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Bioorganic Chemistry

Volumn 39, Issue 2, 2011, Pages 67-72

Application of the bridgehead fragments for the design of conformationally restricted melatonin analogues

(5) Zefirova, Olga N a,b Baranova, Tatiana Yu a Ivanova, Anna A b Ivanov, Andrei A c Zefirov, Nikolay S a,b

a MOSCOW STATE UNIVERSITY (Russian Federation)

b INSTITUTE OF PHYSIOLOGICALLY ACTIVE COMPOUNDS (Russian Federation)

c EMORY UNIVERSITY SCHOOL OF MEDICINE (United States)

Author keywords

Bridgehead fragments; Conformational restriction; Melatonin receptors

Indexed keywords

2 METHOXY 6,7,8,9,10,11 HEXAHYDRO 5H 6,10 METHANOCYCLOOCTA[B]INDOL 9 AMINE; BICARBONATE; BICYCLO[2.2.2]OCTANE DERIVATIVE; BICYCLO[3.2.1]OCTANE DERIVATIVE; BICYCLO[3.3.1]NONANE DERIVATIVE; INDOLE DERIVATIVE; MELATONIN; MELATONIN 1 RECEPTOR; MELATONIN 2 RECEPTOR; MELATONIN DERIVATIVE; MELATONIN RECEPTOR; METHYL 6 METHOXY 2,3,4,9 TETRAHYDRO 1H 1,4 ETHANOCARBAZOLE 3 CARBOXYLATE; METHYL ENDO 2 METHOXY 5,6,7,8,9,10 HEXAHYDRO 6,9 METHANOCYCLOHEPTA[B]INDOL 8 CARBOXYLATE; N (2 METHOXY 5,6,7,8,9,10 HEXAHYDRO 6,9 METANOCYCLOHEPTA[B]INDOL 8 YL)ACETAMIDE; N (ENDO 2 METHOXY 6,7,8,9,10,11 HEXAHYDRO 5H 6,10 METANOCYCLOOCTA[B]INDOL 9 YL)ACETAMIDE; N (EXO 6 METHOXY 2,3,4,9 TETRAHYDRO 1H 1,4 ETHANOCARBAZOL 3 YL)ACETAMIDE; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; CHEMICAL MODIFICATION; CRYSTAL STRUCTURE; DRUG DESIGN; ENZYME SYNTHESIS; MOLECULAR DOCKING; PRIORITY JOURNAL; RECEPTOR BINDING;

BICYCLO COMPOUNDS; COMPUTER SIMULATION; INDOLES; MELATONIN; MOLECULAR CONFORMATION; RECEPTOR, MELATONIN, MT1; RECEPTOR, MELATONIN, MT2;

EID: 79953221772 PISSN: 00452068 EISSN: 10902120 Source Type: Journal
DOI: 10.1016/j.bioorg.2011.02.002 Document Type: Article

Times cited : (15)

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