Structure-activity relationship studies of HIV-1 integrase oligonucleotide inhibitors

ACS Medicinal Chemistry Letters

Volumn 2, Issue 7, 2011, Pages 532-537

  Agapkina, Julia ^a   Zatsepin, Timofei ^a,b   Knyazhanskaya, Ekaterina ^a   Mouscadet, Jean Francois ^c   Gottikh, Marina ^a  

^a MOSCOW STATE UNIVERSITY   (Russian Federation)

^b CENTRAL RESEARCH INSTITUTE OF EPIDEMIOLOGY   (Russian Federation)

^c Ecole Normale Superieure de Cachan   (France)

Author keywords

HIV 1 integrase; inhibitor; oligonucleotide conjugate; xanthene

Indexed keywords

ANTI HUMAN IMMUNODEFICIENCY VIRUS AGENT; INTEGRASE INHIBITOR; OLIGONUCLEOTIDE;

ANTIVIRAL ACTIVITY; ARTICLE; CONTROLLED STUDY; DRUG SYNTHESIS; HUMAN IMMUNODEFICIENCY VIRUS 1 INFECTION; HYDROPHOBICITY; IC 50; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION;

HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 79960386339     PISSN: None     EISSN: 19485875     Source Type: Journal    
DOI: 10.1021/ml200066k     Document Type: Article

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