An efficient synthesis of pyrrolo[1,2-a]quinazolin-5(1H)-one derivatives with the aid of low-valent titanium reagent

Journal of Heterocyclic Chemistry

Volumn 48, Issue 3, 2011, Pages 634-638

  Zhao, Xuan ^a   Shi, Da Qing ^a  

^a SOOCHOW UNIVERSITY   (China)

Author keywords

[No Author keywords available]

Indexed keywords

2,3,3A,4 TETRAHYDROPYRROLO[1,2 A]QUINAZOLIN 5(1H) ONE; 2,3,3A,4 TETRAHYDROPYRROLO[1,2 A]QUINAZOLINE 1,5 DIONE; HALOKETONE; LEVULINIC ACID; QUINAZOLINE DERIVATIVE; TITANIUM; UNCLASSIFIED DRUG;

ARTICLE; CYCLIZATION; SYNTHESIS;

EID: 79957460688     PISSN: 0022152X     EISSN: 19435193     Source Type: Journal    
DOI: 10.1002/jhet.637     Document Type: Article

References (26)

1. Connolly, D. J.; Cusack, D.; O'sullivan, T. P.; Guiry, P. J., Tetrahedron 2005, 61, 10153.
2. Hassanein, H. H.; Abdel, N. G., Bull Fac Pharm 1995, 33, 29.
3. Bekhit, A. A.; Habib, N. S., Et-Din, A.; Bekhit, A., Boll Chim Farm 2001, 140, 297.
4. Malllard, J.; Vincent, M.; Bernard, M., Chim Ther 1968, 3, 100.
5. Merck. Merck Index; Merck: Whithouse Station, NJ, 1996, Vol. 12, p 7897.
6. Merck. Merck Index; Merck: Whithouse Station, NJ, 1996, Vol. 12, p 1512.
7. Merck. Merck Index; Merck: Whithouse Station, NJ, 1996, Vol. 12, p 3489.
8. Stephen, H.; Wedge G., J Chem Soc 1956, 4420.
9. Takeuchi, H.; Hagiwara S.; Eguchi, S., Tetrahedron 1989, 45, 6375.
10. Ferraccioli, R.; Carenzi, D., Synthesis 2003, 1383.
11. Schlapbach, A,;, Heng, R.; Di Padova, F., Bioorg Med Chem Lett 2004, 14, 357.
12. Pastor, G,;, Blanchard, C.; Montginoul, C.; Torreilles, E.; Giral, L.; Texier, A., Bull Soc Chim Fr 1975, 1331.
13. Khalifa, M.; Osman, A. N.; Ibrahim, M. G.; Ossman, A. R. E.; Ismail, M. A., Pharmaizie 1982, 37, 115.
14. Michman, M.; Patai, S.; Wiesel, Y., Org Prep Proced Int 1978, 10, 13.
15. Vorbrueggen, H.; Krolikiewicz, K., Tetrahedron 1994, 50, 6549.
16. Mizuno, T.; Iahino, Y., Tetrahedron 2002, 58, 3155.
17. Tatsuya, O.; Eiji, N.; Takashi, T.; Shingo, M., Tetrahedron 2003, 59, 5603.
18. Aeberli, P.; Houlihan, W. J., J Org Chem 1968, 33, 2402.
19. Iminov, R. T.; Tverdokhlebov, A. V.; Tolmachev, A. A.; Volovenko, Y. M.; Shishkina, S. V.; Shishkin, O. V., Tetrahedron 2009, 65, 8582.
20. Iminov, R. T.; Tverdokhlebov, A. V.; Tolmachev, A. A.; Volovenko, Y. M.; Kostyuk, A. N.; Chernega, A. N.; Rusanov, E. B., Heterocycles 2008, 75, 1673.
21. Shi, D. Q.; Rong, L. C.; Wang, J. X.; Zhuang, Q. Y.; Wang, X. S.; Hu, H. W., Tetrahedron Lett 2003, 44, 3199.
22. Shi, D. Q.; Dou, G. L.; Li, Z. Y.; Ni, S. N.; Li, X. Y.; Wang, X. S.; Wu, H.; Ji, S. J., Tetrahedron 2007, 63, 9764.
23. Shi, D. Q.; Wang, J. X.; Shi, C. L.; Rong, L. C.; Zhuang, Q. Y.; Hu, H. W., Synlett 2004, 1098.
24. Dou, G. L.; Wang, M. M.; Shi, D. Q., J Comb Chem 2009, 11, 151.
25. Houlihan, W. J.; Mountain Lakes, N. J.; Sandoz, Inc., Hanover, N. J. US Patent 1964, 447,566;
26. Chem Abstr 1969, 71, 70630v.