Niementowski reaction: Microwave induced and conventional synthesis of quinazolinones and 3-methyl-1H-5-pyrazolones and their antimicrobial activity

Arkivoc

Volumn 2005, Issue 13, 2005, Pages 98-108

  Desai, Amar R ^a   Desai, Kishor R ^a  

^a VEER NARMAD SOUTH GUJARAT UNIVERSITY   (India)

Author keywords

Microwave; Niementowski reaction; Pyrazolone; Quinazolinone

Indexed keywords

2 METHYL 3 [2 [(3 METHYL 5 OXO 4,5 DIHYDRO 1H PYRAZOL 1 YL) 2 OXOETHYL]]QUINAZOLIN 4(3H) ONE; 2 METHYL 3 [3 [(3 METHYL 5 OXO 4,5 DIHYDRO 1H PYRAZOL 1 YL)CARBONYL]PHENYL]QUINAZOLIN 4(3H) ONE; 2 METHYL 3 [4 [(3 METHYL 5 OXO 4,5 DIHYDRO 1H PYRAZOL 1 YL)CARBONYL]PHENYL]QUINAZOLIN 4(3H) ONE; 3 [2 [(3 METHYL 5 OXO 4,5 DIHYDRO 1H PYRAZOL 1 YL) 2 OXOETHYL] 2 PHENYL]QUINAZOLIN 4(3H) ONE; 3 [3 [(3 METHYL 5 OXO 4,5 DIHYDRO 1H PYRAZOL 1 YL)CARBONYL]PHENYL]2 PHENYLQUINAZOLIN 4(3H) ONE; 3 [4 [(3 METHYL 5 OXO 4,5 DIHYDRO 1H PYRAZOL 1 YL)CARBONYL]PHENYL] 2 PHENYLQUINAZOLIN 4(3H) ONE; 6 BROMO 2 METHYL 3 [2 [(3 METHYL 5 OXO 4,5 DIHYDRO 1H PYRAZOL 1 YL) 2 OXOETHYL]]QUINAZOLIN 4(3H) ONE; 6 BROMO 2 METHYL 3 [3 [(3 METHYL 5 OXO 4,5 DIHYDRO 1H PYRAZOL 1 YL)CARBONYL]PHENYL]QUINAZOLIN 4(3H) ONE; 6 BROMO 2 METHYL 3 [4 [(3 METHYL 5 OXO 2,5 DIHYDRO 1H PYRAZOL 1 YL)CARBONYL]PHENYL]QUINAZOLIN 4(3H) ONE; 6 BROMO 3 [2 [(3 METHYL 5 OXO 4,5 DIHYDRO 1H PYRAZOL 1 YL) 2 OXOETHYL] 2 PHENYL]QUINAZOLIN 4(3H) ONE; 6 BROMO 3 [3 [(3 METHYL 5 OXO 4,5 DIHYDRO 1H PYRAZOL 1 YL)CARBONYL]PHENYL]2 PHENYLQUINAZOLIN 4(3H) ONE; 6 BROMO 3 [4 [(3 METHYL 5 OXO 4,5 DIHYDRO 1H PYRAZOL 1 YL)CARBONYL]PHENYL] 2 PHENYLQUINAZOLIN 4(3H) ONE; AMOXICILLIN; AMPICILLIN; HYDRAZIDE DERIVATIVE; PENICILLIN G; PYRAZOLONE DERIVATIVE; QUINAZOLINONE DERIVATIVE; UNCLASSIFIED DRUG;

ANTIFUNGAL ACTIVITY; ANTIMICROBIAL ACTIVITY; ARTICLE; CANDIDA ALBICANS; CHEMICAL REACTION; COMPARATIVE STUDY; DRUG SCREENING; DRUG SYNTHESIS; GRAM NEGATIVE BACTERIUM; GRAM POSITIVE BACTERIUM; IRRADIATION; MICROWAVE IRRADIATION; MICROWAVE RADIATION; SOLID; SUBSTITUTION REACTION;

EID: 19944393889     PISSN: 14246376     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (26)

1. Xie, W.; Jin, y.; Wang, P. G. Chemtech 1999, 29, 23.
2. Verma, R. S. Green Chem. 1999, 1, 43.
3. Satsangi, R. K. Indian Drugs 1979, 17, 79.
4. Joshi, V.; Chaudhari, R. P. Indian J. Chem. 1987, 26B, 602.
5. Srivastava, V. K.; Gulati, S. S.; Shanker, K. Indian J. Chem. 1987, 26B, 652.
6. Gupta, D. P.; Ahmad, S.; Kumar, A.; Shanker, K. Indian J. Chem. 1988, 27B, 1060.
7. Sakai, K.; Nahata. H. Jpn. Kokai Tokyo Koho JP 6351, 329; Chem. Abstr. 1988, 109, 86338.
8. Niementowski, V. J. Prakt. Chem. 1895, 51, 564;
9. Beilstein 24, 143.
10. Gan, Y.; Lu, D.; Liu, J.; Tian, M. Zhongguo yaouri Zazhi 2001, 11(2), 85;
11. Chem. Abstr. 2002, 136, 216696.
12. Turan-Zitouni, G.; Sivaci, M.; Kilic, F. S.; Erol, K. Eur. J. Med. Chem. 2001, 36, 685.
13. Elguero, J. Comprehensive Heterocyclic Chemistry. The structure, reaction, synthesis and uses of heterocyclic compounds, K. T. Potts, Ed.; Pergamon Press, 1984, Vol. 5, p 167.
14. (a) Sharma, R. S.; Bahel, S. C. J. Ind. Chem. Soc. 1982, 59, 877.
15. (b) Shiba, S. A.; El-Khamry, A, A.; Shaban, M. E.; Atia, K. S. Indian J. Chem. 1997, 36B, 361
16. (a) Jung, J. C.; Watkins, E. B.; Avery, M.A. Synth. Commun. 2002, 32(24), 3767.
17. (b) Scherowsky, G.; Kunda, B. Tetrahedron Lett. 1972, 3169.
18. (a) Kidwai, M.; Saxena, S.; Mohan, R.; Venkataramanan, R. J. Chem. Soc., Perkin Trans. 2002, 16, 1845.
19. (b) Kidwai, M.; Rastogi, S.; Venkataramanan, R. Bull. Chem. Soc. Jpn., 2003, 76, 203.
20. Barry, A. L. The Antimicrobial Susceptibility Test, Principle and Practices., 1993, 180-193.
21. Kidwai, M.; Venkataramanan, R. Green Chem. 2001, 3, 278.
22. Kidwai, M.; Saxena, S.; Mohan, R,; Venkataramanan, R. J. Chem. Soc., Perkin Trans. 2002, 1, 1845.
23. Leiby, R, W. J. Org. Chem. 1985, 50, 2926-2929.
24. Kidwai, M.; Mohan, R.; Org, Proc. Prep. Int. 2003, 35, 426.
25. Kidwai, M.; Rastogi, S.; Mohan, R.; Ruby. Croatica Chemica Acta. 2003, 76, 365.
26. Kidwai, M.; Mohan, R.; J. Korean. Chem. Soc., 2004, 48, 177.