-
1
-
-
0020613394
-
Activity of 8-aminoquinolines against Leishmania tropica within human macrophages in vitro
-
BERMAN J.D. & LEE L.S. Activity of 8-aminoquinolines against Leishmania tropica within human macrophages in vitro. American Journal of Tropical Medicine and Hygiene, 1983, 32, 753-759. (Pubitemid 13041002)
-
(1983)
American Journal of Tropical Medicine and Hygiene
, vol.32
, Issue.4
, pp. 753-759
-
-
Berman, J.D.1
Lee, L.S.2
-
3
-
-
40749149204
-
Selection and phenotype characterisation of sitamaquine-resistant promastigotes of Leishmania donovani
-
DOI 10.1016/j.biopha.2007.12.006, PII S0753332207002892
-
BORIES C., COJEAN S., HUTEAU F. & LOISEAU P.M. Selection and phenotype characterisation of sitamaquine-resistant promastigotes of Leishmania donovani. Biomedicine and Pharmacotherapy, 2008, 62, 164-167. (Pubitemid 351381937)
-
(2008)
Biomedicine and Pharmacotherapy
, vol.62
, Issue.3
, pp. 164-167
-
-
Bories, C.1
Cojean, S.2
Huteau, F.3
Loiseau, P.M.4
-
4
-
-
78149476218
-
Mechanism of interaction of sitamaquine with Leishmania donovani
-
COÏMBRA E.S., LIBONG D., COJEAN S., SAINT-PIERRE-CHAZALET M., SOLGADI A., LE MOYEC L., DUENAS-ROMERO A.M., CHAMINADE P. & LOISEAU P.M. Mechanism of interaction of sitamaquine with Leishmania donovani. The Journal of Antimicrobial Chemotherapy, 2010, 65, 2548-2555.
-
(2010)
The Journal of Antimicrobial Chemotherapy
, vol.65
, pp. 2548-2555
-
-
Coïmbra, E.S.1
Libong, D.2
Cojean, S.3
Saint-Pierre-Chazalet, M.4
Solgadi, A.5
Le Moyec, L.6
Duenas-Romero, A.M.7
Chaminade, P.8
Loiseau, P.M.9
-
5
-
-
3042555141
-
Leishmaniasis: Current situation and new perspectives
-
DOI 10.1016/j.cimid.2004.03.004, PII S0147957104000232
-
DESJEUX P. Leishmaniasis: current situation and new perspectives. Comparative Immunology, Microbiology and Infectious Diseases, 2004, 27, 305-318. (Pubitemid 38842803)
-
(2004)
Comparative Immunology, Microbiology and Infectious Diseases
, vol.27
, Issue.5
, pp. 305-318
-
-
Desjeux, P.1
-
6
-
-
0035687445
-
Phase 2 trial of WR6026, an orally administered 8-aminoquinoline, in the treatment of visceral leishmaniasis caused by Leishmania chagasi
-
DIETZE R., CARVALHO S.F.G., VALLI L.C., BERMAN J., BREWER T., MILHOUS W., SANCHEZ J., SCHUSTER B. & GROGL M. Phase II trial of WR6026, an orally administrated 8-aminoquinoline, in the treatment of visceral leishmaniasis caused by Leishmania chagasi. American Journal of Tropical Medicine and Hygiene, 2001, 65, 685-689. (Pubitemid 34049456)
-
(2001)
American Journal of Tropical Medicine and Hygiene
, vol.65
, Issue.6
, pp. 685-689
-
-
Dietze, R.1
Carvalho, S.F.G.2
Valli, L.C.3
Berman, J.4
Brewer, T.5
Milhous, W.6
Sanchez, J.7
Schuster, B.8
Grogl, M.9
-
7
-
-
33846410660
-
Interaction of sitamaquine with membrane lipids of Leishmania donovani promastigotes
-
DOI 10.1016/j.bbamem.2006.07.003, PII S0005273606002628
-
DUEÑAS-ROMERO A.M., LOISEAU P.M. & SAINT-PIERRE-CHAZALET M. Interaction of sitamaquine with membrane lipids of Leishmania donovani promastigotes. Biochimica et Biophysica Acta, 2007, 1768, 246-252. (Pubitemid 46138097)
-
(2007)
Biochimica et Biophysica Acta - Biomembranes
, vol.1768
, Issue.2
, pp. 246-252
-
-
Duenas-Romero, A.M.1
Loiseau, P.M.2
Saint-Pierre-Chazalet, M.3
-
8
-
-
0001606801
-
Synthesis of primaquine and certain of its analogs
-
ELDERFIELD R.C., MERTEL H.E., MITCH R.T., WEMPEN I.M. & WERBLE E.J. Synthesis of primaquine and certain of its analogs. Journal of the American Chemical Society, 1955, 77, 4816-4819.
-
(1955)
Journal of the American Chemical Society
, vol.77
, pp. 4816-4819
-
-
Elderfield, R.C.1
Mertel, H.E.2
Mitch, R.T.3
Wempen, I.M.4
Werble, E.J.5
-
9
-
-
33747033177
-
In-vitro and in-vivo studies on a topical formulation of sitamaquine dihydrochloride for cutaneous leishmaniasis
-
DOI 10.1211/jpp.58.8.0004
-
GARNIER T., BROWN M.B., LAWRENCE M.J. & CROFT S.L. In vitro and in vivo studies on a topical formulation of sitamaquine dihydrochloride for cutaneous leishmaniasis. Journal of Pharmacy and Pharmacology, 2006, 58, 1043-1054. (Pubitemid 44213636)
-
(2006)
Journal of Pharmacy and Pharmacology
, vol.58
, Issue.8
, pp. 1043-1054
-
-
Garnier, T.1
Brown, M.B.2
Lawrence, M.J.3
Croft, S.L.4
-
10
-
-
0033540005
-
Miltefosine, an oral agent, for the treatment of Indian visceral leishmaniasis
-
JHA T.K., SUNDAR S., THAKUR C.P., BACHMANN P., KARBWANG J., FISCHER C., VOSS A. & BERMAN J. Miltefosine, an oral agent, for the treatment of Indian visceral leishmaniasis. New England Journal of Medicine, 1999, 341, 1795-800.
-
(1999)
New England Journal of Medicine
, vol.341
, pp. 1795-1800
-
-
Jha, T.K.1
Sundar, S.2
Thakur, C.P.3
Bachmann, P.4
Karbwang, J.5
Fischer, C.6
Voss, A.7
Berman, J.8
-
11
-
-
29844441606
-
A phase II dose-ranging study of sitamaquine for the treatment of visceral leishmaniasis in India
-
JHA T.K., SUNDAR S., THAKUR C.P., FELTON J.M., SABIN A.J. & HORTON J. A phase II dose-ranging study of sitamaquine for treatment of visceral leishmaniasis in India. American Journal of Tropical Medicine and Hygiene, 2005, 73, 1005-1011. (Pubitemid 43038244)
-
(2005)
American Journal of Tropical Medicine and Hygiene
, vol.73
, Issue.6
, pp. 1005-1011
-
-
Jha, T.K.1
Sundar, S.2
Thakur, C.P.3
Felton, J.M.4
Sabin, A.J.5
Horton, J.6
-
12
-
-
0018099010
-
The antileishmanial activity of lepidines
-
KINNAMON K.E., STECK E.A., LOIZEAUX P.S., HANSON W.L., CHAPMAN W.L. JR. & WAITS V.B. The antileishmanial activity of lepidines. American Journal of Tropical Medicine and Hygiene, 1978, 27, 751-757. (Pubitemid 8398077)
-
(1978)
American Journal of Tropical Medicine and Hygiene
, vol.27
, Issue.4
, pp. 751-757
-
-
Kinnamon, K.E.1
Steck, E.A.2
Loizeaux, P.S.3
-
13
-
-
0021028292
-
Fine-structural alterations in Leishmania tropica within human macrophages exposed to antileishmanial drugs in vitro
-
LANGRETH S.G., BERMAN J.D., RIORDAN G.P. & LEE L.S. Finestructure alterations in Leishmania tropica within macrophages exposed to antileishmanial drugs in vitro. Journal of Protozoology, 1983, 30, 555-561. (Pubitemid 14232617)
-
(1983)
Journal of Protozoology
, vol.30
, Issue.3
, pp. 555-561
-
-
Langreth, S.G.1
Berman, J.D.2
Riordan, G.P.3
Lee, L.S.4
-
14
-
-
55849137267
-
Sitamaquine sensitivity in Leishmania species is not mediated by drug accumulation in acidocalcisomes
-
LÓPEZ-MARTÍN C., PÉREZ-VICTORIA J.M., CARVALHO L., CASTANYS S. & GAMARRO F. Sitamaquine sensitivity in Leishmania species is not mediated by drug accumulation in acidocalcisomes. Antimicrobial Agents and Chemotherapy, 2008, 52, 4030-4036.
-
(2008)
Antimicrobial Agents and Chemotherapy
, vol.52
, pp. 4030-4036
-
-
López-Martín, C.1
Pérez-Victoria, J.M.2
Carvalho, L.3
Castanys, S.4
Gamarro, F.5
-
15
-
-
0023492646
-
Alkyl phosphocholines: Toxicity and anticancer properties
-
DOI 10.1007/BF02535558
-
MUSCHIOL C., BERGER M.R., SCHULER B., SCHERF H.R., GARZON F.T., ZELLER W.J., UNGER C., EIBL H.J. & SCHMÄHL D. Alkyl phosphocholines: toxicity and anticancer properties. Lipids, 1987, 22, 930-934. (Pubitemid 18001400)
-
(1987)
Lipids
, vol.22
, Issue.11
, pp. 930-934
-
-
Muschiol, C.1
Berger, M.R.2
Schuler, B.3
Scherf, H.R.4
Garzon, F.T.5
Zeller, W.J.6
Unger, C.7
Eibl, H.J.8
Schmahl, D.9
-
16
-
-
0027948991
-
Phase 2 efficacy trial of an oral 8-aminoquinoline (WR6026) for treatment of visceral leishmaniasis
-
SHERWOOD J.A., GACHIHI G.S., MUIGAI R.K., SKILLMAN D.R., MUGO M., RASHID J.R., WASUNNA K.M., WERE J.B., KASILI S.K., MBUGUA J.M. ET AL. Phase II efficacy trial of an oral 8-aminoquinoline (WR6026) for treatment of visceral leishmaniasis. Clinical Infectious Diseases, 1994, 19, 1034-1039. (Pubitemid 24380014)
-
(1994)
Clinical Infectious Diseases
, vol.19
, Issue.6
, pp. 1034-1039
-
-
Sherwood, J.A.1
Gachihi, G.S.2
Muigai, R.K.3
Skillman, D.R.4
Mugo, M.5
Rashid, J.R.6
Wasunna, K.M.A.7
Were, J.B.O.8
Kasili, S.K.9
Mbugua, J.M.10
Kirigi, G.11
Schaefer, K.U.12
Oster, C.N.13
Fleckenstein, L.L.14
Berman, J.D.15
Brewer, T.G.16
Roberts, C.R.17
Johnson, A.J.18
Schuster, B.G.19
-
17
-
-
33749338420
-
Development of miltefosine as an oral treatment for leishmaniasis
-
DOI 10.1016/j.trstmh.2006.02.010, PII S003592030600109X
-
SINDERMANN H. & ENGEL J. Development of miltefosine as an oral treatment for leishmaniasis. Transactions of the Royal Society of Tropical Medicine and Hygiene, 2006, 100 (Suppl 1), S17-S20. (Pubitemid 44490164)
-
(2006)
Transactions of the Royal Society of Tropical Medicine and Hygiene
, vol.100
, Issue.SUPPL. 1
-
-
Sindermann, H.1
Engel, J.2
-
18
-
-
2342538350
-
Miltefosine for new world cutaneous leishmaniasis
-
DOI 10.1086/383321
-
SOTO J., ARANA B.A., TOLEDO J., RIZZO N., VEGA J.C., DIAZ A., LUZ M., GUTIERREZ P., ARBOLEDA M., BERMAN J.D., JUNGE K., ENGEL J. & SINDERMANN H. Miltefosine for new world cutaneous leishmaniasis. Clinical Infectious Diseases, 2004, 38, 1266-1272. (Pubitemid 38608569)
-
(2004)
Clinical Infectious Diseases
, vol.38
, Issue.9
, pp. 1266-1272
-
-
Soto, J.1
Arana, B.A.2
Tolado, J.3
Rizzo, N.4
Vega, J.C.5
Diaz, A.6
Luz, M.7
Gutierrez, P.8
Arboleda, M.9
Berman, J.D.10
Junge, K.11
Engel, J.12
Sindermann, H.13
-
19
-
-
33749336171
-
Treatment of New World cutaneous leishmaniasis with miltefosine
-
DOI 10.1016/j.trstmh.2006.02.022, PII S0035920306002112
-
SOTO J. & BERMAN J. Treatment of New World cutaneous leishmaniasis with miltefosine. Transactions of the Royal Society of Tropical Medicine and Hygiene, 2006, 100 (Suppl 1), S34-S40. (Pubitemid 44490170)
-
(2006)
Transactions of the Royal Society of Tropical Medicine and Hygiene
, vol.100
, Issue.SUPPL. 1
-
-
Soto, J.1
Berman, J.2
-
20
-
-
33845488153
-
Oral miltefosine to treat new world cutaneous leishmaniasis
-
DOI 10.1016/S1473-3099(06)70665-X, PII S147330990670665X
-
SOTO J. & TOLEDO J.T. Oral miltefosine to treat new world cutaneous leishmaniasis. Lancet Infectious Diseases, 2007, 7, 7. (Pubitemid 44917777)
-
(2007)
Lancet Infectious Diseases
, vol.7
, Issue.1
, pp. 7
-
-
Soto, J.1
Toledo, J.T.2
-
21
-
-
0037191710
-
Oral miltefosine for Indian visceral leishmaniasis
-
DOI 10.1056/NEJMoa021556
-
SUNDAR S., JHA T.K., THAKUR C.P., ENGEL J., SINDERMANN H., FISCHER C., JUNGE K., BRYCESON A. & BERMAN J. Oral miltefosine for Indian visceral leishmaniasis. New England Journal of Medicine, 2002, 347, 1739-1746. (Pubitemid 35375612)
-
(2002)
New England Journal of Medicine
, vol.347
, Issue.22
, pp. 1739-1746
-
-
Sundar, S.1
Jha, T.K.2
Thakur, C.P.3
Engel, J.4
Sindermann, H.5
Fischer, C.6
Junge, K.7
Bryceson, A.8
Berman, J.9
-
22
-
-
53349151814
-
New treatment approach in Indian visceral leishmaniasis: Single-dose liposomal amphotericin B followed by short-course oral miltefosine
-
SUNDAR S., RAI M., CHAKRAVARTY J., AGARWAL D., AGRAWAL N., VAILLANT M., OLLIARO P., MURRAY H.W. New treatment approach in Indian visceral leishmaniasis: single-dose liposomal amphotericin B followed by short-course oral miltefosine. Clinical Infectious Diseases, 2008, 47, 1000-1006.
-
(2008)
Clinical Infectious Diseases
, vol.47
, pp. 1000-1006
-
-
Sundar, S.1
Rai, M.2
Chakravarty, J.3
Agarwal, D.4
Agrawal, N.5
Vaillant, M.6
Olliaro, P.7
Murray, H.W.8
-
23
-
-
0021954199
-
Metabolism of a potential 8-aminoquinoline antileishmanial drug in rat liver microsomes
-
THEOHARIDES A.D., CHUNG H., VELAZQUEZ H. Metabolism of a potential 8-aminoquinoline antileishmanial drug in rat liver microsomes. Biochemical Pharmacology, 1985, 34, 181-188. (Pubitemid 15153409)
-
(1985)
Biochemical Pharmacology
, vol.34
, Issue.2
, pp. 181-188
-
-
Theoharides, A.D.1
Chung, H.2
Velazquez, H.3
-
24
-
-
84855284850
-
Identification and quantification of human urinary metabolites of a candidate 8-aminoquinoline antileishmanial drug WR-6026
-
THEOHARIDES A.D., KIM M.M., ASHMORE R.W. & SHIPLEY L.A. Identification and quantification of human urinary metabolites of a candidate 8-aminoquinoline antileishmanial drug WR-6026. Proceedings of American Society of Experimental Biology, 1987, 46, 865.
-
(1987)
Proceedings of American Society of Experimental Biology
, vol.46
, pp. 865
-
-
Theoharides, A.D.1
Kim, M.M.2
Ashmore, R.W.3
Shipley, L.A.4
-
25
-
-
0026696590
-
2+, pentamidine and WR-6026 on mitochondrial membrane potential in situ
-
2+, pentamidine and WR-6026 on mitochondrial membrane potential in situ. Biochemical Journal, 1992, 284, 463-467.
-
(1992)
Biochemical Journal
, vol.284
, pp. 463-467
-
-
Vercesi, A.1
Docampo, R.2
-
26
-
-
0034640341
-
+ exchanger in acidocalcisomes of Leishmania donovani and their alkalization by anti-leishmanial drugs
-
DOI 10.1016/S0014-5793(00)01531-3, PII S0014579300015313
-
VERCESI A., RODRIGUES C., CASTISTI R. & DOCAMPO R. Presence of a Na(+)/H(+) exchanger in acidocalcisomes of Leishmania donovani and their alkalization by anti-leishmanial drugs. FEBS Letters, 2000, 473, 203-206. (Pubitemid 30254291)
-
(2000)
FEBS Letters
, vol.473
, Issue.2
, pp. 203-206
-
-
Vercesi, A.E.1
Rodrigues, C.O.2
Catisti, R.3
Docampo, R.4
-
27
-
-
28044436746
-
A phase II dose-increasing study of sitamaquine for the treatment of visceral leishmaniasis in Kenya
-
WASUNNA M.K., RHASHID J.R., MBUI J., KIRIGI G., KINOTI D., LODENYO H., FELTON J.M., SABIN A.J. & HORTON J. A phase II dose-increasing study of sitamaquine for treatment of visceral leishmaniasis in Kenya. American Journal of Tropical Medicine and Hygiene, 2005, 73, 871-876. (Pubitemid 41688461)
-
(2005)
American Journal of Tropical Medicine and Hygiene
, vol.73
, Issue.5
, pp. 871-876
-
-
Wasunna, M.K.1
Rashid, J.R.2
Mbui, J.3
Kirigi, G.4
Kinoti, D.5
Lodenyo, H.6
Felton, J.M.7
Sabin, A.J.8
Horton, J.9
-
28
-
-
85083142024
-
-
WORLD HEALTH ORGANIZATION. Leishmaniasis Disease Burden. Available from: http://www.who.int/leishmaniasis, 2010.
-
(2010)
Leishmaniasis Disease Burden
-
-
-
29
-
-
0036782986
-
Sitamaquine (GlaxoSmithKline/Walter Reed Army Institute)
-
YEATES C. Sitamaquine (GlaxoSmithKline/Walter Reed Army Institute). Current Opinion in Investigational Drugs, 2002, 3, 1446-1452.
-
(2002)
Current Opinion in Investigational Drugs
, vol.3
, pp. 1446-1452
-
-
Yeates, C.1
|