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Volumn 19, Issue 7, 2011, Pages 2359-2367

Acetyl analogs of combretastatin A-4: Synthesis and biological studies

(19) Lee, Moses a Babu, Balaji a Lee, Megan a Lee, Lauren a Strobel, Raymond a Brockway, Olivia a Nickols, Alexis a Sjoholm, Robert a Tzou, Samuel a Chavda, Sameer a Desta, Dereje a Fraley, Gregory a Siegfried, Adam b Pennington, William b Hartley, Rachel M c Westbrook, Cara c Mooberry, Susan L c Kiakos, Konstantinos d Hartley, John A d

a HOPE COLLEGE (United States)

b CLEMSON UNIVERSITY (United States)

c University of Texas Health Science Center at San Antonio (United States)

d UNIVERSITY COLLEGE LONDON (United Kingdom)

Author keywords

Cancer; Combretastatin A 4; Cytotoxicity; Microtubule; Trimethoxyphenylacetone; Tubulin

Indexed keywords

A 105972; AC 7739; ACETYLCOMBRETASTATIN DERIVATIVE; ALDEHYDE DERIVATIVE; ANTINEOPLASTIC AGENT; COMBRETASTATIN A4; OMBRABULIN; OXADIAZOLINE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL MODEL; ANTINEOPLASTIC ACTIVITY; ARTICLE; CANCER INHIBITION; CANCER MODEL; CELL STRAIN; CELL STRAIN MDA MB 435; CONTROLLED STUDY; DEPOLYMERIZATION; DRUG CYTOTOXICITY; DRUG POTENCY; DRUG SOLUBILITY; DRUG STRUCTURE; DRUG SYNTHESIS; FEMALE; GENETIC MODEL; HUMAN; HUMAN CELL; IC 50; MOLECULAR MODEL; MOUSE; NONHUMAN;

ANIMALS; CRYSTALLOGRAPHY, X-RAY; FEMALE; HUMANS; LEUKEMIA L1210; MELANOMA, EXPERIMENTAL; MICE; MICE, INBRED DBA; MICROTUBULES; MOLECULAR CONFORMATION; STILBENES; STRUCTURE-ACTIVITY RELATIONSHIP;

MURINAE;

EID: 79953200442 PISSN: 09680896 EISSN: None Source Type: Journal
DOI: 10.1016/j.bmc.2011.02.018 Document Type: Article

Times cited : (16)

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