메뉴 건너뛰기




Volumn 65, Issue 10, 2011, Pages 1113-1117

Assessing the sensitivity of [11C]p943, a novel 5-HTIB radioligand, to endogenous serotonin release

Author keywords

5HT1B; 11C P943; Nonhuman primate; PET; Serotonin

Indexed keywords

FENFLURAMINE; P 943; P 943 C 11; RADIOLIGAND; SEROTONIN; SEROTONIN 1B RECEPTOR; UNCLASSIFIED DRUG; 1 (4 (2 METHOXYISOPROPYL)PHENYL) 3 (2 (4 METHYLPIPERAZIN 1 YL)BENZYL)PYRROLIDIN 2 ONE; 1-(4-(2-METHOXYISOPROPYL)PHENYL)-3-(2-(4-METHYLPIPERAZIN-1-YL)BENZYL)PYRROLIDIN-2-ONE; 2 PYRROLIDONE DERIVATIVE; CARBON; DIAGNOSTIC AGENT; LIGAND; PIPERAZINE DERIVATIVE; SEROTONIN ANTAGONIST;

EID: 79960959970     PISSN: 08874476     EISSN: 10982396     Source Type: Journal    
DOI: 10.1002/syn.20942     Document Type: Article
Times cited : (19)

References (28)
  • 3
    • 0033729024 scopus 로고    scopus 로고
    • PET physiological measurements using constant infusion
    • Carson RE. 2000. PET physiological measurements using constant infusion. Nucl Med Biol 27: 657-660.
    • (2000) Nucl Med Biol , vol.27 , pp. 657-660
    • Carson, R.E.1
  • 5
    • 0026005750 scopus 로고
    • Rapid serotonin depletion as a provocative challenge test for patients with major depression: Relevance to antidepressant action and the neurobiology of depression
    • Delgado PL, Price LH, Miller HL, Salomon RM, Licinio J, Krystal JH, Heninger GR, Charney DS. 1991. Rapid serotonin depletion as a provocative challenge test for patients with major depression: Relevance to antidepressant action and the neurobiology of depression. Psychopharmacol Bull 27: 321-330.
    • (1991) Psychopharmacol Bull , vol.27 , pp. 321-330
    • Delgado, P.L.1    Price, L.H.2    Miller, H.L.3    Salomon, R.M.4    Licinio, J.5    Krystal, J.H.6    Heninger, G.R.7    Charney, D.S.8
  • 7
    • 77953860552 scopus 로고    scopus 로고
    • Fenfluramine-induced serotonin release decreases [11C]AZ10419369 binding to 5-HT1B-receptors in the primate brain
    • Finnema SJ, Varrone A, Hwang TJ, Gulyas B, Pierson ME, Halldin C, Farde L. 2010. Fenfluramine-induced serotonin release decreases [11C]AZ10419369 binding to 5-HT1B-receptors in the primate brain. Synapse 64: 573-577.
    • (2010) Synapse , vol.64 , pp. 573-577
    • Finnema, S.J.1    Varrone, A.2    Hwang, T.J.3    Gulyas, B.4    Pierson, M.E.5    Halldin, C.6    Farde, L.7
  • 10
    • 25144447427 scopus 로고    scopus 로고
    • Synthesis of potent and selective serotonin 5-HT1B receptor ligands
    • Huang Y, Bae SA, Roth BL, Laruelle M. 2005. Synthesis of potent and selective serotonin 5-HT1B receptor ligands. Bioorg Med Chem Lett 15: 4786-4789.
    • (2005) Bioorg Med Chem Lett , vol.15 , pp. 4786-4789
    • Huang, Y.1    Bae, S.A.2    Roth, B.L.3    Laruelle, M.4
  • 14
    • 0034018859 scopus 로고    scopus 로고
    • Imaging synaptic neurotransmission with in vivo binding competition techniques: A critical review
    • Laruelle M. 2000. Imaging synaptic neurotransmission with in vivo binding competition techniques: A critical review. J Cereb Blood Flow Metab 20: 423-451.
    • (2000) J Cereb Blood Flow Metab , vol.20 , pp. 423-451
    • Laruelle, M.1
  • 16
    • 0026546675 scopus 로고
    • Mouse 5HT1B serotonin receptor: Cloning, functional expression, and localization in motor control centers
    • Maroteaux L, Saudou F, Amlaiky N, Boschert U, Plassat JL, Hen R. 1992. Mouse 5HT1B serotonin receptor: Cloning, functional expression, and localization in motor control centers. Proc Natl Acad Sci USA 89: 3020-3024.
    • (1992) Proc Natl Acad Sci USA , vol.89 , pp. 3020-3024
    • Maroteaux, L.1    Saudou, F.2    Amlaiky, N.3    Boschert, U.4    Plassat, J.L.5    Hen, R.6
  • 17
    • 0032983836 scopus 로고    scopus 로고
    • The effects of single dose nefazodone and paroxetine upon 5-HT2A binding potential in humans using [18F]-setoperone PET
    • Meyer JH, Cho R, Kennedy S, Kapur S. 1999. The effects of single dose nefazodone and paroxetine upon 5-HT2A binding potential in humans using [18F]-setoperone PET. Psychopharmacology (Berl) 144: 279-281.
    • (1999) Psychopharmacology (Berl) , vol.144 , pp. 279-281
    • Meyer, J.H.1    Cho, R.2    Kennedy, S.3    Kapur, S.4
  • 20
    • 77957718322 scopus 로고    scopus 로고
    • Measuring endogenous 5-HT release by emission tomography: Promises and pitfalls
    • Paterson LM, Tyacke RJ, Nutt DJ, Knudsen GM. 2010. Measuring endogenous 5-HT release by emission tomography: Promises and pitfalls. J Cereb Blood Flow Metab 30: 1682-1706.
    • (2010) J Cereb Blood Flow Metab , vol.30 , pp. 1682-1706
    • Paterson, L.M.1    Tyacke, R.J.2    Nutt, D.J.3    Knudsen, G.M.4
  • 21
    • 0036121286 scopus 로고    scopus 로고
    • Serotonin releasing agents. Neurochemical, therapeutic and adverse effects
    • Rothman RB, Baumann MH. 2002. Serotonin releasing agents. Neurochemical, therapeutic and adverse effects. Pharmacol Biochem Behav 71: 825-836.
    • (2002) Pharmacol Biochem Behav , vol.71 , pp. 825-836
    • Rothman, R.B.1    Baumann, M.H.2
  • 22
    • 70450203483 scopus 로고    scopus 로고
    • The 5-HT1B receptor: A novel target for the pathophysiology of depression
    • Ruf BM, Bhagwagar Z. 2009. The 5-HT1B receptor: A novel target for the pathophysiology of depression. Curr Drug Targets 10: 1118-1138.
    • (2009) Curr Drug Targets , vol.10 , pp. 1118-1138
    • Ruf, B.M.1    Bhagwagar, Z.2
  • 23
    • 7444254932 scopus 로고    scopus 로고
    • Serotonin1B receptors: From protein to physiological function and behavior
    • Sari Y. 2004. Serotonin1B receptors: From protein to physiological function and behavior. Neurosci Biobehav Rev 28: 565-582.
    • (2004) Neurosci Biobehav Rev , vol.28 , pp. 565-582
    • Sari, Y.1
  • 24
    • 0032890427 scopus 로고    scopus 로고
    • Cellular and subcellular localization of 5-hydroxytryptamine1B receptors in the rat central nervous system: Immunocytochemical, autoradiographic and lesion studies
    • Sari Y, Miquel MC, Brisorgueil MJ, Ruiz G, Doucet E, Hamon M, Verge D. 1999. Cellular and subcellular localization of 5-hydroxytryptamine1B receptors in the rat central nervous system: Immunocytochemical, autoradiographic and lesion studies. Neuroscience 88: 899-915.
    • (1999) Neuroscience , vol.88 , pp. 899-915
    • Sari, Y.1    Miquel, M.C.2    Brisorgueil, M.J.3    Ruiz, G.4    Doucet, E.5    Hamon, M.6    Verge, D.7
  • 28
    • 0036323990 scopus 로고    scopus 로고
    • Effect of endogenous serotonin on the binding of the 5-hT1A PET ligand 18F-MPPF in the rat hippocampus: Kinetic beta measurements combined with microdialysis
    • Zimmer L, Mauger G, Le Bars D, Bonmarchand G, Luxen A, Pujol JF. 2002. Effect of endogenous serotonin on the binding of the 5-hT1A PET ligand 18F-MPPF in the rat hippocampus: Kinetic beta measurements combined with microdialysis. J Neurochem 80: 278-286.
    • (2002) J Neurochem , vol.80 , pp. 278-286
    • Zimmer, L.1    Mauger, G.2    Le Bars, D.3    Bonmarchand, G.4    Luxen, A.5    Pujol, J.F.6


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.