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Bioorganic and Medicinal Chemistry

Volumn 19, Issue 20, 2011, Pages 5999-6005

Inhibition of steroid sulfatase with 4-substituted estrone and estradiol derivatives

(5) Phan, Chau Minh a Liu, Yong a Kim, Byoung Moo a Mostafa, Yaser a Taylor, Scott D a

a UNIVERSITY OF WATERLOO (Canada)

Author keywords

Enzyme inhibitors; Hormone therapy; Steroid sulfatase

Indexed keywords

2 FORMYL 17ALPHA BENZYL 17BETA HYDROXYESTRA 1,3,5(10)TRIENE; 2,4 DIFORMYLESTRA 1,3,5(10)TRIENE 17 ONE; 4 ESTRONE; 4 FLUORO 17ALPHA BENZYL 17BETA HYDROXYESTRA 1,3,5(10)TRIENE; 4 FORMYL 2 BROMOESTRA 1,3,5(10)TRIENE 17 ONE; 4 FORMYL 2 NITROESTRA 1,3,5(10)TRIENE 17 ONE; ESTRA 1,3,5(10) TRIENE 17 ONE 3 CARBALDEHYDE; ESTRADIOL DERIVATIVE; ESTRONE DERIVATIVE; STERYL SULFATASE; UNCLASSIFIED DRUG;

ARTICLE; DRUG DETERMINATION; DRUG POTENCY; DRUG PROTEIN BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; ELECTRON; ENZYME INHIBITION; IC 50;

BREAST NEOPLASMS; ENZYME INHIBITORS; ESTRADIOL; ESTRONE; FEMALE; HUMANS; KINETICS; PLACENTA; PREGNANCY; STERYL-SULFATASE;

EID: 80053290725 PISSN: 09680896 EISSN: 14643391 Source Type: Journal
DOI: 10.1016/j.bmc.2011.08.046 Document Type: Article

Times cited : (26)

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