Selective α-glucosidase substrates and inhibitors containing short aromatic peptidyl moieties

Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 8, 2011, Pages 2441-2444

  Park, Sangeun ^a   Hyun, Soonsil ^a   Yu, Jaehoon ^a  

^a Seoul National University   (South Korea)

Author keywords

Glucosidase inhibitor; Glucoside dipeptidyl conjugate; Chromogenic assay; Substrate library

Indexed keywords

4 ACETAMINOPHENYL ALPHA DEXTRO GLUCOPYRANOSIDE; 4 NITROPHENOL; ALPHA GLUCOSIDASE; ALPHA GLUCOSIDASE INHIBITOR; AMYLASE; AROMATIC AMINO ACID; AROMATIC COMPOUND; BACTERIAL ENZYME; BETA GLUCOSE SPACER TRYPTOPHYLTYROSINE; CARBOHYDRATE DERIVATIVE; CHROMOGENIC SUBSTRATE; GLUCOPYRANOSIDE; GLUCOSE DERIVATIVE; PEPTIDE DERIVATIVE; PEPTIDE LIBRARY; SPACER TRYPTOPHYLTYROSINE; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; COMPETITIVE INHIBITION; DRUG DESIGN; DRUG PROTEIN BINDING; DRUG SCREENING; DRUG SELECTIVITY; DRUG SYNTHESIS; ENZYME SUBSTRATE; GEOBACILLUS STEAROTHERMOPHILUS; NONHUMAN; STRUCTURE ACTIVITY RELATION;

ALPHA-GLUCOSIDASES; ANIMALS; BACILLUS; ENZYME INHIBITORS; HYDROPHOBIC AND HYDROPHILIC INTERACTIONS; ORYZA SATIVA; PEPTIDES; RATS; SUBSTRATE SPECIFICITY;

EID: 79953282779     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2011.02.062     Document Type: Article

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