Fac-[TcO3(tacn)]+: A versatile precursor for the labelling of pharmacophores, amino acids and carbohydrates through a new ligand-centred labelling strategy

Chemistry - A European Journal

Volumn 17, Issue 46, 2011, Pages 12967-12974

  Braband, Henrik ^a   Tooyama, Yuji ^a   Fox, Thomas ^a   Simms, Ryan ^b   Forbes, John ^b   Valliant, John F ^b   Alberto, Roger ^a  

^a UNIVERSITY OF ZURICH   (Switzerland)

^b Centre for Probe Development and Commercialization   (Canada)

Author keywords

cycloaddition; glucose; imaging agents; radiopharmaceuticals; technetium

Indexed keywords

BIO-CONJUGATION; BIOCONJUGATES; BIODISTRIBUTIONS; BUILDING BLOCKES; CLINICAL TRANSLATION; CLIP-ON; CYCLOADDUCTS; GLUCOSE DERIVATIVES; IMAGING AGENTS; IN-VIVO; NEUTRAL PH; NON NATURAL AMINO ACIDS; PHARMACOPHORES; RADIOPHARMACEUTICALS; SPECIFIC FUNCTIONAL GROUPS;

AMINO ACIDS; CARBOHYDRATES; FUNCTIONAL GROUPS; GLUCOSE; HYDROPHILICITY; LIGANDS; NITROGEN OXIDES; SCAFFOLDS; TECHNETIUM;

PHARMACODYNAMICS;

AMINO ACID; DIAGNOSTIC AGENT; DRUG DERIVATIVE; GLUCOSE; RADIOPHARMACEUTICAL AGENT; TECHNETIUM COMPLEX;

ANIMAL; ARTICLE; CHEMICAL STRUCTURE; CHEMISTRY; CONFORMATION; DRUG SCREENING; MOUSE; SYNTHESIS;

AMINO ACIDS; ANIMALS; GLUCOSE; MICE; MOLECULAR CONFORMATION; MOLECULAR STRUCTURE; ORGANOTECHNETIUM COMPOUNDS; RADIOPHARMACEUTICALS; XENOGRAFT MODEL ANTITUMOR ASSAYS;

EID: 80555135880     PISSN: 09476539     EISSN: 15213765     Source Type: Journal    
DOI: 10.1002/chem.201101275     Document Type: Article

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