메뉴 건너뛰기




Volumn 18, Issue 2, 2011, Pages 115-119

Sitamaquine as a putative antileishmanial drug candidate: From the mechanism of action to the risk of drug resistance

Author keywords

Aminoquinoline; Drug action; Leishmaniasis; Sitamaquine

Indexed keywords

LEISHMANIA DONOVANI;

EID: 80052050504     PISSN: 1252607X     EISSN: 17761042     Source Type: Journal    
DOI: 10.1051/parasite/2011182115     Document Type: Review
Times cited : (84)

References (29)
  • 1
    • 0020613394 scopus 로고
    • Activity of 8-aminoquinolines against Leishmania tropica within human macrophages in vitro
    • BERMAN J.D. & LEE L.S. Activity of 8-aminoquinolines against Leishmania tropica within human macrophages in vitro. American Journal of Tropical Medicine and Hygiene, 1983, 32, 753-759. (Pubitemid 13041002)
    • (1983) American Journal of Tropical Medicine and Hygiene , vol.32 , Issue.4 , pp. 753-759
    • Berman, J.D.1    Lee, L.S.2
  • 2
  • 3
    • 40749149204 scopus 로고    scopus 로고
    • Selection and phenotype characterisation of sitamaquine-resistant promastigotes of Leishmania donovani
    • DOI 10.1016/j.biopha.2007.12.006, PII S0753332207002892
    • BORIES C., COJEAN S., HUTEAU F. & LOISEAU P.M. Selection and phenotype characterisation of sitamaquine-resistant promastigotes of Leishmania donovani. Biomedicine and Pharmacotherapy, 2008, 62, 164-167. (Pubitemid 351381937)
    • (2008) Biomedicine and Pharmacotherapy , vol.62 , Issue.3 , pp. 164-167
    • Bories, C.1    Cojean, S.2    Huteau, F.3    Loiseau, P.M.4
  • 5
    • 3042555141 scopus 로고    scopus 로고
    • Leishmaniasis: Current situation and new perspectives
    • DOI 10.1016/j.cimid.2004.03.004, PII S0147957104000232
    • DESJEUX P. Leishmaniasis: current situation and new perspectives. Comparative Immunology, Microbiology and Infectious Diseases, 2004, 27, 305-318. (Pubitemid 38842803)
    • (2004) Comparative Immunology, Microbiology and Infectious Diseases , vol.27 , Issue.5 , pp. 305-318
    • Desjeux, P.1
  • 7
    • 33846410660 scopus 로고    scopus 로고
    • Interaction of sitamaquine with membrane lipids of Leishmania donovani promastigotes
    • DOI 10.1016/j.bbamem.2006.07.003, PII S0005273606002628
    • DUEÑAS-ROMERO A.M., LOISEAU P.M. & SAINT-PIERRE-CHAZALET M. Interaction of sitamaquine with membrane lipids of Leishmania donovani promastigotes. Biochimica et Biophysica Acta, 2007, 1768, 246-252. (Pubitemid 46138097)
    • (2007) Biochimica et Biophysica Acta - Biomembranes , vol.1768 , Issue.2 , pp. 246-252
    • Duenas-Romero, A.M.1    Loiseau, P.M.2    Saint-Pierre-Chazalet, M.3
  • 9
    • 33747033177 scopus 로고    scopus 로고
    • In-vitro and in-vivo studies on a topical formulation of sitamaquine dihydrochloride for cutaneous leishmaniasis
    • DOI 10.1211/jpp.58.8.0004
    • GARNIER T., BROWN M.B., LAWRENCE M.J. & CROFT S.L. In vitro and in vivo studies on a topical formulation of sitamaquine dihydrochloride for cutaneous leishmaniasis. Journal of Pharmacy and Pharmacology, 2006, 58, 1043-1054. (Pubitemid 44213636)
    • (2006) Journal of Pharmacy and Pharmacology , vol.58 , Issue.8 , pp. 1043-1054
    • Garnier, T.1    Brown, M.B.2    Lawrence, M.J.3    Croft, S.L.4
  • 13
    • 0021028292 scopus 로고
    • Fine-structural alterations in Leishmania tropica within human macrophages exposed to antileishmanial drugs in vitro
    • LANGRETH S.G., BERMAN J.D., RIORDAN G.P. & LEE L.S. Finestructure alterations in Leishmania tropica within macrophages exposed to antileishmanial drugs in vitro. Journal of Protozoology, 1983, 30, 555-561. (Pubitemid 14232617)
    • (1983) Journal of Protozoology , vol.30 , Issue.3 , pp. 555-561
    • Langreth, S.G.1    Berman, J.D.2    Riordan, G.P.3    Lee, L.S.4
  • 17
    • 33749338420 scopus 로고    scopus 로고
    • Development of miltefosine as an oral treatment for leishmaniasis
    • DOI 10.1016/j.trstmh.2006.02.010, PII S003592030600109X
    • SINDERMANN H. & ENGEL J. Development of miltefosine as an oral treatment for leishmaniasis. Transactions of the Royal Society of Tropical Medicine and Hygiene, 2006, 100 (Suppl 1), S17-S20. (Pubitemid 44490164)
    • (2006) Transactions of the Royal Society of Tropical Medicine and Hygiene , vol.100 , Issue.SUPPL. 1
    • Sindermann, H.1    Engel, J.2
  • 19
    • 33749336171 scopus 로고    scopus 로고
    • Treatment of New World cutaneous leishmaniasis with miltefosine
    • DOI 10.1016/j.trstmh.2006.02.022, PII S0035920306002112
    • SOTO J. & BERMAN J. Treatment of New World cutaneous leishmaniasis with miltefosine. Transactions of the Royal Society of Tropical Medicine and Hygiene, 2006, 100 (Suppl 1), S34-S40. (Pubitemid 44490170)
    • (2006) Transactions of the Royal Society of Tropical Medicine and Hygiene , vol.100 , Issue.SUPPL. 1
    • Soto, J.1    Berman, J.2
  • 20
    • 33845488153 scopus 로고    scopus 로고
    • Oral miltefosine to treat new world cutaneous leishmaniasis
    • DOI 10.1016/S1473-3099(06)70665-X, PII S147330990670665X
    • SOTO J. & TOLEDO J.T. Oral miltefosine to treat new world cutaneous leishmaniasis. Lancet Infectious Diseases, 2007, 7, 7. (Pubitemid 44917777)
    • (2007) Lancet Infectious Diseases , vol.7 , Issue.1 , pp. 7
    • Soto, J.1    Toledo, J.T.2
  • 22
    • 53349151814 scopus 로고    scopus 로고
    • New treatment approach in Indian visceral leishmaniasis: Single-dose liposomal amphotericin B followed by short-course oral miltefosine
    • SUNDAR S., RAI M., CHAKRAVARTY J., AGARWAL D., AGRAWAL N., VAILLANT M., OLLIARO P., MURRAY H.W. New treatment approach in Indian visceral leishmaniasis: single-dose liposomal amphotericin B followed by short-course oral miltefosine. Clinical Infectious Diseases, 2008, 47, 1000-1006.
    • (2008) Clinical Infectious Diseases , vol.47 , pp. 1000-1006
    • Sundar, S.1    Rai, M.2    Chakravarty, J.3    Agarwal, D.4    Agrawal, N.5    Vaillant, M.6    Olliaro, P.7    Murray, H.W.8
  • 23
    • 0021954199 scopus 로고
    • Metabolism of a potential 8-aminoquinoline antileishmanial drug in rat liver microsomes
    • THEOHARIDES A.D., CHUNG H., VELAZQUEZ H. Metabolism of a potential 8-aminoquinoline antileishmanial drug in rat liver microsomes. Biochemical Pharmacology, 1985, 34, 181-188. (Pubitemid 15153409)
    • (1985) Biochemical Pharmacology , vol.34 , Issue.2 , pp. 181-188
    • Theoharides, A.D.1    Chung, H.2    Velazquez, H.3
  • 25
    • 0026696590 scopus 로고
    • 2+, pentamidine and WR-6026 on mitochondrial membrane potential in situ
    • 2+, pentamidine and WR-6026 on mitochondrial membrane potential in situ. Biochemical Journal, 1992, 284, 463-467.
    • (1992) Biochemical Journal , vol.284 , pp. 463-467
    • Vercesi, A.1    Docampo, R.2
  • 26
    • 0034640341 scopus 로고    scopus 로고
    • + exchanger in acidocalcisomes of Leishmania donovani and their alkalization by anti-leishmanial drugs
    • DOI 10.1016/S0014-5793(00)01531-3, PII S0014579300015313
    • VERCESI A., RODRIGUES C., CASTISTI R. & DOCAMPO R. Presence of a Na(+)/H(+) exchanger in acidocalcisomes of Leishmania donovani and their alkalization by anti-leishmanial drugs. FEBS Letters, 2000, 473, 203-206. (Pubitemid 30254291)
    • (2000) FEBS Letters , vol.473 , Issue.2 , pp. 203-206
    • Vercesi, A.E.1    Rodrigues, C.O.2    Catisti, R.3    Docampo, R.4
  • 28
    • 85083142024 scopus 로고    scopus 로고
    • WORLD HEALTH ORGANIZATION. Leishmaniasis Disease Burden. Available from: http://www.who.int/leishmaniasis, 2010.
    • (2010) Leishmaniasis Disease Burden
  • 29
    • 0036782986 scopus 로고    scopus 로고
    • Sitamaquine (GlaxoSmithKline/Walter Reed Army Institute)
    • YEATES C. Sitamaquine (GlaxoSmithKline/Walter Reed Army Institute). Current Opinion in Investigational Drugs, 2002, 3, 1446-1452.
    • (2002) Current Opinion in Investigational Drugs , vol.3 , pp. 1446-1452
    • Yeates, C.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.