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Volumn 38, Issue 5, 2011, Pages 645-651

Fully automated one-pot radiosynthesis of O-(2-[18F]fluoroethyl)-l-tyrosine on the TracerLab FXFN module

Author keywords

18F FET; Amino acids; Automated radiosynthesis; Nucleophilic 18F fluorination; TracerLab FXFN

Indexed keywords

ACETONITRILE; CRYPTAND 2.2.2; FLUOROETHYLTYROSINE F 18; HYDROCHLORIC ACID; POTASSIUM CARBONATE; RADIOPHARMACEUTICAL AGENT; UNCLASSIFIED DRUG;

EID: 79959656783     PISSN: 09698051     EISSN: 18729614     Source Type: Journal    
DOI: 10.1016/j.nucmedbio.2011.01.001     Document Type: Article
Times cited : (39)

References (14)
  • 1
    • 0032616268 scopus 로고    scopus 로고
    • Pitfalls in oncologic diagnosis with FDG PET imaging: physiologic and benign variants
    • Shreve P.D., Anzai Y., Wabl R.L. Pitfalls in oncologic diagnosis with FDG PET imaging: physiologic and benign variants. Radiographics 1999, 19:61-77.
    • (1999) Radiographics , vol.19 , pp. 61-77
    • Shreve, P.D.1    Anzai, Y.2    Wabl, R.L.3
  • 2
    • 0033625413 scopus 로고    scopus 로고
    • O-(2-[18F]Fluoroethyl)-l-tyrosine and l-[methyl-11C]methionine uptake in brain tumours: initial results of a comparative study
    • Weber W.A., Wester H.J., Grosu A.L., Herz M., Dzewas B., Fedlmann H.J., et al. O-(2-[18F]Fluoroethyl)-l-tyrosine and l-[methyl-11C]methionine uptake in brain tumours: initial results of a comparative study. Eur J Nucl Med 2000, 27:542-549.
    • (2000) Eur J Nucl Med , vol.27 , pp. 542-549
    • Weber, W.A.1    Wester, H.J.2    Grosu, A.L.3    Herz, M.4    Dzewas, B.5    Fedlmann, H.J.6
  • 4
    • 0032869487 scopus 로고    scopus 로고
    • Investigation of transport mechanism and uptake kinetics of O-(2-[18F]fluoroethyl)-l-tyrosine in vitro and in vivo
    • Heiss P., Mayer S., Herz M., Wester H.J., Schwaiger M., Senekowitsch-Schmidtke R. Investigation of transport mechanism and uptake kinetics of O-(2-[18F]fluoroethyl)-l-tyrosine in vitro and in vivo. J Nucl Med 1999, 40:1367-1373.
    • (1999) J Nucl Med , vol.40 , pp. 1367-1373
    • Heiss, P.1    Mayer, S.2    Herz, M.3    Wester, H.J.4    Schwaiger, M.5    Senekowitsch-Schmidtke, R.6
  • 6
    • 0036888494 scopus 로고    scopus 로고
    • Efficient routine production of the 18F-labelled amino acid O-(2-[18F]fluoroethyl)-l-tyrosine
    • Hamacher K., Coenen H.H. Efficient routine production of the 18F-labelled amino acid O-(2-[18F]fluoroethyl)-l-tyrosine. Appl Radiat Isot 2002, 57:853-856.
    • (2002) Appl Radiat Isot , vol.57 , pp. 853-856
    • Hamacher, K.1    Coenen, H.H.2
  • 7
    • 73949106339 scopus 로고    scopus 로고
    • New approach for the synthesis of [18F]fluoroethyltyrosine for cancer imaging: simple, fast, and high yielding automated synthesis
    • Zuhayra M., Alfteimi A., Von Forstner C., Lützen U., Meller B., Henze E. New approach for the synthesis of [18F]fluoroethyltyrosine for cancer imaging: simple, fast, and high yielding automated synthesis. Bioorg Med Chem 2009, 17:7441-7448.
    • (2009) Bioorg Med Chem , vol.17 , pp. 7441-7448
    • Zuhayra, M.1    Alfteimi, A.2    Von Forstner, C.3    Lützen, U.4    Meller, B.5    Henze, E.6
  • 8
    • 33746790640 scopus 로고    scopus 로고
    • Remote-controlled module-assisted synthesis of O-(2-[18F]fluoroethyl)-l-tyrosine as tumor PET tracer using two different radiochemical routes
    • Wang M.W., Yin D.Z., Zhang L., Zhou W., Wang Y.X. Remote-controlled module-assisted synthesis of O-(2-[18F]fluoroethyl)-l-tyrosine as tumor PET tracer using two different radiochemical routes. Nucl Sci Tech 2006, 17:148-153.
    • (2006) Nucl Sci Tech , vol.17 , pp. 148-153
    • Wang, M.W.1    Yin, D.Z.2    Zhang, L.3    Zhou, W.4    Wang, Y.X.5
  • 9
    • 33750170963 scopus 로고    scopus 로고
    • Preparation of 18F labelled amino acid O-(2-[18F]fluoroethyl)-l-tyrosine using indirect and direct labelling methods
    • Wang M.W., Yin D.Z., Cheng D.F., Li G., Wang Y.X. Preparation of 18F labelled amino acid O-(2-[18F]fluoroethyl)-l-tyrosine using indirect and direct labelling methods. J Radioanal Nucl Chem 2006, 270:439-443.
    • (2006) J Radioanal Nucl Chem , vol.270 , pp. 439-443
    • Wang, M.W.1    Yin, D.Z.2    Cheng, D.F.3    Li, G.4    Wang, Y.X.5
  • 10
    • 0037161591 scopus 로고    scopus 로고
    • Radiolabeled amino acids for tumor imaging with PET: radiosynthesis and biological evaluation of 2-amino-3-[18F]fluoro-2-methylpropanoic acid and 3-[18F]fluoro-2-methyl-2-(methylamino)propanoic acid
    • McConathy J., Martarello L., Malveaux E.J., Camp V.M., Simpson N.E., Simpson C.P., et al. Radiolabeled amino acids for tumor imaging with PET: radiosynthesis and biological evaluation of 2-amino-3-[18F]fluoro-2-methylpropanoic acid and 3-[18F]fluoro-2-methyl-2-(methylamino)propanoic acid. J Med Chem 2002, 45:2240-2249.
    • (2002) J Med Chem , vol.45 , pp. 2240-2249
    • McConathy, J.1    Martarello, L.2    Malveaux, E.J.3    Camp, V.M.4    Simpson, N.E.5    Simpson, C.P.6
  • 11
    • 12444328823 scopus 로고    scopus 로고
    • Synthesis and evaluation of 2-amino-4-[18F]fluoro-2-methylbutanoic acid (FAMB): relationship of amino acid transport to tumour imaging properties of branched fluorinated amino acids
    • McConathy J., Martarello L., Malveaux E.J., Camp V.M., Simpson N.E., Simpson C.P., et al. Synthesis and evaluation of 2-amino-4-[18F]fluoro-2-methylbutanoic acid (FAMB): relationship of amino acid transport to tumour imaging properties of branched fluorinated amino acids. Nucl Med Biol 2003, 30:477-490.
    • (2003) Nucl Med Biol , vol.30 , pp. 477-490
    • McConathy, J.1    Martarello, L.2    Malveaux, E.J.3    Camp, V.M.4    Simpson, N.E.5    Simpson, C.P.6
  • 12
    • 18844392093 scopus 로고    scopus 로고
    • Evaluation of F-18-labeled amino acid derivatives and [18F]FDG as PET probes in a brain tumor-bearing animal model
    • Wang H.E., Wu S.Y., Chang C.W., Liu R.S., Hwang L.C., Lee T.W., et al. Evaluation of F-18-labeled amino acid derivatives and [18F]FDG as PET probes in a brain tumor-bearing animal model. Nucl Med Biol 2005, 32:367-375.
    • (2005) Nucl Med Biol , vol.32 , pp. 367-375
    • Wang, H.E.1    Wu, S.Y.2    Chang, C.W.3    Liu, R.S.4    Hwang, L.C.5    Lee, T.W.6
  • 13
    • 79959638403 scopus 로고    scopus 로고
    • Radioactively labelled amino acid analogues, their preparation and use. Patent No. WO 2004/110500A1
    • Mertens JJR. Radioactively labelled amino acid analogues, their preparation and use. Patent No. WO 2004/110500A1.
    • Mertens, J.J.R.1
  • 14
    • 33747034214 scopus 로고    scopus 로고
    • Evaluation of d-isomers of O-18F-fluoromethyl, O-18F-fluoroethyl and O-18F-fluoropropyl tyrosine as tumour imaging agents in mice
    • Tsukada H., Sato K., Fukumoto D., Kakiuchi T. Evaluation of d-isomers of O-18F-fluoromethyl, O-18F-fluoroethyl and O-18F-fluoropropyl tyrosine as tumour imaging agents in mice. Eur J Nucl Med Mol Imaging 2006, 33:1017-1024.
    • (2006) Eur J Nucl Med Mol Imaging , vol.33 , pp. 1017-1024
    • Tsukada, H.1    Sato, K.2    Fukumoto, D.3    Kakiuchi, T.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.