Conventional as well as microwave assisted synthesis of some new 4-aryl-3-chloro-1-[(isonicotinamid-4-yl)acetamido]-2-oxo-azetidines: Antibacterial and antifungal agents

Proceedings of the National Academy of Sciences India Section A - Physical Sciences

Volumn 80, Issue 2, 2010, Pages 131-138

  Upadhyay, Apoorva ^a   Srivastava, S K ^a   Srivastava, S D ^a   Yadav, R ^a  

^a DR H S GOUR UNIVERSITY   (India)

Author keywords

Arylidene; Conventional and microwave synthesis; Empirical validation; Evaluation criteria; Isonicotinamide; Thiazolidinone

Indexed keywords

EID: 79953128070     PISSN: 03698203     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Conference Paper

References (19)

1. Caddick S. Microwave assisted organic reactions. Tetrahedron 1995;51:10403-10432.
2. Perreux L & Loupy A. A tentative rationalization of microwave effects in organic synthesis according to the reaction medium and mechanistic consideration. Tetrahedron 2001;57:9199-9223. (Pubitemid 33019218)
3. Galema SA. Microwave chemistry. Chem Soc Rev 1997; 26:233-238. (Pubitemid 127097205)
4. Lidstrom P, Tierney J, Wathey B & Westman J. Microwave assisted organic synthesis a review. Tetrahedron 2001 ; 57 : 9225-9283. (Pubitemid 33016768)
5. Katritzky AR & Singh SK. Microwave assisted heterocyclic synthesis. Arkivoc 2003; 13 : 68-86.
6. Patel VM & Desai KR. Eco-friendly synthesis of pyrazoline derivatives over potassium carbonate. Arkivoc 2004; 1: 123-129. (Pubitemid 38783192)
7. Desai AR & Desai KR. Niementowski reaction: microwave induced and conventional synthesis of quinazolinone and 3-methyl-1H-5-pyrazolone and their antimicrobial activity. Arkivoc 2005; 13: 98-108. (Pubitemid 40757042)
8. Kennedy AD & Summers AL. Chemical constitution and activity of bipyridinium herbicides. Part XIV. Reduction potential and herbicidal activity of 4,4′-(1 ,3,4-Thiadiazole-2,5-diyl) and 4,4′-(1,3,4-oxadiazole-2, 5-diyl) bis(1-methylpyridinium) diiodides. J Heterocyclic Chem 1981 ; 18:409-410.
9. Holla BS, Prasanna CS, Poojary B, Rao KS, Shridhara K & Bhat UG Synthesis and insecticidal activity of some 1,3,4-oxadiazoles derived from 2-chloropyridine-5-acetic acid. Indian J Chem 2004; 43B : 864-868.
10. Kshirsagar A, Turaskar MP, Kulkami VM, Dhanashire S & Kadam V. Microwave assisted synthesis of potential antiinfective and anticonvulsant thiosemicarbazones. International J of chem Tech Research 2009; 1 : 696-701.
11. Arikan N, Sumengen D & Dulger B. Synthesis and antimicrobial activities of 1,2,4-Oxadiazin-5-one, 6-one and 5-thiones. Turk J Chem 2008; 32 : 147-155.
12. Sharma R, Nagda DP & Talesara GL. Synthesis of various isoniazidothiazolidinones and their imidoxy derivatives of potential biological interest. Arkivoc 2006; 1 : 1-12.
13. Sonwane SK, Srivastava SD & Srivastava SK. Synthesis and antimicrobial activity of 2-(2′-arylidene-hydrazino-acetylamino)-4-phenyl- 1,3-thiazoles and 2-[2′-{4″-substituted-aryl-3″-chloro- 2″-oxo-azetidine}-acetyl-amino]-4-phenyl-1,3-thiazoles. Indian J Chem 2008; 47B : 633-636.
14. Singh GS & Pheko T. Formation and antimicrobial activity of 2-azetidinones from selective ester cleavage in 1,3,3-trisubstituted-4- [2′-(O-diarylacyl) hydroxyphenyl]-2-azetidinones. Indian J Chem 2008; 47B : 159-162.
15. Yadav R, Srivastava S, Srivastava SK & Srivastava SD. Synthesis and biological activity of benzothiazolylthiomethyl-1,3,4-thiadiazol-2-oxo- azetidines and 5-arylidene-1,3-thiazolidine-4-ones. Chemistry: An Indian J 2003; 1 : 95-103.
16. Mistry K & Desai KR. Microwave assisted rapid and efficient synthesis of nitrogen and sulphur containing heterocyclic compounds and their pharmacological evaluation. Indian J Chem 2006; 45B : 1762-1766. (Pubitemid 44320361)
17. Kohli P, Srivastava SD & Srivastava SK. Synthesis and pharmacological evaluation of (N-phenothiazinomethyl)-4-[N-(3-chloro-2-oxo-4-substituted- azetidin)]-5-mercapto1,2,4-triazoles. J Ind Chem Soc 2008; 85 : 326-327.
18. Kumar A & Rajput CS. Synthesis and anti-inflammatory activity of newer quinazolin-4-one derivatives. Eur J Med Chem 2009; 44 : 83-90.
19. Srivastava SK, Srivastava S & Srivastava SD. Synthesis of new carbazolyl-thiadiazol-2-oxo-azetidines: antimicrobial, anticonvulsant and anti-inflammatory agents. Indian J Chem 1999; 38B: 183-187.