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Volumn 746, Issue , 2011, Pages 135-164

Radioligand binding methods for membrane preparations and intact cells

Author keywords

Affinity; Assay; Binding; Competition; G protein coupled receptor; Inhibition; Intact cell; Kinetic; Non specific binding; Radioligand; Radioreceptor; Rate constant; Receptor; Saturation

Indexed keywords

ALPHA 2B ADRENERGIC RECEPTOR; G PROTEIN COUPLED RECEPTOR; IODINE 125; NORADRENALIN; OZONE; PRAZOSIN;

EID: 80052792838     PISSN: 10643745     EISSN: None     Source Type: Book Series    
DOI: 10.1007/978-1-61779-126-0_8     Document Type: Article
Times cited : (20)

References (7)
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  • 2
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  • 3
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    • (1949) Ann. N. Y. Acad. Sci , vol.51 , pp. 660-672
    • Scatchard, G.1
  • 4
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    • Graphical method for the determination and presentation of binding parameters in a complex system
    • Rosenthal, H. E. (1967) Graphical method for the determination and presentation of binding parameters in a complex system. Anal. Biochem. 20, 525-532
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  • 5
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    • Jacobs, S., Chang, K. J. and Cuatrecasas, P. (1975) Estimation of hormone-receptor affinity by competitive displacement of labeled ligand: Effect of concentration of receptor and labeled ligand. Biochem. Biophys. Res. Commun. 66, 687-695
    • (1975) Biochem. Biophys. Res. Commun , vol.66 , pp. 687-695
    • Jacobs, S.1    Chang, K.J.2    Cuatrecasas, P.3
  • 6
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    • The power issue: Determination of kb or ki from ic50: A closer look at the cheng-prusoff equation, the schild plot and related power equations
    • Cheng, H. C. (2002) The power issue: Determination of KB or Ki from IC50: A closer look at the Cheng-Prusoff equation, the Schild plot and related power equations. J. Pharmacol. Toxicol. Methods 46, 61-71
    • (2002) J. Pharmacol. Toxicol. Methods , vol.46 , pp. 61-71
    • Cheng, H.C.1
  • 7
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    • Graphic presentation and analysis of inhibition data from ligand-binding experiments
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    • Bylund, D.B.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.