Synthesis and antistaphylococcal activity of N-substituted-1H- benzimidazole-sulphonamides

Archiv der Pharmazie

Volumn 343, Issue 1, 2010, Pages 31-39

  Püsküllü, M Orhan ^a   Yildiz, Sulhiye ^a   Göker, Hakan ^a  

^a ANKARA UNIVERSITY   (Turkey)

Author keywords

1H benzimidazolesulphonamide; Anti staphylococcal activity; Methicillin resistant Staphylococcus aureus; Tautomerism

Indexed keywords

1 BENZYL 2 (3,4 DICHLOROPHENYL) N [2 (DIMETHYLAMINO) ETHYL] 1H BENZIMIDAZOL 5 SULFONAMIDE; 1 BENZYL 2 [4 (4 CHLOROPHENOXY)PHENYL] N [2 (DIMETHYLAMINO)ETHYL] 1H BENZIMIDAZOL 5 SULFONAMIDE; 1 BENZYL N [2 (DIMETHYLAMINO)ETHYL] 2 (2,3,5 TRICHLOROPHENYL) 1H BENZIMIDAZOL 5 SULFONAMIDE; 2 (2,6 DICHLOROPHENYL) 1H BENZIMIDAZOL 5(6) SULFONIC ACID; 2 (3 TERT BUTYL 2 HYDROXYPHENYL) 1H BENZIMIDAZOL 5(6) CARBONITRILE; 2 (3 TERT BUTYL 2 HYDROXYPHENYL) 1H BENZIMIDAZOL 5(6) SULFONAMIDE; 2 (3 TERT BUTYL 2 HYDROXYPHENYL) 1H BENZIMIDAZOL 5(6) SULFONIC ACID; 2 (3 TERT BUTYL 2 HYDROXYPHENYL) N [2 (DIMETHYLAMINO)ETHYL] 1H BENZIMIDAZOL 5(6) SULFONAMIDE; 2 (3,4 DIBENZYLOXYPHENYL) N [2 (DIMETHYLAMINO)ETHYL] 1H BENZIMIDAZOL 5(6) SULFONAMIDE HYDROCHLORIDE; 2 (3,4 DICHLOROPHENYL) 1H BENZIMIDAZOL 5(6) SULFONAMIDE; 2 (3,4 DICHLOROPHENYL) 1H BENZIMIDAZOL 5(6) SULFONIC ACID; 2 (3,4 DICHLOROPHENYL) N [2 (DIMETHYLAMINO)ETHYL] 1H BENZIMIDAZOL 5(6) SULFONAMIDE; 2 (3,5 DI TERT BUTYL 2 HYDROXYPHENYL) 1H BENZIMIDAZOL 5(6) CARBONITRILE; 2 (3,5 DI TERT BUTYL 2 HYDROXYPHENYL) 1H BENZIMIDAZOL 5(6) CARBOXYLIC ACID; 2 (3,5 DI TERT BUTYL 2 HYDROXYPHENYL) 1H BENZIMIDAZOL 5(6) SULFONAMIDE; 2 (3,5 DI TERT BUTYL 2 HYDROXYPHENYL) N [2 (DIMETHYLAMINO)ETHYL] 1H BENZIMIDAZOL 5(6) SULFONAMIDE; 2 (4 (4 CHLOROPHENOXY)PHENYL) N [2 (DIMETHYLAMINO) ETHYL] 1H BENZIMIDAZOL 5(6) SULFONAMIDE; 2 [3,5 BIS(TRIFLUOROMETHYL)PHENYL] 1 BENZYL N [2 (DIMETHYLAMINO)ETHYL] 1H BENZIMIDAZOL 5 SULFONAMIDE; 2 [3,5 BIS(TRIFLUOROMETHYL)PHENYL] N [2 (DIMETHYLAMINO) ETHYL] 1H BENZIMIDAZOL 5(6) SULFONAMIDE; 3 AMINO 4 BENZYLAMINO N [2 (DIMETHYLAMINO)ETHYL]BENZENESULFONAMIDE; 3 NITRO 4 AMINOBENZENESULFONAMIDE; 3,4 DIAMINO N [2 (DIMETHYLAMINO)ETHYL]BENZENESULFONAMIDE; 3,4 DIAMINOBENZENESULFONAMIDE; 3,4 DIAMINOBENZENESULFONIC ACID; 4 AMINO 3 NITROBENZENESULFONIC ACID; 4 CHLORO 3 NITROBENZENESULFONIC ACID; ANTIINFECTIVE AGENT; BENZIMIDAZOLE DERIVATIVE; SULFONAMIDE; UNCLASSIFIED DRUG; UNINDEXED DRUG;

ANTIBACTERIAL ACTIVITY; ANTIFUNGAL ACTIVITY; ARTICLE; BACTERIAL GROWTH; BACTERIAL STRAIN; CANDIDA ALBICANS; CARBON NUCLEAR MAGNETIC RESONANCE; DRUG STRUCTURE; DRUG SYNTHESIS; ESCHERICHIA COLI; GROWTH INHIBITION; IN VITRO STUDY; METHICILLIN RESISTANT STAPHYLOCOCCUS AUREUS; MICROBIOLOGY; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; PRIORITY JOURNAL; PROTON NUCLEAR MAGNETIC RESONANCE; STAPHYLOCOCCUS AUREUS; STAPHYLOCOCCUS INFECTION;

ANTI-BACTERIAL AGENTS; BENZIMIDAZOLES; METHICILLIN-RESISTANT STAPHYLOCOCCUS AUREUS; MICROBIAL SENSITIVITY TESTS; STAPHYLOCOCCUS AUREUS; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONAMIDES;

EID: 74949126821     PISSN: 03656233     EISSN: 15214184     Source Type: Journal    
DOI: 10.1002/ardp.200900199     Document Type: Article

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