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Volumn 38, Issue 8, 2011, Pages 1426-1435

Comparison of biological stability and metabolism of CCK2 receptor targeting peptides, a collaborative project under COST BM0607

Author keywords

177Lu; CCK; Cholecystokinin receptor; Gastrin; In vitro stability; In vivo stability; Metabolism

Indexed keywords

1,4,7,10 TETRAAZACYCLODODECANE 1,4,7,10 TETRAACETIC ACID; CHOLECYSTOKININ B RECEPTOR; GASTRIN DERIVATIVE; PEPTIDE; RADIOLIGAND;

EID: 80052579110     PISSN: 16197070     EISSN: 16197089     Source Type: Journal    
DOI: 10.1007/s00259-011-1818-9     Document Type: Article
Times cited : (80)

References (26)
  • 2
    • 57349195981 scopus 로고    scopus 로고
    • Peptide-based probes for cancer imaging
    • Reubi JC, Maecke HR. Peptide-based probes for cancer imaging. J Nucl Med 2008;49(11):1735-8.
    • (2008) J Nucl Med , vol.49 , Issue.11 , pp. 1735-1738
    • Reubi, J.C.1    Maecke, H.R.2
  • 3
    • 0031945355 scopus 로고    scopus 로고
    • Targeting of cholecystokinin-B/gastrin receptors in vivo: Preclinical and initial clinical evaluation of the diagnostic and therapeutic potential of radiolabelled gastrin
    • DOI 10.1007/s002590050241
    • Behr TM, Jenner N, Radetzky S, Béhé M, Gratz S, Yücekent S, et al. Targeting of cholecystokinin-B/gastrin receptors in vivo: Preclinical and initial clinical evaluation of the diagnostic and therapeutic potential of radiolabelled gastrin. Eur J Nucl Med 1998;25:424-30. (Pubitemid 28211607)
    • (1998) European Journal of Nuclear Medicine , vol.25 , Issue.4 , pp. 424-430
    • Behr, T.M.1    Jenner, N.2    Radetzky, S.3    Behe, M.4    Gratz, S.5    Yucekent, S.6    Raue, F.7    Becker, W.8
  • 5
    • 0030902066 scopus 로고    scopus 로고
    • Cholecystokinin (CCK)-A and CCK-B/gastrin receptors in human tumors
    • Reubi JC, Schaer JC, Waser B. Cholecystokinin (CCK)-A and CCK-B/gastrin receptors in human tumors. Cancer Res 1997;57 (7):1377-86. (Pubitemid 27152565)
    • (1997) Cancer Research , vol.57 , Issue.7 , pp. 1377-1386
    • Reubi, J.C.1    Schaer, J.-C.2    Waser, B.3
  • 6
    • 0036231110 scopus 로고    scopus 로고
    • Cholecystokinin-B/gastrin receptor-targeting peptides for staging and therapy of medullary thyroid cancer and other cholecystokinin-B receptor-expressing malignancies
    • Behr TM, Béhé MP. Cholecystokinin-B/Gastrin receptor-targeting peptides for staging and therapy of medullary throid cancer and other cholecystokinin-B receptor-expressing malignancies. Semin Nucl Med 2002;32(2):97-109. (Pubitemid 34311076)
    • (2002) Seminars in Nuclear Medicine , vol.32 , Issue.2 , pp. 97-109
    • Behr, T.M.1    Behe, M.P.2
  • 11
    • 56249103484 scopus 로고    scopus 로고
    • Optimised labeling, preclinical and initial clinical aspects of CCK-2 receptor-targeting with 3 radiolabeled peptides
    • Breeman WA, Fröberg AC, de Blois E, van Gameren A, Melis M, de Jong M, et al. Optimised labeling, preclinical and initial clinical aspects of CCK-2 receptor-targeting with 3 radiolabeled peptides. Nucl Med Biol 2008;35(8):839-49.
    • (2008) Nucl Med Biol , vol.35 , Issue.8 , pp. 839-849
    • Breeman, W.A.1    Fröberg, A.C.2    De Blois, E.3    Van Gameren, A.4    Melis, M.5    De Jong, M.6
  • 12
    • 77951282548 scopus 로고    scopus 로고
    • Stabilized (111)In-labeled sCCK8 analogues for targeting CCK2-receptor positive tumors: Synthesis and evaluation
    • Roosenburg S, Laverman P, Joosten L, Eek A, Oyen WJ, de Jong M, et al. Stabilized (111)In-labeled sCCK8 analogues for targeting CCK2-receptor positive tumors: Synthesis and evaluation. Bioconjug Chem 2010;21(4):663-70.
    • (2010) Bioconjug Chem , vol.21 , Issue.4 , pp. 663-670
    • Roosenburg, S.1    Laverman, P.2    Joosten, L.3    Eek, A.4    Oyen, W.J.5    De Jong, M.6
  • 13
    • 0034915406 scopus 로고    scopus 로고
    • Radionuclide-labeled somatostatin analogues for diagnostic and therapeutic purposes in nonmedullary thyroid cancer
    • Görges R, Kahaly G, Müller-Brand J, Mäcke H, Roser HW, Bockisch A. Radionuclide-labeled somatostatin analogues for diagnostic and therapeutic purposes in nonmedullary thyroid cancer. Thyroid 2001;11(7):647-59. (Pubitemid 32701585)
    • (2001) Thyroid , vol.11 , Issue.7 , pp. 647-659
    • Gorges, R.1    Kahaly, G.2    Muller-Brand, J.3    Macke, H.4    Roser, H.W.5    Bockisch, A.6
  • 14
    • 4544229980 scopus 로고    scopus 로고
    • Design, synthesis and preclinical evaluation of radiolabeled peptides for diagnosis and therapy
    • DOI 10.2174/1381612043383511
    • Aloj L, Morelli G. Design, synthesis and preclinical evaluation of radiolabeled peptides for diagnosis and therapy. Curr Pharm Des 2004;10(24):3009-31. (Pubitemid 39214008)
    • (2004) Current Pharmaceutical Design , vol.10 , Issue.24 , pp. 3009-3031
    • Aloj, L.1    Morelli, G.2
  • 15
  • 19
    • 0035155042 scopus 로고    scopus 로고
    • Bifunctional chelators for therapeutic lanthanide radiopharmaceuticals
    • DOI 10.1021/bc000070v
    • Liu S, Edwards DS. Bifunctional chelators for therapeutic lanthanide radiopharmaceuticals. Bioconjug Chem 2001;12:7-34. (Pubitemid 32113652)
    • (2001) Bioconjugate Chemistry , vol.12 , Issue.1 , pp. 7-34
    • Liu, S.1    Edwards, S.D.2
  • 20
    • 52449093302 scopus 로고    scopus 로고
    • Macrocyclic chelator-coupled gastrin-based radiopharmaceuticals for targeting of gastrin receptorexpressing tumours
    • Good S, Walter MA, Waser B, Wang X, Müller-Brand J, Béhé MP, et al. Macrocyclic chelator-coupled gastrin-based radiopharmaceuticals for targeting of gastrin receptorexpressing tumours. Eur J Nucl Med Mol Imaging 2008;35 (10):1868-77.
    • (2008) Eur J Nucl Med Mol Imaging , vol.35 , Issue.10 , pp. 1868-1877
    • Good, S.1    Walter, M.A.2    Waser, B.3    Wang, X.4    Müller-Brand, J.5    Béhé, M.P.6
  • 21
    • 33745107170 scopus 로고    scopus 로고
    • Strategies to improve plasma half life time of peptide and protein drugs
    • DOI 10.1007/s00726-005-0289-3
    • Werle M, Bernkop-Schnürch A. Strategies to improve plasma half life time of peptide and protein drugs. Amino Acids 2006;30 (4):351-67. (Pubitemid 43886897)
    • (2006) Amino Acids , vol.30 , Issue.4 , pp. 351-367
    • Werle, M.1    Bernkop-Schnurch, A.2
  • 22
    • 0036257686 scopus 로고    scopus 로고
    • Converting a peptide into a drug: Strategies to improve stability and bioavailability
    • Adessi C, Soto C. Converting a peptide into a drug: Strategies to improve stability and bioavailability. Curr Med Chem 2002;9 (9):963-78. (Pubitemid 34498572)
    • (2002) Current Medicinal Chemistry , vol.9 , Issue.9 , pp. 963-978
    • Adessi, C.1    Soto, C.2
  • 23
    • 79551680701 scopus 로고    scopus 로고
    • Influence of biological assay conditions on stability assessment of radiometal-labelled peptides exemplified using a 177Lu-DOTA-minigastrin derivative
    • Ocak M, Helbok A, von Guggenberg E, Ozsoy Y, Kabasakal L, Kremser L, et al. Influence of biological assay conditions on stability assessment of radiometal-labelled peptides exemplified using a 177Lu-DOTA-minigastrin derivative. Nucl Med Biol 2011;38(2):171-9.
    • (2011) Nucl Med Biol , vol.38 , Issue.2 , pp. 171-179
    • Ocak, M.1    Helbok, A.2    Von Guggenberg, E.3    Ozsoy, Y.4    Kabasakal, L.5    Kremser, L.6
  • 24
    • 0030219801 scopus 로고    scopus 로고
    • Ectoenzymes as sites of peptide regulation
    • DOI 10.1016/0165-6147(96)10036-5
    • Konkoy CS, Davis TP. Ectoenzymes as sites of peptide regulation. Trends Pharmacol Sci 1996;17(8):288-94. (Pubitemid 26261893)
    • (1996) Trends in Pharmacological Sciences , vol.17 , Issue.8 , pp. 288-294
    • Konkoy, C.S.1    Davis, T.P.2
  • 26
    • 0022996585 scopus 로고
    • Phenethyl ester derivative analogues of the C-terminal tetrapeptide of gastrin as potent gastrin antagonists
    • DOI 10.1021/jm00161a012
    • Martinez J, Rodriguez M, Bali JP, Laur J. Phenethyl ester derivative analogues of the C-terminal tetrapeptide of gastrin as potent gastrin antagonists. J Med Chem 1986;29(11):2201-6. (Pubitemid 17182294)
    • (1986) Journal of Medicinal Chemistry , vol.29 , Issue.11 , pp. 2201-2206
    • Martinez, J.1    Rodriguez, M.2    Bali, J.-P.3    Laur, J.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.