Novel jojoba oil-based emulsion gel formulations for clotrimazole delivery

AAPS PharmSciTech

Volumn 12, Issue 1, 2011, Pages 239-247

  Shahin, Mostafa ^a   Abdel Hady, Seham ^b   Hammad, Mohammed ^c   Mortada, Nahed ^a  

^a AIN SHAMS UNIVERSITY   (Egypt)

^b KING ABDULAZIZ UNIVERSITY   (Saudi Arabia)

^c Zagazig University   (Egypt)

Author keywords

Carbopol 934 P; clotrimazole; emulgel; emulsion gel; HPMC; microbiological evaluation; rheology; stability

Indexed keywords

CANDISTAN; CARBOPOL 934; CLOTRIMAZOLE; GELLING AGENT; HYDROXYPROPYLMETHYLCELLULOSE; JOJOBA OIL; LONG CHAIN FATTY ACID; UNCLASSIFIED DRUG;

ANTIFUNGAL ACTIVITY; ARTICLE; CANDIDA ALBICANS; CONTROLLED STUDY; CREAM; DRUG DELIVERY SYSTEM; DRUG EFFICACY; DRUG FORMULATION; DRUG RELEASE; DRUG STABILITY; DRUG STORAGE; EMULGEL FORMULATION; EMULSION; IN VITRO STUDY; NONHUMAN; PRIORITY JOURNAL; ROOM TEMPERATURE; SHEAR STRESS; THIXOTROPY;

ACRYLATES; ADMINISTRATION, TOPICAL; ANTIFUNGAL AGENTS; CANDIDA ALBICANS; CLOTRIMAZOLE; DOSAGE FORMS; DRUG DELIVERY SYSTEMS; DRUG STABILITY; EMULSIONS; EXCIPIENTS; GELS; HUMANS; METHYLCELLULOSE; VISCOSITY; WAXES;

EID: 79954423348     PISSN: None     EISSN: 15309932     Source Type: Journal    
DOI: 10.1208/s12249-011-9583-4     Document Type: Article

References (35)

1. D Marquardt H Sucker 1998 Oil in water emulsion gels: determination and mathematical treatment of flow properties Eur J Pharm Biopharm 46 115 24 9700029 10.1016/S0939-6411(97)00167-7 1:CAS:528:DyaK1cXnsFKhu7w%3D (Pubitemid 29168542)
2. Martindale. The Extra Pharmacopiea. 29 ed. London: Pharmaceutical; 1989
3. D Tettenborn 1972 Acute toxicity and local tolerance of clotrimazole Drugs Made Ger 15 9 94 9 1:CAS:528:DyaE2MXisV0%3D
4. A Bonifaz A Saul 2000 Comparative study between terbinafine 1% emulsion-gel versus ketoconazole 2% cream in tinea cruris and tinea corporis Eur J Dermatol 10 2 107 9 10694308 1:CAS:528:DC%2BD3cXhvFamsbw%3D (Pubitemid 30116422)
5. Borlaug N, Baldwin AR, Estefan R, Harris M, Plucknett DL. Jojoba: new crop for arid lands. New raw material for industry. Washington DC: National Academy Press; 1985.
6. R Habashy A Abdel-Naim A Khalifa M Al-Azizi 2005 Anti-inflammatory effects of jojoba liquid wax in experimental models Pharmacol Res 51 2 95 105 15629254 10.1016/j.phrs.2004.04.011 (Pubitemid 40040539)
7. P Mura MT Faucci P Corti G Bramanti 1997 Formulation studies on topical preparations of clonazepam STP Pharm Sci 7 3 229 34 1:CAS:528:DyaK2sXmtFaksr4%3D
8. MM Jimenez Soriano MJ Fresno Contreras E Selles Flores 2001 Development of a cream from a self emulsifying base and moisturizing actives IL Farmaco 56 513 22 11482788 10.1016/S0014-827X(01)01087-4 1:CAS:528:DC%2BD3MXkvVertLk%3D (Pubitemid 32622127)
9. E Bourret V Ratsimbazafy L Maury C Brossard 1994 Rheological behavior of saturated polyglycolysed glycerides J Pharm Pharmacol 46 538 41 7996378 1:CAS:528:DyaK2cXlvVOhtLo%3D (Pubitemid 24213276)
10. S Simovic J Milic-ASkrabic G Vuleta M Stupar 1998 Physicochemical properties of emulsion gels with different concentrations of polymeric emulsifier pemulen TR1-NF Pharmazie 53 4 276 7 1:CAS:528:DyaK1cXitl2quro%3D (Pubitemid 28186833)
11. D Marquardt P Pedrussio B Herzog H Sucker 1997 Determination of (pseudo)plastic flow properties of pharmaceutical semisolids using rheological AUC parameters Drug Dev Tech 2 2 123 33 1:CAS:528:DyaK2sXjvVygsbw%3D (Pubitemid 28252528)
12. D Krajisink J Milic 2003 Polymer stabilized emulsion systems: structure characteristics and physical stability evaluation Drug Dev Ind Pharm 29 701 11 10.1081/DDC-120021319 (Pubitemid 36840847)
13. N Grigelmo-Miguel O Martin-Belloso 1999 Influence of fruit dietary fiber addition on physical and sensorial properties of strawberry jams J Food Eng 41 13 21 10.1016/S0260-8774(99)00067-9
14. SA Ibrahim E Hafez SM El-shenawy IS El-Gibally EA Mohamed 1991 Formulation and evaluation of clotrimazole ointment Bull Pharm Sci Assi Univ 14 1&2 13 22 1:CAS:528:DyaK38Xmtl2mu7s%3D
15. Harry RG, Harry RG, Rieger MM. Harry's cosmeticology. New York: Chemical Publishing; 2000.
16. Langer RS, Wise DS. Medical applications of controlled release. FL: CRC; 1984.
17. MJ Lucero J Vigo MJ Leon 1994 Study of shear and compression deformations on hydrophilic gels of tretinoin Int J Pharm 106 5 125 33 10.1016/0378-5173(94) 90310-7 1:CAS:528:DyaK2cXktFOrtLw%3D (Pubitemid 24136530)
18. A Abdel-Bary S Shalaby S Abdel-Aal 2001 Formulation and stability of chloramphenicol gel and emulgel Bull Fac Pharm Cairo Univ 39 3 89 99 1:CAS:528:DC%2BD38Xmsl2itLw%3D
19. LW Chan TW Wong PC Chua P York PW Heng 2003 Anti-tack action of polyvinylpyrrolidone on hydroxypropyl methylcellulose solution Chem Pharm Bull 51 2 107 12 12576641 10.1248/cpb.51.107 1:CAS:528:DC%2BD3sXjsFCqu7o%3D (Pubitemid 41701978)
20. B Kovacs G Merenyi 1990 Evaluation of tack behavior of coating solutions Drug Dev Ind Pharm 16 15 2320 3 10.3109/03639049009043801
21. S Rossi F Ferrari MC Bonferoni C Caramella 2001 Rheological and mechanical properties of pharmaceutical gels. Part II: medicated systems: relevance to hydration properties and drug release Boll Chim Farm 140 337 44 11680088 1:CAS:528:DC%2BD3MXot1Crsb8%3D (Pubitemid 32945915)
22. Briceno MI. Rheology of suspensions and emulsions. In: Nelloud F, Marti-Mestres N, editors. Pharmaceutical emulsions and suspensions. New York: Marcel Dekker; 2000. p. 577-607.
23. Perrot EL. Pharmaceutical technology, fundamental pharmaceutics. Minneapolis: Burgress; 1971.
24. LE Pena BI Lee JF Sternes 1994 Structural rheology of model ointment Pharm Res 11 875 81 7937529 10.1023/A:1018990010686 1:CAS:528:DyaK2cXksValsL8%3D (Pubitemid 24210625)
25. MJC Fresno AD Ramirez MM Jimenez 2002 Systematic study of the flow behavior and mechanical properties of carbopol Ultrez 10 hydroalcoholic gels Eur J Pharm Biopharm 54 329 35 12445564 10.1016/S0939-6411(02)00080-2 1:CAS:528:DC%2BD38XoslGguro%3D (Pubitemid 35341834)
26. R Huttenrauch S Fricke 1976 Molecular galenics. 7. Mechanical activation of salves, an indirect proof of their quaternary structure Pharmazie 31 6 408 9 959306 1:STN:280:DyaE283mvFymsQ%3D%3D
27. R Huttenrauch S Fricke V Baumann 1982 Properties and dynamics of structure in shear crystallized ointments Pharmazie. 37 1 25 8 7071108 1:STN:280:DyaL387nsVyjtA%3D%3D
28. E Dickinson SJ Rodford M Golding 2003 Stability and rheology of emulsions containing sodium caseinate: combined effects of ionic calcium and non ionic surfactant Food Hydrocoll 17 211 20 10.1016/S0268-005X(02)00055-3 1:CAS:528:DC%2BD3sXht1Wlsb0%3D
29. P Walkenstrom AM Hermansson 1998 Effect of shear on pure and mixed gels of gelatin and particulate whey protein Food Hydrocoll 12 77 87 10.1016/S0268-005X(98)00048-4 1:CAS:528:DyaK1cXktlyqs7w%3D (Pubitemid 128154435)
30. Jiao J, Burgess DJ. Rheology and stability of w/o/w multiple emulsions containing span 83 and Tween 80. AAPS Pharm Sci Tech. 2003;5(1)
31. P Mura C Nassini D Proietti A Manderioli 1996 Influence of vehicle composition variation on the in vitro and ex vivo clonazepam diffusion from hydrophilic ointment bases Pharm Acta Helv 71 147 54 8810581 10.1016/0031-6865(96)00005-2 (Pubitemid 26281325)
32. A Arellano S Santoyo C Martin P Ygartua 1999 Influence of propylene glycol and isopropyl myristate on the in vitro percutaneous penetration of diclofenac sodium from carbopol gels Eur J Pharm Sci 7 129 35 9845796 10.1016/S0928-0987(98)00010-4 1:CAS:528:DyaK1cXnvVSrsbY%3D (Pubitemid 29056235)
33. Davis SS. Symposium on topical administration of drugs. 1989.
34. JM Petit B Roux XX Zhu 1996 A new physical model for the diffusion of solvents and solutes probes in polymer solutions Macromolecules 29 6031 6 10.1021/ma951159c 1:CAS:528:DyaK28Xks12ktb4%3D (Pubitemid 126520488)
35. SS Davis MS Khanderia 1972 Viscoelastic properties of pharmaceutical semisolids: characterization of the plastibase for bioavailability studies J Pharm Pharmacol 24 176 7 4401981