Synthesis of hexahydro[2]benzopyrano[3,4-c]pyrroles as serotonin 5-HT 2C receptor agonists via intramolecular hetero Diels-Alder reactions

Tetrahedron Letters

Volumn 52, Issue 27, 2011, Pages 3413-3416

  Kiyoi, Takao ^a   Reid, Mark ^a   Francis, Stuart ^a   Davies, Keneth ^a   Laats, Steven ^a   McArthur, Duncan ^a   Easson, Anna Marie ^a   Kiyoi, Yasuko ^a   Tarver, Gary ^a   Caulfield, Wilson ^a   Gibson, Kirsty ^a   Wishart, Grant ^a   Morrison, Angus J ^a   Adam, Julia M ^a   Ray, Peter ^a  

^a MERCK RESEARCH LABORATORIES   (United States)

Author keywords

2 Benzopyrano 3,4 c pyrroles; Intramolecular hetero Diels Alder reaction; Microwave assisted synthesis; Serotonin 5 HT2C receptor agonists

Indexed keywords

BENZOPYRAN DERIVATIVE; HEXAHYDRO[2]BENZOPYRANO[3,4 C]PYRROLE DERIVATIVE; PYRROLE DERIVATIVE; SEROTONIN 2C AGONIST; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL ANALYSIS; DIELS ALDER REACTION; DRUG STRUCTURE; DRUG SYNTHESIS;

ALNUS;

EID: 79957959760     PISSN: 00404039     EISSN: 18733581     Source Type: Journal    
DOI: 10.1016/j.tetlet.2011.03.055     Document Type: Article

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