.K.1    Patel, M.P.2    Patel, R.G.3
  • 12
    • 77952680353 scopus 로고    scopus 로고
    • An ef-ficient three component one-pot synthesis of some new oc-tahydroquinazolinone derivatives and investigation of their antimicrobial activities
    • 2009
    • Ladani, N. K., Patel, M. P., & Patel, R. G. (2009b). An ef-ficient three component one-pot synthesis of some new oc-tahydroquinazolinone derivatives and investigation of their antimicrobial activities. ARKIVOC, 2009(vii), 292-302.
    • (2009) ARKIVOC , vol.7 , pp. 292-302
    • Ladani, N.K.1    Patel, M.P.2    Patel, R.G.3
  • 13
    • 0000525422 scopus 로고
    • A versatile new synthe-sis of quinolines, thienopyridines and related fused pyridines
    • DOI: 10.1016/S0040-4039(01)94745-8
    • Meth-Cohn, O., & Bramha, N. (1978). A versatile new synthe-sis of quinolines, thienopyridines and related fused pyridines. Tetrahedron Letters, 19, 2045-2048. DOI: 10.1016/S0040-4039(01)94745-8.
    • (1978) Tetrahedron Letters , vol.19 , pp. 2045-2048
    • Meth-Cohn, O.1    Bramha, N.2
  • 14
    • 33645821103 scopus 로고    scopus 로고
    • Synthesis and antimycobacterial activities of certain trifluoromethyl- aminoquinoline derivatives
    • Mital, A., Negi, V. S., & Ramachandran, U. (2006). Synthesis and antimycobacterial activities of certain trifluoromethyl-aminoquinoline derivatives. ARKIVOC, 2006(x), 220-227. (Pubitemid 43570425)
    • (2006) Arkivoc , vol.2006 , Issue.10 , pp. 220-227
    • Mital, A.1    Negi, V.S.2    Ramachandran, U.3
  • 15
    • 80052022193 scopus 로고    scopus 로고
    • Microwave-assisted synthesis of some new tetrazolo[1,5-a]quinoline-based benzimidazoles catalyzed by p-TsOH and investiga-tion of their antimicrobial activity
    • DOI: 10.1007/s00044-010-9388-0
    • Mungra, D. C., Patel, M. P., & Patel, R. G. (2011). Microwave-assisted synthesis of some new tetrazolo[1,5-a]quinoline-based benzimidazoles catalyzed by p-TsOH and investiga-tion of their antimicrobial activity Medicinal Chemistry Re-search, OnlineFirst. DOI: 10.1007/s00044-010- 9388-0.
    • (2011) Medicinal Chemistry Re-search, Online First
    • Mungra, D.C.1    Patel, M.P.2    Patel, R.G.3
  • 16
    • 77953177433 scopus 로고    scopus 로고
    • An efficient one-pot synthesis and in vitro antimicrobial activity of new pyridine derivatives bearing the tetrazoloquinoline nucleus
    • 2009
    • Mungra, D. C., Patel, M. P., & Patel, R. G. (2009). An efficient one-pot synthesis and in vitro antimicrobial activity of new pyridine derivatives bearing the tetrazoloquinoline nucleus. ARKIVOC, 2009(xiv), 64-74.
    • (2009) ARKIVOC , Issue.14 , pp. 64-74
    • Mungra, D.C.1    Patel, M.P.2    Patel, R.G.3
  • 17
    • 0012481773 scopus 로고    scopus 로고
    • National Committee for Clinical Laboratory Standards (NC-CLS) Twelfth Informational Supplement. NC-CLS document M100-S12. Wayne, PA, USA: NCCLS
    • National Committee for Clinical Laboratory Standards (NC-CLS) (2002). Performance standards for antimicrobial sus-ceptibility testing. Twelfth Informational Supplement. NC-CLS document M100-S12. Wayne, PA, USA: NCCLS.
    • (2002) Performance Standards for Antimicrobial Sus-ceptibility Testing
  • 18
    • 68149156203 scopus 로고    scopus 로고
    • Microwave-assisted synthesis of some new biquinoline compounds cat-alyzed by DMAP and their biological activities
    • Nirmal, J. P., Patel, M. P., & Patel, R. G. (2009). Microwave-assisted synthesis of some new biquinoline compounds cat-alyzed by DMAP and their biological activities. Indian Journal of Chemistry Section B, 48B, 712-717.
    • (2009) Indian Journal of Chemistry Section B , vol.48 B , pp. 712-717
    • Nirmal, J.P.1    Patel, M.P.2    Patel, R.G.3
  • 19
    • 0037598935 scopus 로고    scopus 로고
    • Synthesis and antimicrobial activity of some novel 2,5- and/or 6-substituted benzoxazole and benzimidazole derivatives
    • DOI: 10.1016/S0928-0987(98)00017-7
    • Oren, I., Temiz, O., Yaļcin, I., Şener, E., & Altanlar, N. (1998). Synthesis and antimicrobial activity of some novel 2,5- and/or 6-substituted benzoxazole and benzimidazole derivatives. European Journal of Pharmaceutical Sciences, 7, 153-160. DOI: 10.1016/S0928-0987(98)00017-7.
    • (1998) European Journal of Pharmaceutical Sciences , vol.7 , pp. 153-160
    • Oren, I.1    Temiz, O.2    Yaļcin, I.3    Şener, E.4    Altanlar, N.5
  • 20
    • 74949126821 scopus 로고    scopus 로고
    • Synthe-sis and antistaphylococcal activity of N-substituted-1H- benzimidazole-sulphonamides
    • DOI 10.1002/ardp.200900199
    • Püsküllü, M. O., Yildiz, S., & G̈oker, H. (2010). Synthe-sis and antistaphylococcal activity of N-substituted-1H-benzimidazole- sulphonamides. Archiv der Pharmazie, 343, 31-39. DOI 10.1002/ardp.200900199.
    • (2010) Archiv der Pharmazie , vol.343 , pp. 31-39
    • Püsküllü, M.O.1    Yildiz, S.2    G̈oker, H.3
  • 21
    • 45149147286 scopus 로고    scopus 로고
    • Scope and limitations of the T-reaction employing some functionalized C-H-acids and naturally oc-curring secondary amines
    • DOI: 10.3987/COM-07-11260
    • Rabong, C., Hametner, C., Mereiter, K., Kartsev, V. G., & Jordis, U. (2008). Scope and limitations of the T-reaction employing some functionalized C-H-acids and naturally oc-curring secondary amines. Heterocycles, 75, 799-838. DOI: 10.3987/COM-07-11260.
    • (2008) Heterocycles , vol.75 , pp. 799-838
    • Rabong, C.1    Hametner, C.2    Mereiter, K.3    Kartsev, V.G.4    Jordis, U.5
  • 22
    • 56049126667 scopus 로고    scopus 로고
    • Green Chemistry: Conventional and microwave induced synthesis of var-ious thiazolidinone derivatives from 3-{[(1E)-(2'-chloro-7'-methoxyquinoline-3'-yl) methylene]amino}-4-(substituted-phenyldiazenyl)phenol and their antimicrobial screening
    • 2008
    • Rana, P. B., Mistry, B. D., & Desai, K. R. (2008). Green Chemistry: conventional and microwave induced synthesis of var-ious thiazolidinone derivatives from 3-{[(1E)-(2'-chloro-7'-methoxyquinoline-3'-yl)methylene]amino}- 4-(substituted-phenyldiazenyl)phenol and their antimicrobial screening. ARKIVOC, 2008(xv), 262-279.
    • (2008) ARKIVOC , Issue.15 , pp. 262-279
    • Rana, P.B.1    Mistry, B.D.2    Desai, K.R.3
  • 23
    • 74849096664 scopus 로고    scopus 로고
    • One-pot, multicomponent condensation reaction in neutral conditions: Synthesis characterization, and biological studies of fused thiazolo[2,3-b] quinazolinone derivatives
    • DOI: 10.1080/10426500802583504
    • Shah, N. K., Patel, M. P., & Patel, R. G. (2009). One-pot, multicomponent condensation reaction in neutral conditions: Synthesis, characterization, and biological studies of fused thiazolo[2,3-b]quinazolinone derivatives. Phosphorus, Sulfur, and Silicon and the Related Elements, 184, 2704-2719. DOI: 10.1080/10426500802583504.
    • (2009) Phosphorus, Sulfur, and Silicon and the Related Elements , vol.184 , pp. 2704-2719
    • Shah, N.K.1    Patel, M.P.2    Patel, R.G.3
  • 24
    • 77950334736 scopus 로고    scopus 로고
    • Synthesis and antibacterial screen-ing of new 4-((5-(difluoromethoxy)-1H- benzo[d]imidazol-2-ylthio)methyl)-tetrazolo[1,5-a]quinoline derivatives
    • DOI: 10.1002/jhet. 340
    • Sonar, S. S., Sadaphal, S. A., Pokalwar, R. U., Shingate, B. B., & Shingare, M. S. (2010). Synthesis and antibacterial screen-ing of new 4-((5-(difluoromethoxy)-1H-benzo[d]imidazol-2-ylthio)methyl)-tetrazolo[1,5-a] quinoline derivatives. Journal of Heterocyclic Chemistry, 47, 441-445. DOI: 10.1002/jhet. 340.
    • (2010) Journal of Heterocyclic Chemistry , vol.47 , pp. 441-445
    • Sonar, S.S.1    Sadaphal, S.A.2    Pokalwar, R.U.3    Shingate, B.B.4    Shingare, M.S.5
  • 25
    • 33947416679 scopus 로고    scopus 로고
    • Synthesis and antibacterial activity of novel pyrazolo[3,4-b]quinoline based heterocyclic azo compounds and their dyeing performance
    • Thakor, S., Patel, D. M., Patel, M. P., & Patel, R. G. (2007). Synthesis and antibacterial activity of novel pyrazolo[3,4-b]quinoline based heterocyclic azo compounds and their dye-ing performance. Saudi Pharmaceutical Journal, 15, 48-54. (Pubitemid 46450508)
    • (2007) Saudi Pharmaceutical Journal , vol.15 , Issue.1 , pp. 48-54
    • Thakor, S.F.1    Patel, D.M.2    Patel, M.P.3    Patel, R.G.4
  • 26
    • 74849128697 scopus 로고    scopus 로고
    • Synthesis, charac-terization, and biological activity of substituted thiazole-5-carboxaldehydes and their ylidenenitriles derivatives
    • DOI: 10.1080/10426500802583520
    • Thumar, N. J., & Patel, M. P. (2009a). Synthesis, charac-terization, and biological activity of substituted thiazole-5-carboxaldehydes and their ylidenenitriles derivatives. Phos-phorus, Sulfur, and Silicon and the Related Elements, 184, 2720-2732. DOI: 10.1080/10426500802583520.
    • (2009) Phos-phorus, Sulfur, and Silicon and the Related Elements , vol.184 , pp. 2720-2732
    • Thumar, N.J.1    Patel, M.P.2
  • 27
    • 77953212666 scopus 로고    scopus 로고
    • Synthesis and in vitro antimicrobial evaluation of 4H-pyrazolopyran, -benzopyran and naphthopyran derivatives of 1H-pyrazole
    • 2009
    • Thumar, N. J., & Patel, M. P. (2009b). Synthesis and in vitro antimicrobial evaluation of 4H-pyrazolopyran, -benzopyran and naphthopyran derivatives of 1H-pyrazole. ARKIVOC, 2009(xiii), 363-380.
    • (2009) ARKIVOC , Issue.13 , pp. 363-380
    • Thumar, N.J.1    Patel, M.P.2


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