A selective, tin-free radical mediated synthesis of indoles based on a sulfonate template

Tetrahedron Letters

Volumn 53, Issue 1, 2012, Pages 41-44

  Gray, Vincent James ^a   Wilden, Jonathan D ^a  

^a UNIVERSITY COLLEGE LONDON   (United Kingdom)

Author keywords

Cyclisation; Indole; Radical; Sulfonate ester

Indexed keywords

ANILINE DERIVATIVE; INDOLE DERIVATIVE; SULFONIC ACID DERIVATIVE; UNCLASSIFIED DRUG; VINYLSULFONIC ACID;

ARTICLE; CHEMICAL ANALYSIS; CHEMICAL REACTION; CHEMICAL STRUCTURE; CYCLIZATION; DRUG SYNTHESIS;

EID: 82955167818     PISSN: 00404039     EISSN: 18733581     Source Type: Journal    
DOI: 10.1016/j.tetlet.2011.10.093     Document Type: Article

References (15)

1. V. Sharma, and D. Pathak J. Heterocycl. Chem. 47 2010 491
2. J.K. Sugden, and T.O. Yoloye Pharm. Acta Helv. 53 1978 65
3. J.A. Joule Indoles E.J. Thomas, Science of Synthesis Knowledge Update 2010/2 Vol. 10 2011 George Thieme Verlag, Stuttgart New York 526
4. G.W. Gribble J. Chem. Soc., Perkin Trans. 1 2000 1045
5. E. Hazai, P. Joshi, E.C. Skoviak, A. Suryanarayanan, M.K. Schulte, and Z. Bikadi Bioorg. Med. Chem. 17 2009 5796
6. A.S. Kalgutkar, B.C. Crews, S. Saleh, D. Prudhomme, and L.J. Marnett Bioorg. Med. Chem. 13 2005 6810
7. Y. Yamamoto, and M. Kurazono Bioorg. Med. Chem. Lett. 17 2007 1626
8. B. Robinson Chem. Rev. 63 1963 373
9. G. Bartoli, and R. Dalpozzo Tetrahedron Lett. 30 1989 2129
10. V. Chudasama, and J.D. Wilden Chem. Commun. 2008 3768
11. G. Aumaitre, J. Chanet-Ray, J. Durand, R. Vessire, and G. Lonchambon Synthesis 1983 816
12. J.A. Murphy, R. Tripoli, T.A. Khan, and U.W. Mali Org. Lett. 7 2005 3287
13. E.J. Corey, D.Y. Gin, and R.S. Kania J. Am. Chem. Soc. 118 1996 9202
14. H.T. Clarke, H.B. Gillespie, and S.Z. Weisshaus J. Am. Chem. Soc. 55 1933 4571
15. K.C. Majumdar, P.K. Basu, and S.K. Chattopadhyay Tetrahedron 63 2007 793